CAS No.: 501437-28-1
BI-D1870 Catalog No. CSN12314
Synonyms: BI-D1870
BI-D1870 is an inhibitor of S6 ribosome which can inhibit RSK1, RSK2, RSK3, RSK4 with IC50 of 31 nM, 24 nM, 18 nM and 15 nM, respectively.
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纯度 & 质量文件
批次:
靶点选择性
生物活性
靶点 RSK1
IC50:31nMRSK2
IC50:24nMRSK3
IC50:18nMRSK4
IC50:15nM- 描述
- 作用机制
- 细胞研究
- Cell Data
- 更多
实验方案
- 计算器
- 储存液制备
技术信息
| CAS号 | 501437-28-1 | 储存条件 |
|
|||||||
| 分子式 | C19H23F2N5O2 | 运输 | 蓝冰 | |||||||
| 分子量 | 391.42 | 别名 | BI-D1870 | |||||||
| 溶解度 |
|
动物实验配方 |
| Cell Lines | Concentration | Assay Type | Time | Activity Description | Data Sources |
|---|
| 22RV1 | - | Growth Inhibition Assay | - | IC50=8.61786 μM | SANGER |
| 23132-87 | - | Growth Inhibition Assay | - | IC50=14.8353 μM | SANGER |
| 5637 | - | Growth Inhibition Assay | - | IC50=4.61444 μM | SANGER |
| 639-V | - | Growth Inhibition Assay | - | IC50=2.71703 μM | SANGER |
| 647-V | - | Growth Inhibition Assay | - | IC50=11.5974 μM | SANGER |
| 697 | - | Growth Inhibition Assay | - | IC50=2.02228 μM | SANGER |
| 769-P | - | Growth Inhibition Assay | - | IC50=28.4533 μM | SANGER |
| 786-0 | - | Growth Inhibition Assay | - | IC50=8.03095 μM | SANGER |
| 8305C | - | Growth Inhibition Assay | - | IC50=3.88943 μM | SANGER |
| 8505C | - | Growth Inhibition Assay | - | IC50=4.45825 μM | SANGER |
| 8-MG-BA | - | Growth Inhibition Assay | - | IC50=2.23461 μM | SANGER |
| A101D | - | Growth Inhibition Assay | - | IC50=4.96865 μM | SANGER |
| A172 | - | Growth Inhibition Assay | - | IC50=0.51705 μM | SANGER |
| A204 | - | Growth Inhibition Assay | - | IC50=9.89755 μM | SANGER |
| A253 | - | Growth Inhibition Assay | - | IC50=14.225 μM | SANGER |
| A375 | - | Growth Inhibition Assay | - | IC50=4.05162 μM | SANGER |
| A388 | - | Growth Inhibition Assay | - | IC50=11.8808 μM | SANGER |
| A3-KAW | - | Growth Inhibition Assay | - | IC50=1.62834 μM | SANGER |
| A427 | - | Growth Inhibition Assay | - | IC50=3.10873 μM | SANGER |
| A431 | - | Growth Inhibition Assay | - | IC50=4.14081 μM | SANGER |
| A498 | - | Growth Inhibition Assay | - | IC50=38.0954 μM | SANGER |
| A549 | - | Growth Inhibition Assay | - | IC50=1.30955 μM | SANGER |
| A704 | - | Growth Inhibition Assay | - | IC50=9.47745 μM | SANGER |
| ACHN | - | Growth Inhibition Assay | - | IC50=8.22529 μM | SANGER |
| ACN | - | Growth Inhibition Assay | - | IC50=2.6679 μM | SANGER |
| AGS | - | Growth Inhibition Assay | - | IC50=2.34404 μM | SANGER |
| AN3-CA | - | Growth Inhibition Assay | - | IC50=15.6468 μM | SANGER |
| ATN-1 | - | Growth Inhibition Assay | - | IC50=4.42341 μM | SANGER |
| AU565 | - | Growth Inhibition Assay | - | IC50=22.7478 μM | SANGER |
| BALL-1 | - | Growth Inhibition Assay | - | IC50=47.8254 μM | SANGER |
| BB30-HNC | - | Growth Inhibition Assay | - | IC50=6.67444 μM | SANGER |
| BB49-HNC | - | Growth Inhibition Assay | - | IC50=11.8375 μM | SANGER |
| BB65-RCC | - | Growth Inhibition Assay | - | IC50=3.45396 μM | SANGER |
| BE-13 | - | Growth Inhibition Assay | - | IC50=1.58709 μM | SANGER |
| Becker | - | Growth Inhibition Assay | - | IC50=2.66078 μM | SANGER |
| BEN | - | Growth Inhibition Assay | - | IC50=17.5626 μM | SANGER |
| BFTC-905 | - | Growth Inhibition Assay | - | IC50=1.56332 μM | SANGER |
| BHT-101 | - | Growth Inhibition Assay | - | IC50=4.10683 μM | SANGER |
| BHY | - | Growth Inhibition Assay | - | IC50=5.5107 μM | SANGER |
| BPH-1 | - | Growth Inhibition Assay | - | IC50=2.12957 μM | SANGER |
| BT-474 | - | Growth Inhibition Assay | - | IC50=8.98872 μM | SANGER |
| BT-549 | - | Growth Inhibition Assay | - | IC50=5.07736 μM | SANGER |
| BV-173 | - | Growth Inhibition Assay | - | IC50=1.98666 μM | SANGER |
