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CAS No.: 890128-81-1
Synonyms: BFH772
BFH772 selectively targets VEGFR2 kinase with IC50 of 3 nM.
生物活性
靶点 | VEGFR2 IC50:3nM |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT00987870 | Psoriasis Art... more >>hritis Collapse << | Phase 1 Phase 2 | Completed | - | Germany ... more >> Novartis Investigator Site Berlin, Germany Collapse << |
NCT01449591 | Erythemato-telangiectatic Rosa... more >>cea Collapse << | Phase 2 | Completed | - | United States, Arkansas ... more >> Novartis Investigative Site Hot Springs, Arkansas, United States United States, Michigan Novartis Investigative Site Ann Abor, Michigan, United States United States, New Jersey Novartis Investigative Site Paramus, New Jersey, United States United States, Oregon Novartis Investigative Site Portland, Oregon, United States United States, Texas Novartis Investigative Site Austin, Texas, United States United States, Washington Novartis Investigative Site Spokane, Washington, United States Collapse << |
实验方案
技术信息
CAS号 | 890128-81-1 | 储存条件 |
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分子式 | C23H16F3N3O3 | 运输 | 蓝冰 | |||||||
分子量 | 439.39 | 别名 | BFH772 | |||||||
溶解度 |
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动物实验配方 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT00987870 | Psoriasis Art... more >>hritis Collapse << | Phase 1 Phase 2 | Completed | - | Germany ... more >> Novartis Investigator Site Berlin, Germany Collapse << |
NCT01449591 | Erythemato-telangiectatic Rosa... more >>cea Collapse << | Phase 2 | Completed | - | United States, Arkansas ... more >> Novartis Investigative Site Hot Springs, Arkansas, United States United States, Michigan Novartis Investigative Site Ann Abor, Michigan, United States United States, New Jersey Novartis Investigative Site Paramus, New Jersey, United States United States, Oregon Novartis Investigative Site Portland, Oregon, United States United States, Texas Novartis Investigative Site Austin, Texas, United States United States, Washington Novartis Investigative Site Spokane, Washington, United States Collapse << |
靶点 | Description | IC50 |
---|---|---|
VEGFR2 | IC50:3nM |
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