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CAS No.: 845614-11-1
Synonyms: RG1678;RO4917838;R-1678
Bitopertin is a noncompetitive inhibitor of glycine reuptake with IC50 of 25 nM.
生物活性
动物研究 | |||||||||||||||||||||||||||||||||||||
剂量 | Mice: 0.1 mg/kg - 10 mg/kg[3] (i.p.); 0.3 mg/kg - 10 mg/kg[1] (p.o.) Rat: 0.3 mg/kg - 3 mg/kg[4] (p.o.), 1 mg/kg - 10 mg/kg[1] (p.o.) | ||||||||||||||||||||||||||||||||||||
给药途径 | i.p., p.o. | ||||||||||||||||||||||||||||||||||||
动物药代数据 |
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NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT01192906 | Schizophrenia | Phase 3 | Completed | - | - |
NCT01234779 | Schizophrenia | Phase 2 | Completed | - | - |
NCT01235559 | Schizophrenia | Phase 3 | Completed | - | - |
实验方案
技术信息
CAS号 | 845614-11-1 | 储存条件 |
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分子式 | C21H20F7N3O4S | 运输 | 蓝冰 | |||||
分子量 | 543.46 | 别名 | RG1678;RO4917838;R-1678;比托派汀 | |||||
溶解度 |
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动物实验配方 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT01192906 | Schizophrenia | Phase 3 | Completed | - | - |
NCT01234779 | Schizophrenia | Phase 2 | Completed | - | - |
NCT01235559 | Schizophrenia | Phase 3 | Completed | - | - |
NCT01235585 | Schizophrenia | Phase 3 | Completed | - | - |
NCT01636492 | Healthy Volunteer | Phase 1 | Completed | - | New Zealand ... more >> Christchurch, New Zealand, 8011 Collapse << |
NCT01192880 | Schizophrenia | Phase 3 | Completed | - | - |
NCT03271541 | Beta-Thalassemia | Phase 2 | Completed | - | Italy ... more >> Centro della Microcitemia e delle Anemie Congenite - Ospedale Galliera; Oncologia /Cardiologia Genova, Liguria, Italy, 16128 Ospedale Maggiore di Milano; Cardio-Metabolic Diseases Milano, Lombardia, Italy, 20122 Lebanon Chronic Care Center Baabda, Lebanon, 1003 Thailand Siriraj Hospital; Division of Haematology-Oncology Bangkok Noi, Thailand, 10700 Collapse << |
NCT01674361 | Obsessive-Compulsive Disorder | Phase 2 | Completed | - | - |
NCT02019290 | Healthy Volunteer | Phase 1 | Withdrawn | March 31, 2014 | - |
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