CAS No.: 1190217-35-6
ASP7663 Catalog No. CSN20581
ASP 7663 is an orally-bioavailabe, selective TRPA1 activator (EC50 values are ~0.5 μM in human, mouse and rat), which displays little or no affinity at more than 60 other related receptors, channels and enzymes. It stimulates 5-HT release from QGP-1 cells and exhibits an abdominal analgesic effect in vivo.
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纯度 & 质量文件
批次:
靶点选择性
生物活性
- 描述
- 参考文献
- [1] Lu Y, Piplani H, et al. Transient Receptor Potential Ankyrin 1 Activation within the Cardiac Myocyte Limits Ischemia-reperfusion Injury in Rodents. Anesthesiology. 2016 Dec;125(6):1171-1180.
- [2] Kojima R, Nozawa K, et al. Effects of novel TRPA1 receptor agonist ASP7663 in models of drug-induced constipation and visceral pain. Eur J Pharmacol. 2014 Jan 15;723:288-93.
实验方案
- 计算器
- 储存液制备
技术信息
| CAS号 | 1190217-35-6 | 储存条件 |
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| 分子式 | C14H14FNO3 | 运输 | 蓝冰 | |
| 分子量 | 263.26 | 别名 |
