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CAS No.: 66085-59-4

尼莫地平 Catalog No. CSN12874

Synonyms: BAY-e 9736;Nimotop;Periplum

Nimodipine is a dihydropyridine derivative and an analogue of the calcium channel blocker nifedipine, with antihypertensive activity. Nimodipine decreases intracellular free Ca2+,Beclin-1 and autophagy.

规格 价格 促销价格 库存 数量
纯度 & 质量文件 批次:

靶点选择性

生物活性

  • 描述
  • 动物研究
    剂量

    Rat: 5 mg/kg - 15 mg/kg[3] (i.p.); 0.001 mg/kg = 0.1 mg/kg[4] (i.v.)

    给药途径

    i.p., i.v.

  • 临床研究
  • NCT号适应症或疾病临床期招募状态预计完成时间地点
    NCT03434314Aortic Aneurysm, Thoracoabdomi... more >>nal Collapse <<Not ApplicableNot yet recruitingSeptember 2021Austria ... more >> Medizinische Universität Innsbruck Not yet recruiting Innsbruck, Austria Contact: Michael Grimm, Prof. Dr.    +43 512 504 22500    michael.grimm@tirol-kliniken.at    Contact: Johannes Holfeld, Dr.       johannes.holfeld@i-med.ac.at    Herzzentrum Hietzing Not yet recruiting Vienna, Austria Contact: Martin Grabenwöger, Prof. Dr.    +43 1 4020585    Martin.Grabenwoeger@wienkav.at    Contact: Gabriel Weiss, Dr.       gabriel.weiss@wienkav.at    France University Hospital of Bordeaux Not yet recruiting Bordeaux, France Contact: Eric Ducasse, Prof. Dr.    +335 56 79 55 25    eric.ducasse@chu-bordeaux.fr    Marie Lannelongue Hospital Not yet recruiting Le Plessis-Robinson, France Contact: Stephan Haulon, Prof. Dr.          Germany Uniklinik RWTH Aachen Not yet recruiting Aachen, Germany Contact: Michael Jacobs, Prof. Dr.    +49 241 8085197    mjacobs@ukaachen.de    Contact: Drosos Kotelis, Dr.       dkotelis@ukaachen.de    Deutsches Herzzentrum Berlin Not yet recruiting Berlin, Germany Contact: Volkmar Falk, Prof. Dr.       falk@dhzb.de    Contact: Semih Buz, Dr.       buz@dhzb.de    Universitätsklinikum Düsseldorf Not yet recruiting Düsseldorf, Germany Contact: Hubert Schelzig, Prof. Dr.    0049 211 81 07211    hubert.schelzig@med.uni-duesseldorf.de    Contact: Alexander Oberhuber, Dr.       Alexander.Oberhuber@med.uni-duesseldorf.de    Westdeutsches Herz und Gefäßzentrum Essen Not yet recruiting Essen, Germany Contact: Heinz Jakob, Prof. Dr.    +49 201 723 4901    heinz.jakob@uk-essen.de    Contact: Konstantinos Tsagakis, Dr.       Konstantinos.Tsagakis@uk-essen.de    Universitäts-Herzzentrum Freiburg/ Bad Krozingen Not yet recruiting Freiburg, Germany Contact: Martin Czerny, Prof. Dr.    +49 7633 402 6216    martin.czerny@universitaets-herzzentrum.de    Herzzentrum Hamburg Not yet recruiting Hamburg, Germany Contact: Tilo Kölbel, Prof. Dr.    +49 40 7410 58609    t.koelbel@uke.de    Medizinische Hochschule Hannover Not yet recruiting Hanover, Germany Contact: Axel Haverich, Prof. Dr.    0049 511- 532 6580    haverich.axel@mh-hannover.de    Contact: Malakh Shrestha, Prof. Dr.    0049 511- 532 6238    Shrestha.Malakh.lal@mh-hannover.de    Universitätsklinikum Heidelberg Not yet recruiting Heidelberg, Germany Contact: Dittmar Böckler, Prof. Dr.    0049 6221 56 6249    dittmar.boeckler@med.uni-heidelberg.de    Contact: Moritz Bischoff, Dr.       moritz.bischoff@med.uni-heidelberg.de    Herzzentrum Leipzig Not yet recruiting Leipzig, Germany Contact: Christian D Etz, Prof. Dr.    +49 341 865 251007    christian.etz@medizin.uni-leipzig.de    UniversitätskIinikum Leipzig Not yet recruiting Leipzig, Germany Contact: Scheinert Dierk, Prof.Dr.    +49 341 97 18770    dierk.scheinert@medizin.uni-leipzig.de    Klinikum rechts der Isar (TU München) Not yet recruiting Munich, Germany Contact: Hans-Henning Eckstein, Prof. Dr.    +49 89 4140 9244    H.H.Eckstein@lrz.tum.de    Contact: Sarah Geisbüsch, Dr.       sarah.geisbuesch@mri.tum.de    Klinikum der Universität München (LMU) Not yet recruiting München, Germany Contact: Maximilian Luehr, Dr.    + 49 89 4400 72436    maximilian.luehr@med.uni-muenchen.de    St. Franziskus-Hospital GmbH Not yet recruiting Münster, Germany Contact: Giovanni Torsello, Prof. Dr.    0049 251 935-3933    giovanni.torsello@ukmuenster.de    Contact: Theodosios Bisdas, Dr.       theodosios.bisdas@sfh-muenster.de    Paracelsus Universität - Klinikum Nürnberg Not yet recruiting Nuremberg, Germany Contact: Eric Verhoeven, Prof. Dr.    0049 911 398 117004    eric.verhoeven@klinikum-nuernberg.de    Contact: Athanasios Katsargyris, Dr.       Athanasios.Katsargyris@klinikum-nuernberg.de    Universitätsklinikum Regensburg Not yet recruiting Regensburg, Germany Contact: Karin Pfister, Prof. Dr.    +49 941 944 6911    Karin.Pfister@klinik.uni-regensburg.de    Contact: Piotr Kasprzak, Prof. Dr.       piotr.kasprzak@ukr.de    Universitätsklinikum Tübingen Not yet recruiting Tübingen, Germany Contact: Christian Schlensak, Prof. Dr.    0049 7071 29 86638    christian.schlensak@med.uni-tuebingen.de    Contact: Mario Lescan, Dr.       mario.lescan@med.uni-tuebingen.de    Italy S.Orsola-Malpighi Hospital Not yet recruiting Bologna, Italy Contact: Davide Pacini, Prof. Dr.    +39 051 6363329    davide.pacini@unibo.it    Ospedale San Raffaele SRL Not yet recruiting Milano, Italy Contact: Roberto Chiesa, Prof. Dr.    +39 02 2643 7148    chiesa.roberto@unisr.it    Contact: Germano Melissano, Prof. Dr.    +39 02 2643 7148    melissano.germano@hsr.it    Netherlands Maastricht University Medical Center Not yet recruiting Maastricht, Netherlands Contact: Michael Jacobs, Prof. Dr.       m.jacobs@mumc.nl    Contact: Barend Mees, Dr.    +31 43 3877478    barend.mees@mumc.nl    Poland Medical University of Warsaw Not yet recruiting Warsaw, Poland Contact: Tomasz Jakimowicz, Dr.       tomj@wum.edu.pl    Silesian Center for Heart Diseases Not yet recruiting Zabrze, Poland Contact: Marian Zembala, Prof. Dr.    +48 323733689    m.zembala@sccs.pl; sek.kch@sccs.pl    Contact: Maciej K Kolowca, Dr.       maciej@kolowca.eu    Sweden Lund University Hospital Malmoe Not yet recruiting Malmö, Sweden Contact: Tim Resch, Dr.       tim.resch@med.lu.se    Örebro University Hospital Not yet recruiting Örebro, Sweden Contact: Thomas Larzon, Prof. Dr.       thomas.larzon@regionorebrolan.se    Switzerland Bern University Hospital Not yet recruiting Bern, Switzerland Contact: Jürg Schmidli, Prof. Dr.    +41 31 632 26 02    juerg.schmidli@insel.ch    United Kingdom St Bartholomews Hospital Not yet recruiting London, United Kingdom Contact: Aung Y Oo, Prof. Dr.       AungYe.OO@Bartshealth.nhs.uk Collapse <<
    NCT03718780Pulmonary Disease, Chronic Obs... more >>tructive Lung Diseases, Interstitial Chronic Heart Failure Pulmonary Arterial Hypertension Hyperventilation Syndrome Healthy Collapse <<Not ApplicableNot yet recruitingMarch 2020France ... more >> Service de pneumologie Not yet recruiting Béthune, France, 62408 Contact: Frédéric BART          Principal Investigator: Frédéric BART          Service de pneumologie CHMS Not yet recruiting Chambéry, France, 73000 Contact: Serge Kouzan          Sub-Investigator: Julien PERNOT          Sub-Investigator: Marie COUDURIER          Principal Investigator: Serge KOUZAN          Service de réanimation médicale - CHMS Not yet recruiting Chambéry, France, 73000 Contact: Jean-Marc THOURET       Jean-Marc.Thouret@ch-metropole-savoie.fr    Contact: Vincent PEIGNE       vincent.peigne@ch-metropole-savoie.fr    Sub-Investigator: Jean-Marc THOURET          Principal Investigator: Vincent PEIGNE          Service de Pneumologie CHU Grenoble Not yet recruiting La Tronche, France, 38700 Contact: Bernard AGUILANIU          Principal Investigator: Bernard AGUILANIU Collapse <<
    NCT00001478--Completed-United States, Maryland ... more >> National Institute of Mental Health (NIMH) Bethesda, Maryland, United States, 20892 Collapse <<
  • 更多
  • 参考文献

实验方案

技术信息

CAS号 66085-59-4 储存条件
分子式 C21H26N2O7 运输 蓝冰
分子量 418.44 别名 BAY-e 9736;Nimotop;Periplum;尼莫地平
溶解度
DMSO250.0 mg/mL (597.5 mM)
Waterinsoluble
动物实验配方

大规格询价

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