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CAS No.: 1365267-27-1
Synonyms: Ensartinib;Ensartinib-analog;X 396-analog
Ensartinib is a potent inhibitor ofALK, which is used to treat non-small-cell lung cancer.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT03574402 | Carcinoma, Non-Small-Cell Lung | Phase 2 | Not yet recruiting | December 30, 2024 | - |
NCT03155620 | Advanced Malignant Solid Neopl... more >>asm Ann Arbor Stage III Childhood Non-Hodgkin Lymphoma Ann Arbor Stage IV Childhood Non-Hodgkin Lymphoma Childhood Langerhans Cell Histiocytosis Histiocytic Sarcoma Juvenile Xanthogranuloma Malignant Glioma Recurrent Central Nervous System Neoplasm Recurrent Childhood Ependymoma Recurrent Childhood Malignant Germ Cell Tumor Recurrent Childhood Medulloblastoma Recurrent Childhood Non-Hodgkin Lymphoma Recurrent Childhood Rhabdomyosarcoma Recurrent Childhood Soft Tissue Sarcoma Recurrent Ewing Sarcoma Recurrent Glioma Recurrent Hepatoblastoma Recurrent Langerhans Cell Histiocytosis Recurrent Malignant Solid Neoplasm Recurrent Neuroblastoma Recurrent Osteosarcoma Recurrent Peripheral Primitive Neuroectodermal Tumor Recurrent Rhabdoid Tumor Refractory Central Nervous System Neoplasm Refractory Childhood Malignant Germ Cell Tumor Refractory Ewing Sarcoma Refractory Glioma Refractory Hepatoblastoma Refractory Langerhans Cell Histiocytosis Refractory Malignant Solid Neoplasm Refractory Medulloblastoma Refractory Neuroblastoma Refractory Non-Hodgkin Lymphoma Refractory Osteosarcoma Refractory Peripheral Primitive Neuroectodermal Tumor Refractory Rhabdoid Tumor Refractory Rhabdomyosarcoma Rhabdoid Tumor Stage III Osteosarcoma AJCC v7 Stage III Soft Tissue Sarcoma AJCC v7 Stage IV Osteosarcoma AJCC v7 Stage IV Soft Tissue Sarcoma AJCC v7 Stage IVA Osteosarcoma AJCC v7 Stage IVB Osteosarcoma AJCC v7 Wilms Tumor Collapse << | Phase 2 | Recruiting | September 30, 2027 | - |
NCT03215693 | Non-Small Cell Lung Cancer | Phase 2 | Recruiting | December 2018 | China ... more >> Beijing Cancer Hospital Recruiting Beijing, China Contact: Jian Fang, MD 13701224460 fangjian5555@163.com Principal Investigator: Jun Zhao, MD Beijing Chest Hospital,Capital Medical University Recruiting Beijing, China Contact: Shucai Zhang, MD 13901297065 sczhang6304@163.com Department of Medical Oncology, Cancer Institute/Hospital, Chinese Academy of Medical Sciences Recruiting Beijing, China Contact: Junling Li, MD 13801178891 drlijunling@vip.163.com Peking Union College Hospital Recruiting Beijing, China Contact: Wei Zhong, MD 13810616395 zw_pumch@126.com Collapse << |
实验方案
技术信息
CAS号 | 1365267-27-1 | 储存条件 |
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分子式 | C25H25Cl2FN6O3 | 运输 | 蓝冰 | |
分子量 | 547.41 | 别名 | Ensartinib;Ensartinib-analog;X 396-analog |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT03574402 | Carcinoma, Non-Small-Cell Lung | Phase 2 | Not yet recruiting | December 30, 2024 | - |
