CAS No.: 802906-73-6
Basimglurant Catalog No. CSN15700
Synonyms: RG7090;CTEP Derivative
RG7090 is a potent, selective and orally available mGlu5 negative allosteric modulator with a Kd of 1.1 nM.
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纯度 & 质量文件
批次:
靶点选择性
生物活性
- 描述
- 参考文献
- [1] Lindemann L, Porter RH, et al. Pharmacology of basimglurant (RO4917523, RG7090), a unique metabotropic glutamate receptor 5 negative allosteric modulator in clinical development for depression. J Pharmacol Exp Ther. 2015 Apr;353(1):213-33.
- [2] Jaeschke G, Kolczewski S, et al. Metabotropic glutamate receptor 5 negative allosteric modulators: discovery of 2-chloro-4-[1-(4-fluorophenyl)-2,5-dimethyl-1H-imidazol-4-ylethynyl] pyridine (basimglurant, RO4917523), a promising novel medicine for psychiatric diseases. J Med Chem. 2015 Feb
实验方案
- 计算器
- 储存液制备
技术信息
| CAS号 | 802906-73-6 | 储存条件 |
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| 分子式 | C18H13ClFN3 | 运输 | 蓝冰 | |||||
| 分子量 | 325.77 | 别名 | RG7090;CTEP Derivative | |||||
| 溶解度 |
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动物实验配方 |
