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CAS No.: 1643913-93-2

(E)-3-(6-aminopyridin-3-yl)-N-((5-(4-(4,4-difluoropiperidine-1-carbonyl)phenyl)-7-(4-fluorophenyl)benzofuran-2-yl)methyl)acrylamide Catalog No. CSN17983

Synonyms: PAK4-IN-1

PAK4-IN-1 is an inhibitor of p21-activated kinases (PAKs), with IC50 of ≤100 nM in MTT assay.

规格 价格 促销价格 库存 数量
纯度 & 质量文件 批次:

靶点选择性

生物活性

  • 描述
  • 临床研究
  • NCT号适应症或疾病临床期招募状态预计完成时间地点
    NCT02702492NHL Solid Tum... more >>ors Collapse <<Phase 1RecruitingNovember 2019United States, Colorado ... more >> University of Colorado Cancer Center Recruiting Aurora, Colorado, United States, 80045 Contact: Stephen Leong, MD       Stephen.Leong@ucdenver.edu    Principal Investigator: Stephen Leong, MD          United States, District of Columbia Georgetown University, Lombardi Comprehensive Cancer Center Recruiting Washington, District of Columbia, United States, 20007 Contact: Michael Pishvaian, MD, PhD       pishvaim@georgetown.edu    Principal Investigator: Michael Pishvaian, MD, PhD          United States, Minnesota Mayo Clinic Rochester Recruiting Rochester, Minnesota, United States, 55905 Contact: Amit Mahipal, MBBS, MPH    507-293-0462    mahipal.amit@mayo.edu    Principal Investigator: Amit Mahipal, MBBS, MPH          United States, New York NYU-Laura & Isaac Perlmutter Cancer Center Recruiting New York, New York, United States, 100016 Contact: Daniel Cho    212-731-5871    daniel.cho@nyumc.org    Principal Investigator: Daniel Cho, MD          United States, Tennessee Vanderbilt-Ingram Cancer Center Recruiting Nashville, Tennessee, United States, 37232 Contact: Jordan Berlin, MD          Contact       Jordan.Berlin@vanderbilt.edu    Principal Investigator: Jordan Berlin, MD          United States, Texas MD Anderson Cancer Center Recruiting Houston, Texas, United States, 77030 Contact: Aung Naing    713-563-0803    anaing@mdanderson.org    Principal Investigator: Aung Naing, MD          Canada, Ontario Princess Margaret Hospital Recruiting Toronto, Ontario, Canada, M5G 2M9 Contact: Albiruni Razak, MB, BCh    416-586-4800 ext 3883       Principal Investigator: Albiruni Razak, MB, Bch Collapse <<

实验方案

技术信息

CAS号 1643913-93-2 储存条件
分子式 C35H29F3N4O3 运输 蓝冰
分子量 610.63 别名 PAK4-IN-1

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