|1-(4-氟苯基)-4-(4-(吡啶-2-基)哌嗪-1-基)丁-1-酮|CsnPharm

CAS No.: 1649-18-9

Azaperone/阿扎佩隆 Catalog No. CSN12577

Synonyms: R-1929;NSC 170976;Stresnil

Azaperone functions as a dopamine antagonist that can bind to D1 and D2 receptors. It has the characteristics of antihistamines and anticholinergics.

规格	价格	促销价格	库存	数量

400-920-2911

sales@csnpharm.cn

tech@csnpharm.cn

加入购物车大规格询价

加入收藏

产品咨询

400-920-2911

sales@csnpharm.cn

tech@csnpharm.cn

纯度 & 质量文件批次:

靶点选择性

生物活性

实验方案

技术信息

生物活性

描述Administration of azaperone at weaning had a profound effect on preovulatory LH secretion as well as growth kinetics and estrogenicity of ovarian antral follicles^[3]. Thiafentanil and azaperone, with or without etorphine, delivered rapid safe, effective, reversible field anaesthesia in healthy swamp buffalo^[4]. Using azaperone alone the duration of immobility was 1.9 to 10.8 hours for mice and 0.9 to 2.4 hours for rats. The withdrawal reflex was not eliminated from mice receiving azaperone alone; however, the withdrawal reflex was eliminated from 0.9 to 2.4 hours in rats receiving azaperone. Azaperone produced a tachypnea in rats and male mice while a depressed respiratory rate was observed in female mice. Overall, azaperone alone was shown to provide sedation in mice as compared to a dose dependent anesthesia in rats. Azaperone and the azaperone-ketamine combination appear to be a suitable alternative to sedatives and anesthetics currently used in rats and mice^[5].
临床研究

NCT号	适应症或疾病	临床期	招募状态	预计完成时间	地点
NCT01486615	Anxiety	Phase 4	Completed	-	Nepal ... more >> B. P. Koirala Institute of Health Sciences Dharan, Koshi, Nepal, 56700 Dr Krishna Pokharel Dharan, Koshi, Nepal, 56700 Collapse <<
NCT01486615	-	-	Completed	-	-

参考文献

实验方案

计算器摩尔计算器总药量计算器工作液计算器
储存液制备
- 1 mg
- 5 mg
- 10 mg
- 1 mM
- 3.0544 mL
- 15.2720 mL
- 30.5441 mL
- 5 mM
- 0.6109 mL
- 3.0544 mL
- 6.1088 mL
- 10 mM
- 0.3054 mL
- 1.5272 mL
- 3.0544 mL

技术信息

CAS号

1649-18-9

储存条件

粉末: Sealed in dry,2-8°C

液体: -20°C:3-6 月 -80°C:12月

分子式

C19H22FN3O

运输

蓝冰

分子量

327.40

别名

R-1929;NSC 170976;Stresnil;Azaperon;Suicalm;Eucalmyl;阿扎哌隆

溶解度

DMSO	330.0 mg/mL (1008.0 mM) warming
Water	insoluble

动物实验配方

IP	2% DMSO+2% Tween80+30% PEG300+water	6 mg/mL	clear
PO	0.5% CMC-Na	62 mg/mL	suspension

大规格询价

号为必填项

姓名: 邮箱: 手机号:

留言:

提交

Azaperone/阿扎佩隆 Catalog No. CSN12577

靶点选择性

请登录您的专属账户

确认信息