CAS No.: 244101-02-8
L-798106 Catalog No. CSN20466
Synonyms: CM9;GW671021;L-798,106
L-798106 is a potent and highly selective prostanoid EP3 receptor antagonist (Ki values are 0.3, 916, > 5000 and > 5000 nM at EP3, EP4, EP1 and EP2, respectively), and it can attenuate sulprostone-induced inhibition of EFS-evoked twitch and contractile responses in vivo.
| 规格 | 价格 | 促销价格 | 库存 | 数量 |
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纯度 & 质量文件
批次:
靶点选择性
生物活性
- 描述
- 参考文献
- [1] Li C, Liu X, et al. Tuberin Regulates Prostaglandin Receptor-mediated Viability, via Rheb, in mTORC1-hyperactive Cells. Mol Cancer Res. 2017 Jul 14. pii: molcanres.0077.2017.
- [2] Bassil AK, Borman RA, et al. Activation of prostaglandin EP receptors by lubiprostone in rat and human stomach and colon. Br J Pharmacol. 2008 May;154(1):126-35.
实验方案
- 计算器
- 储存液制备
技术信息
| CAS号 | 244101-02-8 | 储存条件 |
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| 分子式 | C27H22BrNO4S | 运输 | 蓝冰 | |
| 分子量 | 536.44 | 别名 | CM9;GW671021;L-798,106 |
