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CAS No.: 475479-34-6
Synonyms: R1439;RO0728804;RG-1439
Aleglitazar is a dual PPAR-α/γ agonist with IC50 of 2.8 nM/4.6 nM.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT01615354 | Healthy Volunteer | Phase 1 | Completed | - | United Kingdom ... more >> Manchester, United Kingdom, M13 9WL Collapse << |
NCT00388518 | Diabetes Mellitus Type 2 | Phase 2 | Completed | - | - |
NCT00461058 | Diabetes Mellitus Type 2 | Phase 2 | Completed | - | - |
实验方案
技术信息
CAS号 | 475479-34-6 | 储存条件 |
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分子式 | C24H23NO5S | 运输 | 蓝冰 | |
分子量 | 437.51 | 别名 | R1439;RO0728804;RG-1439;阿格列扎 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT01615354 | Healthy Volunteer | Phase 1 | Completed | - | United Kingdom ... more >> Manchester, United Kingdom, M13 9WL Collapse << |
NCT00388518 | Diabetes Mellitus Type 2 | Phase 2 | Completed | - | - |
NCT00461058 | Diabetes Mellitus Type 2 | Phase 2 | Completed | - | - |
NCT01398267 | Diabetes Mellitus Type 2 | Phase 1 | Completed | - | United States, California ... more >> Chula Vista, California, United States, 91911 United States, Nebraska Omaha, Nebraska, United States, 68154 United States, Texas Dallas, Texas, United States, 75247 San Antonio, Texas, United States, 78209 Collapse << |
NCT00461006 | Diabetes Mellitus Type 2 | Phase 2 | Completed | - | - |
NCT01729403 | Diabetes Mellitus Type 2 | Phase 2 | Completed | - | Germany ... more >> Neuss, Germany, 41460 Collapse << |
NCT01691989 | Diabetes Mellitus Type 2 | Phase 3 | Completed | - | - |
NCT01680978 | Diabetes Mellitus Type 2 | Phase 2 | Completed | - | United Kingdom ... more >> Oxford, United Kingdom, OX3 9DU Collapse << |
NCT01188317 | Healthy Volunteer | Phase 1 | Completed | - | United States, Nebraska ... more >> Omaha, Nebraska, United States, 68154 Collapse << |
NCT01893242 | Diabetes Mellitus Type 2, Kidn... more >>ey Disease, Chronic Collapse << | Phase 3 | Withdrawn | January 2019 | - |
NCT01042769 | Diabetes Mellitus Type 2 | Phase 3 | Completed | - | - |
NCT01691846 | Diabetes Mellitus Type 2 | Phase 3 | Completed | - | - |
NCT01871415 | Diabetes Mellitus Type 2 | Phase 3 | Completed | - | China ... more >> Shanghai, China, 200003 ShenYang, China, 110004 Shiyan, China, 442000 Suzhou, China, 215004 Korea, Republic of Gyeonggi-do, Korea, Republic of, 463-712 Incheon, Korea, Republic of, 405-760 Seoul, Korea, Republic of, 150-950 Collapse << |
NCT01188304 | Healthy Volunteer | Phase 1 | Completed | - | United States, Texas ... more >> San Antonio, Texas, United States, 78209 Collapse << |
NCT01715818 | Cardiovascular Disease, Diabet... more >>es Mellitus Type 2 Collapse << | Phase 3 | Completed | - | - |
NCT01871428 | Diabetes Mellitus Type 2 | Phase 3 | Completed | - | China ... more >> Chongqing, China, 400016 Shanghai, China, 200003 Shiyan, China, 442000 Suzhou, China, 215004 Hong Kong Hong Kong, Hong Kong Malaysia Alor Setar, Malaysia, 05400 Perak, Malaysia, 33400 Collapse << |
NCT01711775 | Healthy Volunteer | Phase 1 | Completed | - | China ... more >> Beijing, China, 100083 Collapse << |
NCT01691755 | Diabetes Mellitus Type 2 | Phase 3 | Completed | - | - |
NCT01679639 | Healthy Volunteer | Phase 1 | Completed | - | United Kingdom ... more >> Manchester, United Kingdom, M13 9WL Collapse << |
NCT01701739 | Healthy Volunteer | Phase 1 | Completed | - | United Kingdom ... more >> Manchester, United Kingdom, M13 9WL Collapse << |
NCT01197911 | - | - | Completed | - | - |
NCT01197911 | Healthy Volunteer | Phase 1 | Completed | - | United States, Florida ... more >> Orlando, Florida, United States, 32809 United States, Tennessee Knoxville, Tennessee, United States, 37920 Collapse << |
NCT01043029 | Diabetes Mellitus Type 2 | Phase 2 | Completed | - | - |
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