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CAS No.: 5579-84-0
Synonyms: PT-9;Betahistine (hydrochloride);Betahistine HCl
Betahistine 2HCl is histamine H3 receptor inhibitor with IC50 of 1.9 μM. It is an antivertigo drug.
生物活性
靶点 | Histamine Receptor H3 IC50:1.9μM |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT02516072 | Remote Ischaemic Preconditioni... more >>ng Contrast Induced Nephropathy Collapse << | Not Applicable | Recruiting | October 2019 | Singapore ... more >> Changi General Hospital Recruiting Singapore, Singapore, 529889 Contact: Tjun Yip Tang 81610293 Tjun_Yip_Tang@cgh.com.sg Principal Investigator: Tjun Yip Tang Collapse << |
NCT02475239 | Benign Paroxysmal Positional V... more >>ertigo Collapse << | Not Applicable | Unknown | June 2017 | Thailand ... more >> Yuvatiya Plodpoai Recruiting Hatyai, Songkhla, Thailand, 90110 Contact: Yuvatiya Plodpoa, MD 66015988403 yuvatiya.plodpai@gmail.com Collapse << |
NCT01287975 | Stroke | Not Applicable | Completed | - | Singapore ... more >> Tan Tock Seng Hospital Rehabilitation Centre Singapore, Singapore, 569766 Collapse << |
实验方案
技术信息
CAS号 | 5579-84-0 | 储存条件 |
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分子式 | C8H14Cl2N2 | 运输 | 蓝冰 | |||||||
分子量 | 209.12 | 别名 | PT-9;Betahistine (hydrochloride);Betahistine HCl;brand names Veserc;Serc;Hiserk;Betaserc;Vergo;盐酸倍他司汀 | |||||||
溶解度 |
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动物实验配方 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT02516072 | Remote Ischaemic Preconditioni... more >>ng Contrast Induced Nephropathy Collapse << | Not Applicable | Recruiting | October 2019 | Singapore ... more >> Changi General Hospital Recruiting Singapore, Singapore, 529889 Contact: Tjun Yip Tang 81610293 Tjun_Yip_Tang@cgh.com.sg Principal Investigator: Tjun Yip Tang Collapse << |
NCT02475239 | Benign Paroxysmal Positional V... more >>ertigo Collapse << | Not Applicable | Unknown | June 2017 | Thailand ... more >> Yuvatiya Plodpoai Recruiting Hatyai, Songkhla, Thailand, 90110 Contact: Yuvatiya Plodpoa, MD 66015988403 yuvatiya.plodpai@gmail.com Collapse << |
NCT01287975 | Stroke | Not Applicable | Completed | - | Singapore ... more >> Tan Tock Seng Hospital Rehabilitation Centre Singapore, Singapore, 569766 Collapse << |
NCT02648945 | Aerobic Exercise | Not Applicable | Unknown | - | Malaysia ... more >> Universiti Tunku Abdul Rahman Recruiting Kajang, Selangor, Malaysia, 43000 Contact: Manisha Parai, MPT 0173128276 Collapse << |
NCT02649452 | Healthy | Not Applicable | Unknown | - | Malaysia ... more >> Universiti Tunku Abdul Rahman Recruiting Kajang, Selangor, Malaysia, 43000 Contact: Manisha Parai, MPT 0173128276 Collapse << |
NCT02645292 | Sedentary Lifestyle | Phase 1 | Completed | - | - |
NCT02781402 | Overweight | Not Applicable | Completed | - | - |
NCT03376334 | Balance | Not Applicable | Completed | - | Malaysia ... more >> Universiti Tunku Abdul Rahman Cheras, Selangor, Malaysia, 43000 Collapse << |
NCT03737890 | Pulmonary Function in Frail El... more >>derly Collapse << | Not Applicable | Completed | - | Malaysia ... more >> Universiti Tunku Abdul Rahman Kajang, Selangor, Malaysia, 43000 Collapse << |
NCT02185222 | Memory Disorders ... more >> Age-Related Cognitive Decline Collapse << | Phase 3 | Recruiting | July 2018 | France ... more >> Chu Angers Recruiting Angers, France, 49933 Contact: Cédric ANNWEILER, PH CeAnnweiler@chu-angers.fr Principal Investigator: Cédric ANNWEILER, PH CH BLOIS Recruiting Blois, France Contact: Patrick FRIOCOURT, PH pfriocourt@ch-blois.fr Principal Investigator: Patrick FRIOCOURT, PH CHU BREST - Hôpital de la Cavale Blanche Not yet recruiting Brest, France, 29200 Contact: Armelle GENTRIC, PU-PH armelle.gentric@chu-brest.fr Principal Investigator: Armelle GENTRIC, PU-PH CHI ELBEUF Louviers Val-de-Reuil Recruiting Elbeuf, France Contact: Thibault SIMON, PH thibault.simon@chi-elbeuf-louviers.fr Principal Investigator: Thibault SIMON, PH CHU NANTES - Hôpital Bellier Recruiting Nantes, France, 44093 Contact: Sophie PICHIERRI, PH sophie.pichierri@chu-nantes.fr Principal Investigator: Sophie PICHIERRI, PH CHU NANTES - Hôpital Laënnec Recruiting Nantes, France, 44093 Contact: Claire BOUTOLEAU-BRETONNIERE claire.boutoleaubretonniere@chu-nantes.fr Principal Investigator: Claire BOUTOLEAU-BRETONNIERE, PH Chr Orleans Recruiting Orléans, France, 45067 Contact: Jean-Bernard GAUVAIN, PH jean-bernard.gauvain@chr-orleans.fr Principal Investigator: Jean-Bernard GAUVAIN, PH CHU POITIERS - Hôpital de la Milétrie Recruiting Poitiers, France, 86021 Contact: Marc PACCALIN, PU-PH m.paccalin@chu-poitiers.fr Principal Investigator: Marc PACCALIN, PU-PH CHU RENNES - Hôpital Hôtel Dieu Recruiting Rennes, France, 35064 Contact: Aline CORVOL, PH aline.corvol@chu-rennes.fr Principal Investigator: Aline CORVOL, PH CHU ROUEN - Hôpital Charles Nicolle Recruiting Rouen, France, 76031 Contact: Caroline LEVASSEUR, PH caroline.levasseur@chu-rouen.fr Principal Investigator: Caroline LEVASSEUR, PH CHRU TOURS - Hôpital Bretonneau Not yet recruiting Tours, France, 37044 Contact: Fanny HENNEKINNE, PH fanny.hennekinne@univ-tours.fr Principal Investigator: Fanny HENNEKINNE, PH Collapse << |
NCT01717131 | Invasive Breast Cancer | Phase 3 | Recruiting | July 2028 | France ... more >> Gilles HOUVENAEGHEL, PHD Recruiting Marseille, France, 13009 Contact: Gilles HOUVENAEGHEL, PhD 33(0)491223778 drci.up@ipc.unicancer.fr Collapse << |
NCT01660087 | Lung Cancer | Not Applicable | Withdrawn | - | Singapore ... more >> Institute of Microelectronics Singapore, Singapore, 117685 National University Hospital/ National University of Singapore Singapore, Singapore, 119074 Collapse << |
NCT02717793 | No Condition, Healthy Females | Phase 1 | Completed | - | Malaysia ... more >> Manisha Kajang, Selangor, Malaysia, 43000 Collapse << |
NCT03581396 | - | - | Recruiting | June 2019 | France ... more >> Service Imagerie 1 Recruiting Strasbourg, France, 67091 Contact: Aïna VENKATASAMY, MD 33 3 88 12 78 65 aina.venkatasamy@chru-strasbourg.fr Contact: Pauline BRETZ, MD 33 3 88 12 78 65 paulinebretz@hotmail.com Principal Investigator: Aïna VENKATASAMY, MD Sub-Investigator: Pauline BRETZ, MD Sub-Investigator: Francis VEILLON, MD, PhD Collapse << |
NCT02724982 | - | - | Completed | - | Malaysia ... more >> Universiti Tunku Abdul Rahman Kajang, Selangor, Malaysia, 43000 Collapse << |
NCT01077622 | - | - | Completed | - | - |
NCT01580345 | Pregnancy | Phase 3 | Completed | - | India ... more >> KLEUs Jawaharlal Nehru Medical College- Prabhakar Kore Charitable Hospital Belgaum, Karnataka, India, 590010 Collapse << |
NCT00474409 | Vertigo | Phase 4 | Withdrawn(Due to poor enrollme... more >>nt, this study was withdrawn/ terminated.) Collapse << | - | China, Beijing ... more >> Beijing Tiantan Hospital Beijing, Beijing, China, 100050 Beijing Hospital Beijing, Beijing, China, 100730 China, Shanghai Shanghai Renji Hospital Shanghai, Shanghai, China, 20001 Shanghai Huashan Hospital Shanghai, Shanghai, China, 200040 Collapse << |
NCT02896374 | Schizophrenia | Not Applicable | Completed | - | France ... more >> Centre Hospitalier de Versailles Le Chesnay, France, 78150 Collapse << |
NCT01077622 | Leukaemia, Lymphocytic, Chroni... more >>c Collapse << | Phase 2 | Completed | - | Japan ... more >> GSK Investigational Site Aichi, Japan, 466-8650 GSK Investigational Site Kanagawa, Japan, 259-1143 GSK Investigational Site Nagasaki, Japan, 852-8501 GSK Investigational Site Tokyo, Japan, 104-0045 GSK Investigational Site Tokyo, Japan, 135-8550 Korea, Republic of GSK Investigational Site Seoul, Korea, Republic of, 110-744 GSK Investigational Site Seoul, Korea, Republic of, 138-736 Collapse << |
NCT02026778 | Nausea and Vomiting | Not Applicable | Unknown | December 2014 | Korea, Republic of ... more >> Department of Anesthesiology and Pain Medicine, Yonsei University College of Medicine Recruiting Seoul, Korea, Republic of, 120-752 Contact: Bon Nyeo Koo, MD 82-2-2227-7897 koobn@yuhs.ac Collapse << |