NCT03155620 | Advanced Malignant Solid Neopl... more >>asm Ann Arbor Stage III Childhood Non-Hodgkin Lymphoma Ann Arbor Stage IV Childhood Non-Hodgkin Lymphoma Childhood Langerhans Cell Histiocytosis Histiocytic Sarcoma Juvenile Xanthogranuloma Malignant Glioma Recurrent Central Nervous System Neoplasm Recurrent Childhood Ependymoma Recurrent Childhood Malignant Germ Cell Tumor Recurrent Childhood Medulloblastoma Recurrent Childhood Non-Hodgkin Lymphoma Recurrent Childhood Rhabdomyosarcoma Recurrent Childhood Soft Tissue Sarcoma Recurrent Ewing Sarcoma Recurrent Glioma Recurrent Hepatoblastoma Recurrent Langerhans Cell Histiocytosis Recurrent Malignant Solid Neoplasm Recurrent Neuroblastoma Recurrent Osteosarcoma Recurrent Peripheral Primitive Neuroectodermal Tumor Recurrent Rhabdoid Tumor Refractory Central Nervous System Neoplasm Refractory Childhood Malignant Germ Cell Tumor Refractory Ewing Sarcoma Refractory Glioma Refractory Hepatoblastoma Refractory Langerhans Cell Histiocytosis Refractory Malignant Solid Neoplasm Refractory Medulloblastoma Refractory Neuroblastoma Refractory Non-Hodgkin Lymphoma Refractory Osteosarcoma Refractory Peripheral Primitive Neuroectodermal Tumor Refractory Rhabdoid Tumor Refractory Rhabdomyosarcoma Rhabdoid Tumor Stage III Osteosarcoma AJCC v7 Stage III Soft Tissue Sarcoma AJCC v7 Stage IV Osteosarcoma AJCC v7 Stage IV Soft Tissue Sarcoma AJCC v7 Stage IVA Osteosarcoma AJCC v7 Stage IVB Osteosarcoma AJCC v7 Wilms Tumor Collapse << | Phase 2 | Recruiting | September 30, 2027 | - |
NCT03215693 | Non-Small Cell Lung Cancer | Phase 2 | Recruiting | December 2018 | China ... more >> Beijing Cancer Hospital Recruiting Beijing, China Contact: Jian Fang, MD 13701224460 fangjian5555@163.com Principal Investigator: Jun Zhao, MD Beijing Chest Hospital,Capital Medical University Recruiting Beijing, China Contact: Shucai Zhang, MD 13901297065 sczhang6304@163.com Department of Medical Oncology, Cancer Institute/Hospital, Chinese Academy of Medical Sciences Recruiting Beijing, China Contact: Junling Li, MD 13801178891 drlijunling@vip.163.com Peking Union College Hospital Recruiting Beijing, China Contact: Wei Zhong, MD 13810616395 zw_pumch@126.com Collapse << |
NCT03737994 | ALK Gene Rearrangement ... more >> ALK Positive Non-Squamous Non-Small Cell Lung Carcinoma Stage IV Lung Cancer AJCC v8 Stage IVA Lung Cancer AJCC v8 Stage IVB Lung Cancer AJCC v8 Collapse << | Phase 2 | Not yet recruiting | December 13, 2025 | - |
NCT01625234 | Advanced Solid Tumors ... more >> Non-small Cell Lung Cancer Collapse << | Phase 1 Phase 2 | Recruiting | November 2021 | - |
NCT03213652 | Advanced Malignant Solid Neopl... more >>asm ALK Fusion Protein Expression ALK Gene Mutation ALK Gene Translocation Ann Arbor Stage III Childhood Non-Hodgkin Lymphoma Ann Arbor Stage IV Childhood Non-Hodgkin Lymphoma Histiocytosis Recurrent Childhood Central Nervous System Neoplasm Recurrent Childhood Non-Hodgkin Lymphoma Recurrent Malignant Solid Neoplasm Recurrent Neuroblastoma Refractory Central Nervous System Neoplasm Refractory Malignant Solid Neoplasm Refractory Neuroblastoma Refractory Non-Hodgkin Lymphoma ROS1 Fusion Positive ROS1 Gene Mutation ROS1 Gene Translocation Collapse << | Phase 2 | Recruiting | September 30, 2024 | - |
NCT03753685 | Nonsmall Cell Lung Cancer ... more >> Brain Metastases Collapse << | Phase 2 | Not yet recruiting | October 2020 | - |
NCT03510611 | Non-Small Cell Lung Cancer | Phase 1 | Enrolling by invitation | July 2018 | China, Zhejiang ... more >> The 1st Phase Clinical Research Center of the Second Affiliated Hospital of Zhejiang University Medical College Hangzhou, Zhejiang, China, 311009 Collapse << |
