CAS No.: 1187595-84-1
Baricitinib phosphate/磷酸巴瑞克替尼 Catalog No. CSN17535
Synonyms: LY3009104 phosphate;INCB028050 phosphate;INCB-028050
Baricitinib Phosphate can selectively inhibit JAK1/2 inhibitor with IC50 values of 5.9 nM and 5.7 nM.
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纯度 & 质量文件
批次:
靶点选择性
生物活性
靶点 JAK2
IC50:5.7nMJAK1
IC50:5.9nM- 描述
- 临床研究
NCT号 适应症或疾病 临床期 招募状态 预计完成时间 地点 NCT01398475 Chronic Inflammatory Disorder ... more >> Arthritis, Rheumatoid Collapse << Phase 1 Completed - Singapore ... more >> For additional information regarding investigative sites for this trial, contact 1-877-CTLILLY (1-877-285-4559, 1-317-615-4559) Mon - Fri from 9 AM to 5 PM Eastern Time (UTC/GMT - 5 hours, EST), or speak with your personal physician. Singapore, Singapore, 117597 Collapse << NCT01398475 - - Completed - - - 参考文献
- [1] Jabbari A, Dai Z, et al. Reversal of Alopecia Areata Following Treatment With the JAK1/2 Inhibitor Baricitinib. EBioMedicine. 2015 Feb 26;2(4):351-5.
- [2] Fridman JS, Scherle PA, et al. Selective inhibition of JAK1 and JAK2 is efficacious in rodent models of arthritis: preclinical characterization of INCB028050. J Immunol. 2010 May 1;184(9):5298-307.
实验方案
- 计算器
- 储存液制备
技术信息
| CAS号 | 1187595-84-1 | 储存条件 |
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| 分子式 | C16H20N7O6PS | 运输 | 蓝冰 | |||
| 分子量 | 469.41 | 别名 | LY3009104 phosphate;INCB028050 phosphate;INCB-028050;INCB-28050;LY-3009104;Baricitinib Phosphate;Olumiant;磷酸巴瑞克替尼 | |||
| 溶解度 |
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动物实验配方 |