NCT01969513 | Benign Positional Paroxysmal V... more >>ertigo Collapse << | Not Applicable | Completed | - | Spain ... more >> CAP Florida L'Hospitalet de Llobregat, Barcelona, Spain, 08905 Collapse << |
NCT03624283 | Vestibular Disorder | Not Applicable | Recruiting | July 31, 2020 | China, Shanghai ... more >> Otorhinolaryngology Department of Affiliated Eye and ENT Hospital, Fudan University, Shanghai, China Recruiting Shanghai, Shanghai, China, 200031 Contact: Huawei Li, Phd &MD hwli@shmu.edu.cn Contact: Peixia Wu, MS &MD 13524844652@163.com Collapse << |
NCT00160238 | Meniere's Disease | Phase 4 | Completed | - | France ... more >> Site 1 Marseille, France Collapse << |
NCT00409305 | Obesity | Phase 2 | Completed | - | United States, Alabama ... more >> Cahaba Research, Inc. Birmingham, Alabama, United States, 35242 United States, California Scripps Clinic, Nutrition Metabolic Research San Diego, California, United States, 92130 Diablo Clinical Research, Inc. Walnut Creek, California, United States, 94598 United States, Florida Miami Research Associates, Inc., Nutrition Division Miami, Florida, United States, 33143 United States, Georgia CSRA Partners in Health, Inc. Augusta, Georgia, United States, 30909 United States, Illinois Radiant Research, Inc. Chicago, Illinois, United States, 60610 NCCR Chicago, Illinois, United States, 60611 United States, Indiana American Health Network Indianapolis, Indiana, United States, 46254 Midwest Institute for Clinical Research Indianapolis, Indiana, United States, 46260 United States, Kansas Radiant Research, Inc. Overland Park, Kansas, United States, 66215 United States, Kentucky L-MARC Research Center Louisville, Kentucky, United States, 40213 United States, Louisiana Pennington Biomedical Research Center Baton Rouge, Louisiana, United States, 70808 United States, Minnesota Radiant Research, Inc. Edina, Minnesota, United States, 55435 United States, Missouri Diabetes & Endocrinology Specialists Chesterfield, Missouri, United States, 63017 United States, New York Comprehensive Weight Control Program New York, New York, United States, 10021 Rochester Clinical Research, Inc. Rochester, New York, United States, 14609 United States, Ohio Lindner Clinical Trial Center Cincinnati, Ohio, United States, 45219 United States, Oregon Covance CRU, Inc. Portland, Oregon, United States, 97239 United States, Texas Diabetes & Glandular Disease Research Associates, Inc. San Antonio, Texas, United States, 78229 Collapse << |
NCT00428168 | Weight Gain | Phase 2 | Terminated(Interim Analysis re... more >>sult indicated the study will not show a significant benefit of the study medication on the primary endpoint.) Collapse << | - | Canada, Alberta ... more >> Capital Health, Edmonton Mental Health Clinic Edmonton, Alberta, Canada, T5K 2J5 Canada, British Columbia Dr. Alexander McIntyre Penticton, British Columbia, Canada, V2A 4M4 Vancouver Island Health Authority Victoria, British Columbia, Canada, V8R 4Z3 Canada, Manitoba Dr. Ivan Kowalchuk Winnipeg, Manitoba, Canada, R3K 2E2 Canada, Nova Scotia Capital District Health Authority Halifax, Nova Scotia, Canada, B3H 2E2 Canada, Ontario Queen's University Kingston, Ontario, Canada, K7L 5G2 Canada, Quebec Douglas Hospital Research Centre Verdun (Montreal), Quebec, Canada, H4H 1R3 Israel Abarbanel Hospital Bat Yam, Israel Geha Psychiatric Hospital Petach Tikva, Israel, 49100 Lev Hasharon Tirat Hacarmel, Israel Collapse << |
NCT00466869 | Hypercholesterolemia | Phase 2 | Terminated(Sponsor decision) | - | Israel ... more >> Internal Medicine Department A-Wolfson Medical Center Holon, Israel Internal Medicine Department A-Meir Medical Center Kfar Saba, Israel Collapse << |
