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CAS No.: 1029939-86-3

Artefenomel Catalog No. CSN18863

Synonyms: OZ439

Artefenomel is an antimalarial ozonide artefenomel which can maintain the rapid onset of action and potent activity of the artemisinin derivatives while exhibits greatly improved pharmacokinetics, low projected cost of goods, prophylactic activity, and the potential for a single dose cure.

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实验方案

技术信息

生物活性

描述Artefenomel is an antimalarial ozonide artefenomel which can maintain the rapid onset of action and potent activity of the artemisinin derivatives while exhibits greatly improved pharmacokinetics, low projected cost of goods, prophylactic activity, and the potential for a single dose cure.
临床研究

NCT号	适应症或疾病	临床期	招募状态	预计完成时间	地点
NCT01213966	Malaria, Falciparum ... more >> Malaria, Vivax Collapse <<	Phase 2	Completed	-	-
NCT03542149	Malaria	Phase 1	Recruiting	July 15, 2019	Australia, Queensland ... more >> Q-Pharm Recruiting Herston, Queensland, Australia, 4006 Contact: Brenda Cerqueira, MSc +61 (0) 439 726 233 B.Cerqueira@qpharm.com.au Contact: Priscila White, MSc +61 (0) 439 726 233 P.White@qpharm.com.au Collapse <<
NCT02573857	Malaria	Phase 1 Phase 2	Terminated	-	Australia, Queensland ... more >> Q-Pharm Clinics Herston, Queensland, Australia, 4006 Collapse <<

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参考文献

[1] Kim HS, Hammill JT, et al. Seeking the Elusive Long-Acting Ozonide: Discovery of Artefenomel (OZ439). J Med Chem. 2017 Apr 13;60(7):2651-2653.
[2] McCarthy JS, Baker M, et al. Efficacy of OZ439 (artefenomel) against early Plasmodium falciparum blood-stage malaria infection in healthy volunteers. J Antimicrob Chemother. 2016 Sep;71(9):2620-7.

实验方案

计算器摩尔计算器总药量计算器工作液计算器
储存液制备
- 1 mg
- 5 mg
- 10 mg
- 1 mM
- 2.1294 mL
- 10.6471 mL
- 21.2941 mL
- 5 mM
- 0.4259 mL
- 2.1294 mL
- 4.2588 mL
- 10 mM
- 0.2129 mL
- 1.0647 mL
- 2.1294 mL

技术信息

CAS号	1029939-86-3	储存条件	粉末液体 -20°C:3-6 月 -80°C:12月
分子式	C28H39NO5	运输	蓝冰
分子量	469.61	别名	OZ439

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NCT号	适应症或疾病	临床期	招募状态	预计完成时间	地点

NCT01213966	Malaria, Falciparum ... more >> Malaria, Vivax Collapse <<	Phase 2	Completed	-	-
NCT03542149	Malaria	Phase 1	Recruiting	July 15, 2019	Australia, Queensland ... more >> Q-Pharm Recruiting Herston, Queensland, Australia, 4006 Contact: Brenda Cerqueira, MSc +61 (0) 439 726 233 B.Cerqueira@qpharm.com.au Contact: Priscila White, MSc +61 (0) 439 726 233 P.White@qpharm.com.au Collapse <<
NCT02573857	Malaria	Phase 1 Phase 2	Terminated	-	Australia, Queensland ... more >> Q-Pharm Clinics Herston, Queensland, Australia, 4006 Collapse <<
NCT01213966	-	-	Completed	-	-
NCT02497612	Plasmodium Falciparum Infectio... more >>n Collapse <<	Phase 2	Recruiting	April 2, 2021	Benin ... more >> Investigational Site Number 204001 Recruiting Cotonou, Benin Burkina Faso Investigational Site Number 854001 Recruiting Nanoro, Burkina Faso Investigational Site Number 854003 Recruiting Niangoloko, Burkina Faso Investigational Site Number 854002 Recruiting Ouagadougou, Burkina Faso Gabon Investigational Site Number 266002 Recruiting Lambaréné, Gabon Investigational Site Number 266001 Recruiting Libreville, Gabon, B.P. 4009 Kenya Investigational Site Number 404002 Recruiting Kisian, Kenya Investigational Site Number 404003 Recruiting Kisumu, Kenya, 40100 Mozambique Investigational Site Number 508001 Recruiting Chokwe, Mozambique Uganda Investigational Site Number 800002 Recruiting Tororo, Uganda Vietnam Investigational Site Number 704003 Recruiting Binh Phuoc, Vietnam Investigational Site Number 704004 Recruiting Gia Lai, Vietnam Investigational Site Number 704001 Recruiting Khanh Hoa, Vietnam Investigational Site Number 704002 Recruiting Quang Tri, Vietnam Collapse <<
NCT03660839	Plasmodium Falciparum Infectio... more >>n Collapse <<	Phase 2	Recruiting	October 2019	Benin ... more >> Investigational Site Number 2040001 Recruiting Cotonou, Benin Burkina Faso Investigational Site Number 8540002 Recruiting Ouagadougou, Burkina Faso, 01 BP 2208 Investigational Site Number 8540001 Recruiting Ouagadougou, Burkina Faso, 01 BP218 Gabon Investigational Site Number 2660001 Recruiting Libreville, Gabon, B.P. 4009 Collapse <<
NCT02083380	Uncomplicated Plasmodium Falci... more >>parum Malaria Collapse <<	Phase 2 Phase 3	Completed	-	Benin ... more >> Centre D'Étude Et de Recherchesur Le Paludisme Associé À La Grossesse Et À L'Enfance (Cerpage) Cerpage Cotonou, Benin, FSS 01 BP 188 Burkina Faso Centre National de Recherche et de Formation sur le paludisme (CNRFP) Ouagadougou, Kadiogo Ouagadougou, Burkina Faso Clinical research Unit of Nanoro (CRUN)/CMA Saint Camille de Nanoro, 11 BP 218 Ouagadougou CMS 11 Ouagadougou, Burkina Faso Congo, The Democratic Republic of the Kinshasa School of Public Health, School of Medicine University of Kinshasa Kinshasa, Congo, The Democratic Republic of the Gabon Centre de Recherches Medicales de Lambarene, Albert Schweitzer Hospital Lambarene, Gabon arielle K. Bouyou-Akotet, Department of Parasitology-Mycology and Tropical Medicine, Faculty of Medicine, Université des Sciences de la Santé, BP 4009, Libreville, Gabon Libreville, Gabon Mozambique MANHIÇA HEALTH RESEARCH CENTER, Rua 12, Vila da Manhica, Maputa, Chefe Maputa, Mozambique Uganda Tororo District Hospital Tororo, Uganda Vietnam National Institute of Malariology, Parasitology and Entomology, 245 Luong The Vinh Street, Trung van, Tu Liem, Hanoi, Vietnam Hanoi, Vietnam Collapse <<
NCT02083380	-	-	Completed	-	-

Artefenomel Catalog No. CSN18863

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