| C2BBe1 | - | Growth Inhibition Assay | - | IC50=9.86204 μM | SANGER |
| C32 | - | Growth Inhibition Assay | - | IC50=3.96581 μM | SANGER |
| C-33-A | - | Growth Inhibition Assay | - | IC50=7.4782 μM | SANGER |
| C8166 | - | Growth Inhibition Assay | - | IC50=8.86772 μM | SANGER |
| Ca9-22 | - | Growth Inhibition Assay | - | IC50=2.65933 μM | SANGER |
| CAL-120 | - | Growth Inhibition Assay | - | IC50=10.7597 μM | SANGER |
| CAL-12T | - | Growth Inhibition Assay | - | IC50=4.05795 μM | SANGER |
| CAL-27 | - | Growth Inhibition Assay | - | IC50=8.1272 μM | SANGER |
| CAL-33 | - | Growth Inhibition Assay | - | IC50=3.53362 μM | SANGER |
| CAL-39 | - | Growth Inhibition Assay | - | IC50=4.93988 μM | SANGER |
| CAL-51 | - | Growth Inhibition Assay | - | IC50=4.86843 μM | SANGER |
| CAL-54 | - | Growth Inhibition Assay | - | IC50=5.93314 μM | SANGER |
| CAL-62 | - | Growth Inhibition Assay | - | IC50=0.88152 μM | SANGER |
| CAL-72 | - | Growth Inhibition Assay | - | IC50=28.5561 μM | SANGER |
| CAL-85-1 | - | Growth Inhibition Assay | - | IC50=25.1544 μM | SANGER |
| Calu-3 | - | Growth Inhibition Assay | - | IC50=14.8743 μM | SANGER |
| Calu-6 | - | Growth Inhibition Assay | - | IC50=21.1005 μM | SANGER |
| CAMA-1 | - | Growth Inhibition Assay | - | IC50=26.4876 μM | SANGER |
| CaR-1 | - | Growth Inhibition Assay | - | IC50=5.20726 μM | SANGER |
| Ca-Ski | - | Growth Inhibition Assay | - | IC50=3.47514 μM | SANGER |
| CFPAC-1 | - | Growth Inhibition Assay | - | IC50=24.6272 μM | SANGER |
| CGTH-W-1 | - | Growth Inhibition Assay | - | IC50=3.93504 μM | SANGER |
| ChaGo-K-1 | - | Growth Inhibition Assay | - | IC50=12.7649 μM | SANGER |
| CHL-1 | - | Growth Inhibition Assay | - | IC50=1.95792 μM | SANGER |
| CHP-134 | - | Growth Inhibition Assay | - | IC50=3.48758 μM | SANGER |
| CHP-212 | - | Growth Inhibition Assay | - | IC50=8.82267 μM | SANGER |
| COLO-320-HSR | - | Growth Inhibition Assay | - | IC50=40.041 μM | SANGER |
| COLO-678 | - | Growth Inhibition Assay | - | IC50=45.7032 μM | SANGER |
| COLO-679 | - | Growth Inhibition Assay | - | IC50=15.1013 μM | SANGER |
| COLO-680N | - | Growth Inhibition Assay | - | IC50=34.1397 μM | SANGER |
| COLO-684 | - | Growth Inhibition Assay | - | IC50=18.9956 μM | SANGER |
| COLO-800 | - | Growth Inhibition Assay | - | IC50=2.54166 μM | SANGER |
| COLO-824 | - | Growth Inhibition Assay | - | IC50=4.90408 μM | SANGER |
| COLO-829 | - | Growth Inhibition Assay | - | IC50=3.66618 μM | SANGER |
| COR-L23 | - | Growth Inhibition Assay | - | IC50=4.74256 μM | SANGER |
| COR-L88 | - | Growth Inhibition Assay | - | IC50=6.79791 μM | SANGER |
| CP50-MEL-B | - | Growth Inhibition Assay | - | IC50=41.0797 μM | SANGER |
| CP66-MEL | - | Growth Inhibition Assay | - | IC50=17.301 μM | SANGER |
| CTB-1 | - | Growth Inhibition Assay | - | IC50=1.44679 μM | SANGER |
| CTV-1 | - | Growth Inhibition Assay | - | IC50=0.47872 μM | SANGER |
| CW-2 | - | Growth Inhibition Assay | - | IC50=15.0223 μM | SANGER |
| D-247MG | - | Growth Inhibition Assay | - | IC50=15.8533 μM | SANGER |
| D-283MED | - | Growth Inhibition Assay | - | IC50=2.23695 μM | SANGER |
| D-336MG | - | Growth Inhibition Assay | - | IC50=43.1152 μM | SANGER |
| D-392MG | - | Growth Inhibition Assay | - | IC50=14.1211 μM | SANGER |
| D-423MG | - | Growth Inhibition Assay | - | IC50=4.80803 μM | SANGER |
| D-502MG | - | Growth Inhibition Assay | - | IC50=3.07019 μM | SANGER |
| D-542MG | - | Growth Inhibition Assay | - | IC50=6.7309 μM | SANGER |
| D-566MG | - | Growth Inhibition Assay | - | IC50=2.91295 μM | SANGER |
| Daoy | - | Growth Inhibition Assay | - | IC50=0.98767 μM | SANGER |
| DB | - | Growth Inhibition Assay | - | IC50=2.55013 μM | SANGER |
