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CAS No.: 1620576-64-8
AZD8835 ia a mixed inhibitor of PI3Kα and PI3Kδ with IC50 of 6.2 nM and 5.7 nM, respectively, also with selectivity against PI3Kβ (IC50=431 nM) and PI3Kγ (IC50=90 nM).
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT02260661 | Advanced Solid Malignancies ... more >> Breast Cancer - ER+, HER2 - Breast Cancer - ER+, HER2-, PIK3CA Gene Mutation Collapse << | Phase 1 | Completed | - | United States, Colorado ... more >> Research Site Denver, Colorado, United States United States, South Carolina Research Site Greenville, South Carolina, United States United States, Tennessee Research Site Nashville, Tennessee, United States United States, Texas Research Site Houston, Texas, United States United States, Wisconsin Research Site Milwaukee, Wisconsin, United States United Kingdom Research Site Cambridge, United Kingdom Sarah Cannon Research Institute, United Kingdom London, United Kingdom, W1G 6AD Research Site London, United Kingdom Research Site Manchester, United Kingdom Collapse << |
实验方案
技术信息
CAS号 | 1620576-64-8 | 储存条件 |
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分子式 | C22H31N9O3 | 运输 | 蓝冰 | |
分子量 | 469.54 | 别名 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT02260661 | Advanced Solid Malignancies ... more >> Breast Cancer - ER+, HER2 - Breast Cancer - ER+, HER2-, PIK3CA Gene Mutation Collapse << | Phase 1 | Completed | - | United States, Colorado ... more >> Research Site Denver, Colorado, United States United States, South Carolina Research Site Greenville, South Carolina, United States United States, Tennessee Research Site Nashville, Tennessee, United States United States, Texas Research Site Houston, Texas, United States United States, Wisconsin Research Site Milwaukee, Wisconsin, United States United Kingdom Research Site Cambridge, United Kingdom Sarah Cannon Research Institute, United Kingdom London, United Kingdom, W1G 6AD Research Site London, United Kingdom Research Site Manchester, United Kingdom Collapse << |
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