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CAS No.: 183232-66-8
AM251 is a potent CB1 receptor antagonist (IC50 = 8 nM, Ki = 7.49 nM) that displays 306-fold selectivity over CB2 receptors and also a potent GPR55 agonist (EC50 = 39 nM).
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT03160326 | - | - | Recruiting | March 2020 | United States, California ... more >> San Francisco VA Medical Center Recruiting San Francisco, California, United States, 94121 Contact: Julie Doyle 415-221-4810 ext 2597 Julie.Doyle2@va.gov Principal Investigator: Cynthia Delgado, MD United States, District of Columbia Washington DC VA Medical Center Recruiting Washington, District of Columbia, United States, 20422 Contact: Brian M Hoover, MS 202-745-8000 ext 55826 Brian.Hoover@va.gov Principal Investigator: Michael Harris-Love, DSc Sub-Investigator: Haniel Hernandez, DPT Sub-Investigator: Sholey Argani, MD Sub-Investigator: Marc Blackman, MD Collapse << |
实验方案
技术信息
CAS号 | 183232-66-8 | 储存条件 |
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分子式 | C22H21Cl2IN4O | 运输 | 蓝冰 | |
分子量 | 555.24 | 别名 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT03160326 | - | - | Recruiting | March 2020 | United States, California ... more >> San Francisco VA Medical Center Recruiting San Francisco, California, United States, 94121 Contact: Julie Doyle 415-221-4810 ext 2597 Julie.Doyle2@va.gov Principal Investigator: Cynthia Delgado, MD United States, District of Columbia Washington DC VA Medical Center Recruiting Washington, District of Columbia, United States, 20422 Contact: Brian M Hoover, MS 202-745-8000 ext 55826 Brian.Hoover@va.gov Principal Investigator: Michael Harris-Love, DSc Sub-Investigator: Haniel Hernandez, DPT Sub-Investigator: Sholey Argani, MD Sub-Investigator: Marc Blackman, MD Collapse << |
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