| DBTRG-05MG | - | Growth Inhibition Assay | - | IC50=44.6996 μM | SANGER |
| DEL | - | Growth Inhibition Assay | - | IC50=5.39023 μM | SANGER |
| Detroit562 | - | Growth Inhibition Assay | - | IC50=6.85991 μM | SANGER |
| DJM-1 | - | Growth Inhibition Assay | - | IC50=4.79729 μM | SANGER |
| DMS-114 | - | Growth Inhibition Assay | - | IC50=4.81386 μM | SANGER |
| DMS-273 | - | Growth Inhibition Assay | - | IC50=8.89623 μM | SANGER |
| DOK | - | Growth Inhibition Assay | - | IC50=3.76526 μM | SANGER |
| DoTc2-4510 | - | Growth Inhibition Assay | - | IC50=24.7575 μM | SANGER |
| DSH1 | - | Growth Inhibition Assay | - | IC50=21.3879 μM | SANGER |
| DU-145 | - | Growth Inhibition Assay | - | IC50=2.11056 μM | SANGER |
| DU-4475 | - | Growth Inhibition Assay | - | IC50=0.50417 μM | SANGER |
| ECC10 | - | Growth Inhibition Assay | - | IC50=0.70094 μM | SANGER |
| EFM-19 | - | Growth Inhibition Assay | - | IC50=12.7717 μM | SANGER |
| EFO-27 | - | Growth Inhibition Assay | - | IC50=5.06329 μM | SANGER |
| EGI-1 | - | Growth Inhibition Assay | - | IC50=47.1833 μM | SANGER |
| EM-2 | - | Growth Inhibition Assay | - | IC50=2.92193 μM | SANGER |
| EoL-1-cell | - | Growth Inhibition Assay | - | IC50=1.01878 μM | SANGER |
| EPLC-272H | - | Growth Inhibition Assay | - | IC50=4.17596 μM | SANGER |
| ES1 | - | Growth Inhibition Assay | - | IC50=5.0013 μM | SANGER |
| ES3 | - | Growth Inhibition Assay | - | IC50=9.05156 μM | SANGER |
| ES4 | - | Growth Inhibition Assay | - | IC50=1.85143 μM | SANGER |
| ES5 | - | Growth Inhibition Assay | - | IC50=2.23633 μM | SANGER |
| ES7 | - | Growth Inhibition Assay | - | IC50=0.91607 μM | SANGER |
| ES8 | - | Growth Inhibition Assay | - | IC50=1.87724 μM | SANGER |
| ETK-1 | - | Growth Inhibition Assay | - | IC50=4.36203 μM | SANGER |
| EW-1 | - | Growth Inhibition Assay | - | IC50=2.75328 μM | SANGER |
| EW-11 | - | Growth Inhibition Assay | - | IC50=3.41224 μM | SANGER |
| EW-16 | - | Growth Inhibition Assay | - | IC50=24.0926 μM | SANGER |
| EW-18 | - | Growth Inhibition Assay | - | IC50=0.62211 μM | SANGER |
| EW-22 | - | Growth Inhibition Assay | - | IC50=8.91382 μM | SANGER |
| EW-3 | - | Growth Inhibition Assay | - | IC50=0.0358 μM | SANGER |
| FADU | - | Growth Inhibition Assay | - | IC50=8.17543 μM | SANGER |
| FTC-133 | - | Growth Inhibition Assay | - | IC50=6.46551 μM | SANGER |
| G-361 | - | Growth Inhibition Assay | - | IC50=2.1221 μM | SANGER |
| G-401 | - | Growth Inhibition Assay | - | IC50=9.90449 μM | SANGER |
| G-402 | - | Growth Inhibition Assay | - | IC50=16.8565 μM | SANGER |
| GAMG | - | Growth Inhibition Assay | - | IC50=0.74717 μM | SANGER |
| GB-1 | - | Growth Inhibition Assay | - | IC50=6.02068 μM | SANGER |
| GCIY | - | Growth Inhibition Assay | - | IC50=4.71015 μM | SANGER |
| GCT | - | Growth Inhibition Assay | - | IC50=2.31358 μM | SANGER |
| GI-1 | - | Growth Inhibition Assay | - | IC50=3.15255 μM | SANGER |
| GI-ME-N | - | Growth Inhibition Assay | - | IC50=7.29158 μM | SANGER |
| GMS-10 | - | Growth Inhibition Assay | - | IC50=3.09388 μM | SANGER |
| GOTO | - | Growth Inhibition Assay | - | IC50=3.28004 μM | SANGER |
| GP5d | - | Growth Inhibition Assay | - | IC50=16.1171 μM | SANGER |
| GR-ST | - | Growth Inhibition Assay | - | IC50=11.298 μM | SANGER |
| GT3TKB | - | Growth Inhibition Assay | - | IC50=3.75604 μM | SANGER |
| H4 | - | Growth Inhibition Assay | - | IC50=2.48393 μM | SANGER |
| H9 | - | Growth Inhibition Assay | - | IC50=0.06019 μM | SANGER |
| HAL-01 | - | Growth Inhibition Assay | - | IC50=22.0418 μM | SANGER |
| HCC1187 | - | Growth Inhibition Assay | - | IC50=16.6557 μM | SANGER |
| HCC1395 | - | Growth Inhibition Assay | - | IC50=48.992 μM | SANGER |
