CAS No.: 900515-16-4
AS-252424 Catalog No. CSN16052
AS-252424 is a potent PI3Kγ inhibitor with IC50 of 30 nM in a cell-free assay with 30-fold selectivity for PI3Kγ than PI3Kα, and low inhibitory activity towards PI3Kδ/β.
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纯度 & 质量文件
批次:
靶点选择性
生物活性
- 描述
- 细胞研究
- Cell Data
- 参考文献
- [1] Graves BM, Simerly T, et al. Phosphoinositide-3-kinase/akt - dependent signaling is required for maintenance of [Ca(2+)] (i), I(Ca), and Ca(2+) transients in HL-1 cardiomyocytes. J Biomed Sci. 2012 Jun 20;19:59.
- [2] Pomel V, Klicic J, et al. Furan-2-ylmethylene thiazolidinediones as novel, potent, and selective inhibitors of phosphoinositide 3-kinase gamma. J Med Chem. 2006 Jun 29;49(13):3857-71.
实验方案
- 计算器
- 储存液制备
技术信息
| CAS号 | 900515-16-4 | 储存条件 |
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| 分子式 | C14H8FNO4S | 运输 | 蓝冰 | |
| 分子量 | 305.28 | 别名 |
