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CAS No.: 802904-66-1
Synonyms: AZD1981
AZD1981 is a potent and selective CRTh2 antagonist and displaces radio-labelled PGD2 from human recombinant DP2 with high potency (pIC50 = 8.4).
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT02367066 | Type 2 Diabetes Mellitus | Phase 1 | Completed | - | United States, California ... more >> Research Site Chula Vista, California, United States Collapse << |
NCT00766415 | Chronic Obstructive Pulmonary ... more >>Disease Collapse << | Phase 2 | Completed | - | Germany ... more >> Research Site Frieburg, Germany Research Site GROßHANSDORF, Germany Research Site Hannover, Germany Netherlands Research Site Amsterdam, Netherlands United Kingdom Research Site Leicester, United Kingdom Research Site London, United Kingdom Research Site Manchester, United Kingdom Research Site Newcastle upon Tyne, United Kingdom Collapse << |
NCT00766415 | - | - | Completed | - | - |
实验方案
技术信息
CAS号 | 802904-66-1 | 储存条件 |
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分子式 | C19H17ClN2O3S | 运输 | 蓝冰 | |||||||
分子量 | 388.87 | 别名 | AZD1981 | |||||||
溶解度 |
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动物实验配方 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT02367066 | Type 2 Diabetes Mellitus | Phase 1 | Completed | - | United States, California ... more >> Research Site Chula Vista, California, United States Collapse << |
NCT00766415 | Chronic Obstructive Pulmonary ... more >>Disease Collapse << | Phase 2 | Completed | - | Germany ... more >> Research Site Frieburg, Germany Research Site GROßHANSDORF, Germany Research Site Hannover, Germany Netherlands Research Site Amsterdam, Netherlands United Kingdom Research Site Leicester, United Kingdom Research Site London, United Kingdom Research Site Manchester, United Kingdom Research Site Newcastle upon Tyne, United Kingdom Collapse << |
NCT00766415 | - | - | Completed | - | - |
NCT01196689 | Asthma | Phase 1 | Completed | - | Sweden ... more >> Research Site Uppsala, Sweden Collapse << |
NCT00758589 | Asthma | Phase 2 | Completed | - | Argentina ... more >> Research Site Quilmes, Buenos Aires, Argentina Research Site San Miguel de Tucuman, Tucuman, Argentina Research Site Buenos Aires, Argentina Research Site Santa Fe, Argentina Brazil Research Site Porto Alegre, Brasil, Brazil Research Site Rio de Janeiro, RJ, Brazil Research Site Santo Andre, SP, Brazil Research Site Sao Paulo, SP, Brazil Costa Rica Research Site Barrio Los Yoses, San Jose, Costa Rica Research Site San Francisco de Dos Rios, San Jose, Costa Rica Poland Research Site Bialystok, Poland Research Site Bydgoszcz, Poland Research Site Gdalsk, Poland Research Site Kielce, Poland Research Site Krakow, Poland Research Site Lublin, Poland Research Site Poznal, Poland Research Site Szczecin, Poland Research Site Tarnow, Poland Research Site Turek, Poland Research Site Wroclaw, Poland Collapse << |
NCT00698282 | Healthy | Phase 1 | Completed | - | United Kingdom ... more >> Research Site Berkshire, United Kingdom Collapse << |
NCT00758589 | - | - | Completed | - | - |
NCT01254461 | Drug Interaction | Phase 1 | Completed | - | Sweden ... more >> Research Site Uppsala, Sweden Collapse << |
NCT01058447 | Healthy | Phase 1 | Completed | - | - |
NCT00918398 | Healthy Postm... more >>enopausal Surgically Sterile Women Collapse << | Phase 1 | Completed | - | Sweden ... more >> Research Site Uppsala, Sweden Collapse << |
NCT00690482 | - | - | Completed | - | - |
NCT01197794 | Asthma Patients | Phase 2 | Completed | - | - |
NCT02367066 | - | - | Completed | - | - |
NCT01265641 | Asthma | Phase 1 | Completed | - | United Kingdom ... more >> Researche Site London, UK, United Kingdom Collapse << |
NCT01110525 | Oral Contraceptives | Phase 1 | Completed | - | Sweden ... more >> Research Site Lulea, Sweden Research Site Uppsala, Sweden Collapse << |
NCT01199341 | Pharmakokinetic | Phase 1 | Completed | - | Sweden ... more >> Research Site Uppsala, Sweden Collapse << |
NCT00859352 | Healthy Male Volunteer | Phase 1 | Completed | - | Sweden ... more >> Research Site Uppsala, Sweden Collapse << |
NCT00690482 | Moderate to Severe COPD | Phase 2 | Completed | - | Bulgaria ... more >> Research Site Pleven, Bulgaria Research Site Russe, Bulgaria Research Site Sofia, Bulgaria Research Site Varna, Bulgaria Denmark Research Site Arhus C, Denmark Research Site Hellerup, Denmark Research Site Hvidovre, Denmark Research Site Vaerlose, Denmark Poland Research Site Krakow, Poland Research Site Lublin, Poland Research Site Ostrow Wielkopolski, Poland Research Site Przemysl, Poland Research Site Rzeszow, Poland Slovakia Research Site Bojnice, Slovakia Research Site Liptovsky Hradok, Slovakia Research Site Poprad, Slovakia Research Site Spisska Nova Ves, Slovakia Research Site Zilina, Slovakia Sweden Research Site Lund, Sweden Research Site Stockholm, Sweden Research Site Uppsala, Sweden Collapse << |
NCT01311635 | Healthy | Phase 1 | Completed | - | Sweden ... more >> Research Site Uppsala, Sweden Collapse << |
NCT02031679 | Chronic Idiopathic Urticaria | Phase 2 | Completed | - | United States, Maryland ... more >> Johns Hopkins Asthma and Allergy Center Baltimore, Maryland, United States, 21224-6821 Collapse << |
NCT02031679 | - | - | Completed | - | - |
NCT01197794 | - | - | Completed | - | - |
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