| HCC1806 | - | Growth Inhibition Assay | - | IC50=11.6134 μM | SANGER |
| HCC1954 | - | Growth Inhibition Assay | - | IC50=4.25746 μM | SANGER |
| HCC38 | - | Growth Inhibition Assay | - | IC50=17.7698 μM | SANGER |
| HCC70 | - | Growth Inhibition Assay | - | IC50=24.1323 μM | SANGER |
| HCE-4 | - | Growth Inhibition Assay | - | IC50=12.2699 μM | SANGER |
| HCT-116 | - | Growth Inhibition Assay | - | IC50=39.058 μM | SANGER |
| HD-MY-Z | - | Growth Inhibition Assay | - | IC50=3.36542 μM | SANGER |
| HEC-1 | - | Growth Inhibition Assay | - | IC50=7.25387 μM | SANGER |
| HEL | - | Growth Inhibition Assay | - | IC50=2.70254 μM | SANGER |
| HGC-27 | - | Growth Inhibition Assay | - | IC50=6.35786 μM | SANGER |
| HH | - | Growth Inhibition Assay | - | IC50=2.80001 μM | SANGER |
| HL-60 | - | Growth Inhibition Assay | - | IC50=0.88362 μM | SANGER |
| HLE | - | Growth Inhibition Assay | - | IC50=5.11734 μM | SANGER |
| HMV-II | - | Growth Inhibition Assay | - | IC50=2.16633 μM | SANGER |
| HN | - | Growth Inhibition Assay | - | IC50=1.61368 μM | SANGER |
| HO-1-N-1 | - | Growth Inhibition Assay | - | IC50=3.79801 μM | SANGER |
| HOP-62 | - | Growth Inhibition Assay | - | IC50=4.30856 μM | SANGER |
| HOP-92 | - | Growth Inhibition Assay | - | IC50=13.7997 μM | SANGER |
| HOS | - | Growth Inhibition Assay | - | IC50=4.46453 μM | SANGER |
| HPAF-II | - | Growth Inhibition Assay | - | IC50=11.8356 μM | SANGER |
| Hs-578-T | - | Growth Inhibition Assay | - | IC50=5.83607 μM | SANGER |
| HSC-2 | - | Growth Inhibition Assay | - | IC50=6.12353 μM | SANGER |
| HSC-3 | - | Growth Inhibition Assay | - | IC50=0.81769 μM | SANGER |
| HT | - | Growth Inhibition Assay | - | IC50=17.1964 μM | SANGER |
| HT-1080 | - | Growth Inhibition Assay | - | IC50=6.54042 μM | SANGER |
| HT-1376 | - | Growth Inhibition Assay | - | IC50=4.23059 μM | SANGER |
| HT-144 | - | Growth Inhibition Assay | - | IC50=5.86832 μM | SANGER |
| HT-3 | - | Growth Inhibition Assay | - | IC50=2.51024 μM | SANGER |
| HT55 | - | Growth Inhibition Assay | - | IC50=16.8751 μM | SANGER |
| HTC-C3 | - | Growth Inhibition Assay | - | IC50=5.77644 μM | SANGER |
| HuCCT1 | - | Growth Inhibition Assay | - | IC50=9.47406 μM | SANGER |
| HuH-7 | - | Growth Inhibition Assay | - | IC50=8.73012 μM | SANGER |
| HuO-3N1 | - | Growth Inhibition Assay | - | IC50=16.2473 μM | SANGER |
| HuO9 | - | Growth Inhibition Assay | - | IC50=2.36824 μM | SANGER |
| HuP-T4 | - | Growth Inhibition Assay | - | IC50=31.4837 μM | SANGER |
| HUTU-80 | - | Growth Inhibition Assay | - | IC50=3.66621 μM | SANGER |
| IA-LM | - | Growth Inhibition Assay | - | IC50=11.3486 μM | SANGER |
| IGR-1 | - | Growth Inhibition Assay | - | IC50=4.10274 μM | SANGER |
| IGROV-1 | - | Growth Inhibition Assay | - | IC50=6.92583 μM | SANGER |
| IST-MEL1 | - | Growth Inhibition Assay | - | IC50=26.7177 μM | SANGER |
| IST-MES1 | - | Growth Inhibition Assay | - | IC50=40.7653 μM | SANGER |
| IST-SL1 | - | Growth Inhibition Assay | - | IC50=0.84574 μM | SANGER |
| JEG-3 | - | Growth Inhibition Assay | - | IC50=3.6919 μM | SANGER |
| J-RT3-T3-5 | - | Growth Inhibition Assay | - | IC50=5.80794 μM | SANGER |
| JVM-2 | - | Growth Inhibition Assay | - | IC50=25.2122 μM | SANGER |
| JVM-3 | - | Growth Inhibition Assay | - | IC50=3.06756 μM | SANGER |
| K5 | - | Growth Inhibition Assay | - | IC50=7.8742 μM | SANGER |
| KALS-1 | - | Growth Inhibition Assay | - | IC50=13.095 μM | SANGER |
| KARPAS-299 | - | Growth Inhibition Assay | - | IC50=27.4701 μM | SANGER |
| KARPAS-45 | - | Growth Inhibition Assay | - | IC50=0.16525 μM | SANGER |
| KE-37 | - | Growth Inhibition Assay | - | IC50=1.59478 μM | SANGER |
| KG-1 | - | Growth Inhibition Assay | - | IC50=3.61106 μM | SANGER |
