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CAS No.: 924298-51-1

3-((6-Methylpyridin-2-yl)ethynyl)cyclohex-2-en-1-one O-methyl oxime Catalog No. CSN22662

ABP 688 is a high affinity human mGlu5 receptor antagonist with Ki of 1.7 nM.

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靶点选择性

生物活性

  • 临床研究
  • NCT号适应症或疾病临床期招募状态预计完成时间地点
    NCT02727972Major Depressive Disorder ... more >> Post-Traumatic Stress Disorder Bipolar Disorder Collapse <<Not ApplicableRecruitingAugust 2020United States, Connecticut ... more >> PET Center Recruiting New Haven, Connecticut, United States, 06519 Contact: Sarah O, MA    203-737-7066       Principal Investigator: Irina Esterlis, PhD Collapse <<
    NCT01691092Major Depressive Disorder ... more >> Post-Traumatic Stress Disorder (PTSD) Collapse <<Not ApplicableCompleted-United States, Connecticut ... more >> Connecticut Mental Health Center New Haven, Connecticut, United States, 06519 Yale University Magnetic Resonance Research Center (MRRC) New Haven, Connecticut, United States, 06519 Yale University PET Center New Haven, Connecticut, United States, 06519 Collapse <<
    NCT01528241DepressionPhase 1Completed-United States, New York ... more >> Novartis Investigative Site New York, New York, United States United States, Pennsylvania Novartis Investigative Site Pittsburgh, Pennsylvania, United States Collapse <<
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实验方案

技术信息

CAS号 924298-51-1 储存条件
分子式 C15H16N2O 运输 蓝冰
分子量 240.30 别名

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