NCT02898116 | Non-small Cell Lung Cancer ... more >> Carcinoma NSCLC Collapse << | Phase 1 Phase 2 | Completed | - | United States, New York ... more >> Research Facility New York, New York, United States, 10016 Collapse << |
NCT02767804 | Non-small Cell Lung Cancer | Phase 3 | Recruiting | April 2020 | - |
NCT03420508 | Melanoma | Phase 2 | Recruiting | January 2020 | United States, New Jersey ... more >> Memoral Sloan Kettering Monmouth Recruiting Middletown, New Jersey, United States, 07748 Contact: Alexander Shoushtari, MD 646-888-4161 Memorial Sloan Kettering Bergen Recruiting Montvale, New Jersey, United States, 07645 Contact: Alexander Shoushtari, MD 646-888-4161 United States, New York Memorial Sloan Kettering Westchester Recruiting Harrison, New York, United States, 10604 Contact: Alexander Shoushtari, MD 646-888-4161 Memorial Sloan Kettering Cancer Center Recruiting New York, New York, United States, 10065 Contact: Alexander Shoushtari, MD 646-888-4161 Contact: Paul Chapman, MD 646-888-4162 Principal Investigator: Alexander Shoushtari, MD Collapse << |
NCT02898116 | - | - | Completed | - | - |
NCT02959619 | Solid Tumor N... more >>on-Small Cell Lung Cancer Metastatic Collapse << | Phase 1 | Recruiting | June 2019 | China, Guangdong ... more >> Sun yat-sen Univerisity Cancer Center Recruiting Guanzhou, Guangdong, China, 510060 Principal Investigator: Li Zhang, MD Collapse << |
NCT03608007 | Lung Cancer R... more >>OS1 Gene Rearrangement Collapse << | Phase 2 | Recruiting | May 2020 | China, Zhejiang ... more >> Jinxiao Xu Recruiting Hangzhou, Zhejiang, China, 311100 Contact: Jinxiao Xu Principal Investigator: Shun Lu, Ph.D Collapse << |
NCT03536481 | Lung Cancer | Phase 1 | Not yet recruiting | December 31, 2018 | China, Shanghai ... more >> Shanghai Public Health Clinical Center Not yet recruiting Shanghai, Shanghai, China, 201508 Contact: Xianmin Meng 86 18916081980 scmxm@126.com Collapse << |
NCT03142906 | Anesthesia Ul... more >>trasound Emergencies Operation Ultrasonography Surgery Collapse << | Not Applicable | Recruiting | September 30, 2018 | Canada, Ontario ... more >> London Health Sciences Centre Recruiting London, Ontario, Canada, N6A 5A5 Contact: Ahmed Hegazy, Assist. Prof 5198604917 ahegazy@uwo.ca Contact: Osama Sefein, Resident 2263762815 osama.sefein@londonhospitals.ca Sub-Investigator: Osama Sefein, Resident Sub-Investigator: Kiarash Mohajer, Resident Sub-Investigator: Philip Jones, Assoc. Prof Sub-Investigator: Ramiro Arellano, Assoc. Prof Sub-Investigator: Robert Arntfield, Assist. Prof Sub-Investigator: Wilfredo Puentes, Assist. Prof Sub-Investigator: Jonathan Borger, Assist. Prof Collapse << |
NCT01980641 | Stroke | Not Applicable | Recruiting | February 2018 | Spain ... more >> IBIMA Recruiting Malaga, Malaag, Spain, 29017 Contact: Antonio Cuesta-Vargas, PhD Contact: Marina Tirado, MD Patronato Municipal de deportes de Torremolinos Completed Torremolinos, Malaga, Spain, 29620 Collapse << |