| KGN | - | Growth Inhibition Assay | - | IC50=11.8589 μM | SANGER |
| KINGS-1 | - | Growth Inhibition Assay | - | IC50=9.6937 μM | SANGER |
| KM12 | - | Growth Inhibition Assay | - | IC50=3.12273 μM | SANGER |
| KM-H2 | - | Growth Inhibition Assay | - | IC50=33.1699 μM | SANGER |
| KNS-42 | - | Growth Inhibition Assay | - | IC50=5.2616 μM | SANGER |
| KNS-62 | - | Growth Inhibition Assay | - | IC50=25.018 μM | SANGER |
| KNS-81-FD | - | Growth Inhibition Assay | - | IC50=5.50092 μM | SANGER |
| KOSC-2 | - | Growth Inhibition Assay | - | IC50=1.13385 μM | SANGER |
| KP-N-YN | - | Growth Inhibition Assay | - | IC50=5.0567 μM | SANGER |
| KP-N-YS | - | Growth Inhibition Assay | - | IC50=0.68223 μM | SANGER |
| KS-1 | - | Growth Inhibition Assay | - | IC50=6.52147 μM | SANGER |
| KU-19-19 | - | Growth Inhibition Assay | - | IC50=3.60304 μM | SANGER |
| KU812 | - | Growth Inhibition Assay | - | IC50=0.62623 μM | SANGER |
| KURAMOCHI | - | Growth Inhibition Assay | - | IC50=34.6425 μM | SANGER |
| KY821 | - | Growth Inhibition Assay | - | IC50=0.88812 μM | SANGER |
| KYSE-140 | - | Growth Inhibition Assay | - | IC50=21.7271 μM | SANGER |
| KYSE-150 | - | Growth Inhibition Assay | - | IC50=2.15234 μM | SANGER |
| KYSE-270 | - | Growth Inhibition Assay | - | IC50=5.53536 μM | SANGER |
| KYSE-410 | - | Growth Inhibition Assay | - | IC50=10.0615 μM | SANGER |
| KYSE-450 | - | Growth Inhibition Assay | - | IC50=7.63791 μM | SANGER |
| KYSE-510 | - | Growth Inhibition Assay | - | IC50=4.2609 μM | SANGER |
| KYSE-520 | - | Growth Inhibition Assay | - | IC50=7.2929 μM | SANGER |
| KYSE-70 | - | Growth Inhibition Assay | - | IC50=47.7222 μM | SANGER |
| L-363 | - | Growth Inhibition Assay | - | IC50=5.69476 μM | SANGER |
| LAMA-84 | - | Growth Inhibition Assay | - | IC50=1.12794 μM | SANGER |
| LAN-6 | - | Growth Inhibition Assay | - | IC50=17.8485 μM | SANGER |
| LB1047-RCC | - | Growth Inhibition Assay | - | IC50=4.10441 μM | SANGER |
| LB2241-RCC | - | Growth Inhibition Assay | - | IC50=3.68625 μM | SANGER |
| LB831-BLC | - | Growth Inhibition Assay | - | IC50=3.54016 μM | SANGER |
| LC-2-ad | - | Growth Inhibition Assay | - | IC50=6.86292 μM | SANGER |
| LCLC-103H | - | Growth Inhibition Assay | - | IC50=18.051 μM | SANGER |
| LCLC-97TM1 | - | Growth Inhibition Assay | - | IC50=2.60028 μM | SANGER |
| LK-2 | - | Growth Inhibition Assay | - | IC50=18.7723 μM | SANGER |
| LN-405 | - | Growth Inhibition Assay | - | IC50=11.5927 μM | SANGER |
| LNCaP-Clone-FGC | - | Growth Inhibition Assay | - | IC50=3.70041 μM | SANGER |
| LoVo | - | Growth Inhibition Assay | - | IC50=1.46755 μM | SANGER |
| LOXIMVI | - | Growth Inhibition Assay | - | IC50=2.04434 μM | SANGER |
| LS-123 | - | Growth Inhibition Assay | - | IC50=20.0194 μM | SANGER |
| LS-411N | - | Growth Inhibition Assay | - | IC50=22.2869 μM | SANGER |
| LU-134-A | - | Growth Inhibition Assay | - | IC50=3.95422 μM | SANGER |
| LU-135 | - | Growth Inhibition Assay | - | IC50=33.7086 μM | SANGER |
| LU-139 | - | Growth Inhibition Assay | - | IC50=0.84958 μM | SANGER |
| LU-65 | - | Growth Inhibition Assay | - | IC50=18.4043 μM | SANGER |
| LXF-289 | - | Growth Inhibition Assay | - | IC50=4.40202 μM | SANGER |
| M059J | - | Growth Inhibition Assay | - | IC50=3.71468 μM | SANGER |
| M14 | - | Growth Inhibition Assay | - | IC50=5.86726 μM | SANGER |
| MC116 | - | Growth Inhibition Assay | - | IC50=19.5331 μM | SANGER |
| MC-IXC | - | Growth Inhibition Assay | - | IC50=0.79589 μM | SANGER |
| MDA-MB-157 | - | Growth Inhibition Assay | - | IC50=4.30656 μM | SANGER |
| MDA-MB-175-VII | - | Growth Inhibition Assay | - | IC50=6.6209 μM | SANGER |
| MDA-MB-231 | - | Growth Inhibition Assay | - | IC50=4.72115 μM | SANGER |
