|2,2',2''-(苯-1,2,3-三基三(氧基))三(N,N,N-三乙基乙铵)碘化物|CsnPharm

CAS No.: 65-29-2

三碘季胺酚 Catalog No. CSN11077

Synonyms: Gallamine (iodide);Flaxedil;Tricuran

Gallamine triethiodide is a competitive cholinergic receptor blocker with an IC50 of 68.0 ± 8.4 μM, used as a non-depolarising muscle relaxant.

规格	价格	促销价格	库存	数量

400-920-2911

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靶点选择性

生物活性

实验方案

技术信息

生物活性

靶点 AChR

IC50:68.0±8.4μM
描述Gallamine Triethiodine is a cholinergic receptor inhibitor. It acts by combining with the cholinergic receptor sites in muscle and competitively blocking the transmitter action of acetylcholine. Gallamine triethiodide has a parasympatholytic effect on the cardiac vagus nerve which causes tachycardia and occasionally hypertension. Very high doses cause histamine release^[3]. Internal gallamine triethiodide modifies Na⁺ channel kinetics in Myxicola axons but does not alter K⁺ conductance^[4]. Slight accumulation of gallamine was noted in two of the four patients with biliary disease receiving multiple doses of gallamine, but this was also characteristic of data obtained in the patients without obstruction^[5].
参考文献

实验方案

计算器摩尔计算器总药量计算器工作液计算器
储存液制备
- 1 mg
- 5 mg
- 10 mg
- 1 mM
- 1.1217 mL
- 5.6083 mL
- 11.2167 mL
- 5 mM
- 0.2243 mL
- 1.1217 mL
- 2.2433 mL
- 10 mM
- 0.1122 mL
- 0.5608 mL
- 1.1217 mL

技术信息

CAS号

65-29-2

储存条件

粉末: Keep in dark place,Inert atmosphere,2-8°C

液体: -20°C:3-6 月 -80°C:12月

分子式

C30H60I3N3O3

运输

蓝冰

分子量

891.53

别名

Gallamine (iodide);Flaxedil;Tricuran;Gallamoni jodidum;Gallaminii iodidum;Iodide;Gallamonium;Gallamine Triethochloride;三碘季胺酚

溶解度

DMSO	150.0 mg/mL (168.3 mM)
Water	50.0 mg/mL (56.1 mM)

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