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CAS No.: 950736-05-7

B-Raf IN 1 Catalog No. CSN16988

Synonyms: B-RAF IN 1;B-RAF Inhibitor 1;MDK-36057

B-Raf IN 1 is a highlt potent and selective B-Raf inhibitor with IC50 of 24 nM, equipotent against c-Raf (IC50= 25 nM).

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靶点选择性

生物活性

  • 描述
  • 临床研究
  • NCT号适应症或疾病临床期招募状态预计完成时间地点
    NCT03430947Malignant Melanoma Stage IV ... more >> BRAF V600 Mutation Brain Metastases Collapse <<Phase 2RecruitingAugust 31, 2021Germany ... more >> Technische Universität Dresden Recruiting Dresden, Germany, 01307 Contact: Friedegund Meier, MD    +49 351 458 ext 2497    friedegund.meier@uniklinikum-dresden.de    Contact: Esther Troost, MD    +49 351 458 ext 2394    esther.troost@uniklinikum-dresden.de    Principal Investigator: Friedegund Meier, MD          Principal Investigator: Esther Troost, MD, PhD          Ruprecht-Karls-University of Heidelberg, Faculty of Medicine Not yet recruiting Heidelberg, Germany, 69120 Contact: Jessica Hassel, MD          Eberhard Karls University of Tübingen, University Medical Center Not yet recruiting Tuebingen, Germany, 72076 Contact: Thomas Eigentler, MD Collapse <<
    NCT01340846CancerPhase 1Completed-United States, Arizona ... more >> GSK Investigational Site Scottsdale, Arizona, United States, 85259 United States, Florida GSK Investigational Site Sarasota, Florida, United States, 34232 United States, Michigan GSK Investigational Site Detroit, Michigan, United States, 48201 United States, Ohio GSK Investigational Site Columbus, Ohio, United States, 43210 United States, Oklahoma GSK Investigational Site Oklahoma City, Oklahoma, United States, 73104 United States, South Carolina GSK Investigational Site Greenville, South Carolina, United States, 29605 United States, Tennessee GSK Investigational Site Nashville, Tennessee, United States, 37203 United States, Utah GSK Investigational Site Salt Lake City, Utah, United States, 84112 Australia, Western Australia GSK Investigational Site Nedlands, Western Australia, Australia, 6009 United Kingdom GSK Investigational Site Headington, United Kingdom, OX3 7LJ GSK Investigational Site London, United Kingdom, W1G 6AD Collapse <<
    NCT01909453MelanomaPhase 3Active, not recruitingMarch 31, 2019-
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实验方案

技术信息

CAS号 950736-05-7 储存条件
分子式 C29H24F3N5O 运输 蓝冰
分子量 515.53 别名 B-RAF IN 1;B-RAF Inhibitor 1;MDK-36057

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