| MDA-MB-361 | - | Growth Inhibition Assay | - | IC50=48.046 μM | SANGER |
| MDA-MB-415 | - | Growth Inhibition Assay | - | IC50=13.1609 μM | SANGER |
| ME-180 | - | Growth Inhibition Assay | - | IC50=2.77736 μM | SANGER |
| MEG-01 | - | Growth Inhibition Assay | - | IC50=5.36274 μM | SANGER |
| MEL-HO | - | Growth Inhibition Assay | - | IC50=9.402 μM | SANGER |
| MEL-JUSO | - | Growth Inhibition Assay | - | IC50=8.68675 μM | SANGER |
| MFM-223 | - | Growth Inhibition Assay | - | IC50=8.80735 μM | SANGER |
| MHH-ES-1 | - | Growth Inhibition Assay | - | IC50=4.82504 μM | SANGER |
| MHH-NB-11 | - | Growth Inhibition Assay | - | IC50=26.5851 μM | SANGER |
| MHH-PREB-1 | - | Growth Inhibition Assay | - | IC50=4.39773 μM | SANGER |
| MIA-PaCa-2 | - | Growth Inhibition Assay | - | IC50=4.36227 μM | SANGER |
| MKN1 | - | Growth Inhibition Assay | - | IC50=3.20875 μM | SANGER |
| MKN7 | - | Growth Inhibition Assay | - | IC50=22.687 μM | SANGER |
| ML-2 | - | Growth Inhibition Assay | - | IC50=0.85575 μM | SANGER |
| MLMA | - | Growth Inhibition Assay | - | IC50=5.23436 μM | SANGER |
| MN-60 | - | Growth Inhibition Assay | - | IC50=2.44883 μM | SANGER |
| MOLT-13 | - | Growth Inhibition Assay | - | IC50=3.96856 μM | SANGER |
| MOLT-16 | - | Growth Inhibition Assay | - | IC50=9.16655 μM | SANGER |
| MOLT-4 | - | Growth Inhibition Assay | - | IC50=3.39098 μM | SANGER |
| Mo-T | - | Growth Inhibition Assay | - | IC50=33.8593 μM | SANGER |
| MPP-89 | - | Growth Inhibition Assay | - | IC50=8.91341 μM | SANGER |
| MS-1 | - | Growth Inhibition Assay | - | IC50=19.6103 μM | SANGER |
| MV-4-11 | - | Growth Inhibition Assay | - | IC50=0.97897 μM | SANGER |
| MZ1-PC | - | Growth Inhibition Assay | - | IC50=3.82883 μM | SANGER |
| MZ2-MEL | - | Growth Inhibition Assay | - | IC50=10.662 μM | SANGER |
| NB10 | - | Growth Inhibition Assay | - | IC50=1.7763 μM | SANGER |
| NB12 | - | Growth Inhibition Assay | - | IC50=9.34081 μM | SANGER |
| NB14 | - | Growth Inhibition Assay | - | IC50=2.11321 μM | SANGER |
| NB17 | - | Growth Inhibition Assay | - | IC50=9.14535 μM | SANGER |
| NB5 | - | Growth Inhibition Assay | - | IC50=10.5405 μM | SANGER |
| NB6 | - | Growth Inhibition Assay | - | IC50=2.45779 μM | SANGER |
| NB69 | - | Growth Inhibition Assay | - | IC50=12.7585 μM | SANGER |
| NB7 | - | Growth Inhibition Assay | - | IC50=19.1753 μM | SANGER |
| NBsusSR | - | Growth Inhibition Assay | - | IC50=1.82961 μM | SANGER |
| NCI-H1048 | - | Growth Inhibition Assay | - | IC50=2.68321 μM | SANGER |
| NCI-H1092 | - | Growth Inhibition Assay | - | IC50=16.6297 μM | SANGER |
| NCI-H1155 | - | Growth Inhibition Assay | - | IC50=14.2747 μM | SANGER |
| NCI-H1299 | - | Growth Inhibition Assay | - | IC50=2.93736 μM | SANGER |
| NCI-H1304 | - | Growth Inhibition Assay | - | IC50=33.6036 μM | SANGER |
| NCI-H1395 | - | Growth Inhibition Assay | - | IC50=2.47121 μM | SANGER |
| NCI-H1437 | - | Growth Inhibition Assay | - | IC50=4.9293 μM | SANGER |
| NCI-H1573 | - | Growth Inhibition Assay | - | IC50=48.6785 μM | SANGER |
| NCI-H1581 | - | Growth Inhibition Assay | - | IC50=12.2819 μM | SANGER |
| NCI-H1648 | - | Growth Inhibition Assay | - | IC50=11.4629 μM | SANGER |
| NCI-H1651 | - | Growth Inhibition Assay | - | IC50=29.8503 μM | SANGER |
| NCI-H1703 | - | Growth Inhibition Assay | - | IC50=20.8173 μM | SANGER |
| NCI-H1755 | - | Growth Inhibition Assay | - | IC50=33.811 μM | SANGER |
| NCI-H1770 | - | Growth Inhibition Assay | - | IC50=17.9491 μM | SANGER |
| NCI-H1792 | - | Growth Inhibition Assay | - | IC50=2.73738 μM | SANGER |
| NCI-H1838 | - | Growth Inhibition Assay | - | IC50=48.3458 μM | SANGER |
| NCI-H2009 | - | Growth Inhibition Assay | - | IC50=16.9266 μM | SANGER |