NCT03677661 | Post-Concussion Syndrome ... more >> Mild Traumatic Brain Injury Vestibular Disorder Whiplash Injuries Concussion, Brain Collapse << | Not Applicable | Not yet recruiting | October 1, 2020 | Canada, Quebec ... more >> Clinique Cortex Not yet recruiting Quebec city, Quebec, Canada, G1W 0C5 Contact: Pierre Langevin, pht, MClSc 418-955-7853 pierre.langevin@fmed.ulaval.ca Collapse << |
NCT00281580 | Hypertension | Phase 3 | Completed | - | - |
NCT00281580 | - | - | Completed | - | - |
NCT03256500 | Delirium Conf... more >>usion Collapse << | Not Applicable | Recruiting | June 30, 2020 | United States, Florida ... more >> Malcolm Randall Veterans Affairs Medical Center Recruiting Gainesville, Florida, United States, 32608 Contact: Uma Suryadevara, MD Contact: Colleen Campbell 352-376-1611 ext 6114 colleen.campbell@va.gov Principal Investigator: Uma Suryadevara, M.D Sub-Investigator: Colleen Campbell Sub-Investigator: Kenneth Heilman, M.D Sub-Investigator: Ronald Shorr, M.D Sub-Investigator: Joseph Thornton, M.D Sub-Investigator: Laurence Solberg, M.D Sub-Investigator: Adam Woods, Ph.D Sub-Investigator: Andrew Pierce, M.D Collapse << |
NCT02248701 | Spinal Cord Injury ... more >> Spinal Cord Injuries Trauma, Nervous System Wounds and Injuries Central Nervous System Diseases Nervous System Diseases Spinal Cord Diseases Gonadal Disorders Endocrine System Diseases Hypogonadism Genital Diseases, Male Collapse << | Phase 2 | Recruiting | June 1, 2019 | United States, Florida ... more >> North Florida/South Georgia Veterans Health System, Gainesville, FL Recruiting Gainesville, Florida, United States, 32608 Contact: Joshua F Yarrow, PhD MS BS 352-376-1611 ext 6477 joshua.yarrow@va.gov Contact: Dana M Otzel, PhD (352) 376-1611 ext 6917 Dana.Otzel@va.gov Principal Investigator: Joshua F Yarrow, PhD MS BS James A. Haley Veterans' Hospital, Tampa, FL Recruiting Tampa, Florida, United States, 33612 Contact: Joshua F Yarrow, PhD 352-376-1611 ext 6477 Joshua.Yarrow@va.gov Contact: Dana M Otzel, PhD 3523761611 ext 6917 Dana.Otzel@va.gov Collapse << |
NCT01641926 | Hepatitis B, Chronic | Phase 3 | Terminated(This study was term... more >>inated early due to poor recruitment) Collapse << | - | - |
NCT02672592 | Hypogonadism ... more >>Metabolic Syndrome X Obesity Collapse << | Phase 3 | Completed | - | Switzerland ... more >> University Department of Medicine, Kantonsspital Aarau Aarau, Switzerland, 5001 University Hospital Basel Basel, Switzerland, 4031 Collapse << |
NCT02667392 | Stroke | Phase 1 | Recruiting | January 31, 2019 | United States, Florida ... more >> North Florida/South Georgia Veterans Health System, Gainesville, FL Recruiting Gainesville, Florida, United States, 32608 Contact: Heidi Parrish (352) 376-1611 ext 105246 heidi.parrish@va.gov Contact: Margaret H McCallum (352) 376-1611 ext 5223 Margaret.McCallum@va.gov Principal Investigator: Dorian Kay Rose, PhD MS BS Collapse << |
NCT01641926 | - | - | Terminated(This study was term... more >>inated early due to poor recruitment) Collapse << | - | - |
NCT03719794 | Metabolic Syndrome | Not Applicable | Recruiting | September 2019 | Canada, Quebec ... more >> Cardiovascular Prevention and Rehabilitation Center Recruiting Montreal, Quebec, Canada, H1T 1N6 Contact: Julie Lalongé 5143741480 ext 4259 julie.lalonge@icm-mhi.org Principal Investigator: Anil Nigam, MD Collapse << |
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