NCT01759251 | - | - | Completed | - | Russian Federation ... more >> Site reference ID 89414 Belgorod, Russian Federation, 308007 Research facility ID ORG-000838 Irkutsk, Russian Federation, 664047 Site reference ID 89433 Kazan, Russian Federation, 420012 Site reference ID 89454 Moscow, Russian Federation, 119991 Site reference ID 89419 Moscow, Russian Federation, 123007 Research facility ID ORG-000837 Moscow, Russian Federation, 125047 Site reference ID 94374 Moscow, Russian Federation, 127006 Site reference ID 89416 Moscow, Russian Federation, 129110 Site reference ID 89435 Novosibirsk, Russian Federation, 630091 Research facility ID ORG-000841 Odintsovo, Russian Federation, 143007 Site reference ID 89453 Rostov-on-Don, Russian Federation, 344010 Site reference ID 89418 Saratow, Russian Federation, 410012 Site reference ID 89456 St. Petersburg, Russian Federation, 198255 Site reference ID 89415 Ufa, Russian Federation, 450009 Site reference ID 89455 Volgograd, Russian Federation, 400134 Ukraine Research facility ID ORG-000345 Donetsk, Ukraine, 83045 Site reference ID 93715 Ivano-Frankivsk, Ukraine, 76014 Site reference ID 93713 Kharkiv, Ukraine, 61000 Site reference ID 93454 Kiev, Ukraine, 04112 Site reference ID 93475 Mykolaiv, Ukraine, 54001 Site reference ID 93714 Sevastopol, Ukraine, 99011 Site reference ID 93474 Simferopol, Ukraine, 95006 Site reference ID 95738 Zaporizhzhia, Ukraine, 69032 Site reference ID 93455 Zaporizhzhia, Ukraine, 69060 Collapse << |
NCT00829881 | Attention Deficit Disorder Wit... more >>h Hyperactivity Collapse << | Phase 1 | Completed | - | United States, Ohio ... more >> University of Cincinnati; Department of Psychiatry Cincinnati, Ohio, United States, 45219 Collapse << |
NCT01759251 | - | - | Completed | - | - |
NCT00709202 | Schizophrenia ... more >> Schizoaffective Disorder Schizophreniform Disorder Bipolar I Disorder Bipolar II Bipolar NOS Psychotic Disorder Not Otherwise Specified Autism Collapse << | Phase 2 | Completed | - | United States, New York ... more >> Nathan Kline Insitute for Psychiatric Research Orangeburg, New York, United States, 10962 Collapse << |
NCT00459992 | Obesity Overw... more >>eight Overnutrition Collapse << | Phase 1 | Completed | - | United States, Maryland ... more >> National Institutes of Health Clinical Center, 9000 Rockville Pike Bethesda, Maryland, United States, 20892 Collapse << |
NCT01468285 | Gait or Balance Disorder Probl... more >>ems Collapse << | Phase 4 | Completed | - | Singapore ... more >> Site Reference ID/Investigator# 63545 Singapore, Singapore, 169608 Site Reference ID/Investigator# 63544 Singapore, Singapore, 308433 Collapse << |
NCT00748436 | Obesity | Phase 2 | Completed | - | Belgium ... more >> GP: Dr. Van Mulders Aalst, Belgium, 9310 UZ Antwerpen Edegem, Belgium, 2650 UZ Gent Gent, Belgium, 9000 UZ Leuven Leuven, Belgium, 3000 Germany Zentrum für Therapiestudien Leipzig, Germany, 04103 CRS Clinical Research Services Mönchengladbach, Germany, 41061 Netherlands Emotional Brain Almere, Netherlands, 1311 GP: Dr. Rol Bennebroek, Netherlands, 2121 AMWO Den Haag, Netherlands, 2582 Wecor Etten-leur, Netherlands, 4873 PT&R Geleen, Netherlands, 6166 AMWO Rotterdam, Netherlands, 3081 Collapse << |
NCT00852956 | Healthy | Phase 1 | Completed | - | Romania ... more >> IFE Human Pharmacology Arad, Romania IFE Human Pharmacology Timisoara, Romania Collapse << |
NCT01168336 | Healthy | Phase 1 | Completed | - | Romania ... more >> Pierrel Research HP-RO Arad, Romania Pierrel Research HP-RO Timisoara, Romania, RO-300244 Collapse << |
NCT00585585 | Recurrent Major Depressive Dis... more >>order With Atypical Features Collapse << | Phase 2 | Terminated(Lack of participant... more >>s) Collapse << | - | United States, Ohio ... more >> University of Cincinnati Cincinnati, Ohio, United States, 45267-0559 Collapse << |
NCT00585585 | - | - | Terminated(Lack of participant... more >>s) Collapse << | - | - |
靶点 | Description | IC50 |
---|---|---|
Histamine Receptor H3 | IC50:1.9μM |
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