| NCI-H2029 | - | Growth Inhibition Assay | - | IC50=1.97241 μM | SANGER |
| NCI-H2052 | - | Growth Inhibition Assay | - | IC50=13.3848 μM | SANGER |
| NCI-H2087 | - | Growth Inhibition Assay | - | IC50=8.36158 μM | SANGER |
| NCI-H209 | - | Growth Inhibition Assay | - | IC50=0.7682 μM | SANGER |
| NCI-H2122 | - | Growth Inhibition Assay | - | IC50=8.40479 μM | SANGER |
| NCI-H2228 | - | Growth Inhibition Assay | - | IC50=11.4928 μM | SANGER |
| NCI-H2291 | - | Growth Inhibition Assay | - | IC50=49.5988 μM | SANGER |
| NCI-H23 | - | Growth Inhibition Assay | - | IC50=12.3125 μM | SANGER |
| NCI-H2342 | - | Growth Inhibition Assay | - | IC50=29.3803 μM | SANGER |
| NCI-H2347 | - | Growth Inhibition Assay | - | IC50=25.4249 μM | SANGER |
| NCI-H2405 | - | Growth Inhibition Assay | - | IC50=6.74855 μM | SANGER |
| NCI-H2452 | - | Growth Inhibition Assay | - | IC50=11.3927 μM | SANGER |
| NCI-H28 | - | Growth Inhibition Assay | - | IC50=8.85185 μM | SANGER |
| NCI-H292 | - | Growth Inhibition Assay | - | IC50=1.46069 μM | SANGER |
| NCI-H358 | - | Growth Inhibition Assay | - | IC50=19.2673 μM | SANGER |
| NCI-H446 | - | Growth Inhibition Assay | - | IC50=3.6834 μM | SANGER |
| NCI-H460 | - | Growth Inhibition Assay | - | IC50=18.8466 μM | SANGER |
| NCI-H520 | - | Growth Inhibition Assay | - | IC50=18.3281 μM | SANGER |
| NCI-H526 | - | Growth Inhibition Assay | - | IC50=37.2772 μM | SANGER |
| NCI-H596 | - | Growth Inhibition Assay | - | IC50=12.4798 μM | SANGER |
| NCI-H650 | - | Growth Inhibition Assay | - | IC50=5.57114 μM | SANGER |
| NCI-H661 | - | Growth Inhibition Assay | - | IC50=34.8448 μM | SANGER |
| NCI-H69 | - | Growth Inhibition Assay | - | IC50=2.71601 μM | SANGER |
| NCI-H720 | - | Growth Inhibition Assay | - | IC50=0.17194 μM | SANGER |
| NCI-H727 | - | Growth Inhibition Assay | - | IC50=21.3493 μM | SANGER |
| NCI-H747 | - | Growth Inhibition Assay | - | IC50=8.04457 μM | SANGER |
| NCI-H810 | - | Growth Inhibition Assay | - | IC50=3.22155 μM | SANGER |
| NCI-H82 | - | Growth Inhibition Assay | - | IC50=19.6878 μM | SANGER |
| NCI-SNU-1 | - | Growth Inhibition Assay | - | IC50=6.79022 μM | SANGER |
| NCI-SNU-5 | - | Growth Inhibition Assay | - | IC50=15.5589 μM | SANGER |
| NEC8 | - | Growth Inhibition Assay | - | IC50=1.70115 μM | SANGER |
| NH-12 | - | Growth Inhibition Assay | - | IC50=3.11456 μM | SANGER |
| NKM-1 | - | Growth Inhibition Assay | - | IC50=9.83964 μM | SANGER |
| no-10 | - | Growth Inhibition Assay | - | IC50=22.5004 μM | SANGER |
| no-11 | - | Growth Inhibition Assay | - | IC50=21.1602 μM | SANGER |
| NOMO-1 | - | Growth Inhibition Assay | - | IC50=11.8597 μM | SANGER |
| NOS-1 | - | Growth Inhibition Assay | - | IC50=7.20415 μM | SANGER |
| NTERA-S-cl-D1 | - | Growth Inhibition Assay | - | IC50=10.5475 μM | SANGER |
| NUGC-3 | - | Growth Inhibition Assay | - | IC50=23.1199 μM | SANGER |
| NY | - | Growth Inhibition Assay | - | IC50=19.1567 μM | SANGER |
| OAW-42 | - | Growth Inhibition Assay | - | IC50=40.0542 μM | SANGER |
| OCI-AML2 | - | Growth Inhibition Assay | - | IC50=19.7032 μM | SANGER |
| OCUB-M | - | Growth Inhibition Assay | - | IC50=6.6077 μM | SANGER |
| OE19 | - | Growth Inhibition Assay | - | IC50=14.0075 μM | SANGER |
| OE33 | - | Growth Inhibition Assay | - | IC50=30.1342 μM | SANGER |
| OMC-1 | - | Growth Inhibition Assay | - | IC50=6.35441 μM | SANGER |
| OVCAR-3 | - | Growth Inhibition Assay | - | IC50=33.4127 μM | SANGER |
| OVCAR-4 | - | Growth Inhibition Assay | - | IC50=7.5526 μM | SANGER |
| OVCAR-5 | - | Growth Inhibition Assay | - | IC50=7.82329 μM | SANGER |
| OVCAR-8 | - | Growth Inhibition Assay | - | IC50=6.94229 μM | SANGER |
| P12-ICHIKAWA | - | Growth Inhibition Assay | - | IC50=2.52559 μM | SANGER |
| P30-OHK | - | Growth Inhibition Assay | - | IC50=25.6318 μM | SANGER |
| PANC-03-27 | - | Growth Inhibition Assay | - | IC50=4.30083 μM | SANGER |
| PANC-08-13 | - | Growth Inhibition Assay | - | IC50=18.7889 μM | SANGER |
| PC-14 | - | Growth Inhibition Assay | - | IC50=20.1834 μM | SANGER |
| PC-3 | - | Growth Inhibition Assay | - | IC50=4.94648 μM | SANGER |
| PFSK-1 | - | Growth Inhibition Assay | - | IC50=9.95669 μM | SANGER |
| PSN1 | - | Growth Inhibition Assay | - | IC50=3.05786 μM | SANGER |
| QIMR-WIL | - | Growth Inhibition Assay | - | IC50=2.07849 μM | SANGER |
| Ramos-2G6-4C10 | - | Growth Inhibition Assay | - | IC50=1.70444 μM | SANGER |
| RCC10RGB | - | Growth Inhibition Assay | - | IC50=33.9433 μM | SANGER |
| RCM-1 | - | Growth Inhibition Assay | - | IC50=8.96486 μM | SANGER |
| RD | - | Growth Inhibition Assay | - | IC50=3.43132 μM | SANGER |
| RERF-LC-MS | - | Growth Inhibition Assay | - | IC50=17.9129 μM | SANGER |
| RH-1 | - | Growth Inhibition Assay | - | IC50=21.883 μM | SANGER |
| RH-18 | - | Growth Inhibition Assay | - | IC50=50.0884 μM | SANGER |
| RKO | - | Growth Inhibition Assay | - | IC50=4.72817 μM | SANGER |
| RMG-I | - | Growth Inhibition Assay | - | IC50=42.4921 μM | SANGER |
| RPMI-2650 | - | Growth Inhibition Assay | - | IC50=19.012 μM | SANGER |
| RPMI-7951 | - | Growth Inhibition Assay | - | IC50=3.3973 μM | SANGER |
| RPMI-8226 | - | Growth Inhibition Assay | - | IC50=24.3155 μM | SANGER |
| RS4-11 | - | Growth Inhibition Assay | - | IC50=7.70196 μM | SANGER |
| RT-112 | - | Growth Inhibition Assay | - | IC50=6.79463 μM | SANGER |
| RVH-421 | - | Growth Inhibition Assay | - | IC50=8.75398 μM | SANGER |
| RXF393 | - | Growth Inhibition Assay | - | IC50=22.2789 μM | SANGER |
| S-117 | - | Growth Inhibition Assay | - | IC50=33.7286 μM | SANGER |
| Saos-2 | - | Growth Inhibition Assay | - | IC50=12.2003 μM | SANGER |
| SAS | - | Growth Inhibition Assay | - | IC50=9.58455 μM | SANGER |
| SBC-1 | - | Growth Inhibition Assay | - | IC50=0.69524 μM | SANGER |
| SCC-15 | - | Growth Inhibition Assay | - | IC50=8.87196 μM | SANGER |
| SCC-25 | - | Growth Inhibition Assay | - | IC50=5.19046 μM | SANGER |
| SCC-4 | - | Growth Inhibition Assay | - | IC50=3.09276 μM | SANGER |
| SCC-9 | - | Growth Inhibition Assay | - | IC50=6.8255 μM | SANGER |
| SCH | - | Growth Inhibition Assay | - | IC50=5.74767 μM | SANGER |
| SF126 | - | Growth Inhibition Assay | - | IC50=15.7285 μM | SANGER |
| SF268 | - | Growth Inhibition Assay | - | IC50=2.87225 μM | SANGER |
| SF539 | - | Growth Inhibition Assay | - | IC50=10.7188 μM | SANGER |
| SH-4 | - | Growth Inhibition Assay | - | IC50=16.992 μM | SANGER |
| SHP-77 | - | Growth Inhibition Assay | - | IC50=43.1828 μM | SANGER |
| SiHa | - | Growth Inhibition Assay | - | IC50=6.14097 μM | SANGER |
| SJRH30 | - | Growth Inhibition Assay | - | IC50=5.39213 μM | SANGER |
| SJSA-1 | - | Growth Inhibition Assay | - | IC50=2.6687 μM | SANGER |
| SKG-IIIa | - | Growth Inhibition Assay | - | IC50=6.56263 μM | SANGER |
| SK-HEP-1 | - | Growth Inhibition Assay | - | IC50=12.2613 μM | SANGER |
| SK-LU-1 | - | Growth Inhibition Assay | - | IC50=8.43997 μM | SANGER |
| SK-MEL-1 | - | Growth Inhibition Assay | - | IC50=40.2927 μM | SANGER |
| SK-MEL-2 | - | Growth Inhibition Assay | - | IC50=10.1588 μM | SANGER |
| SK-MEL-28 | - | Growth Inhibition Assay | - | IC50=5.20313 μM | SANGER |
| SK-MEL-3 | - | Growth Inhibition Assay | - | IC50=18.6679 μM | SANGER |
| SK-MES-1 | - | Growth Inhibition Assay | - | IC50=3.7303 μM | SANGER |
| SK-N-AS | - | Growth Inhibition Assay | - | IC50=2.29059 μM | SANGER |
| SK-N-DZ | - | Growth Inhibition Assay | - | IC50=25.0904 μM | SANGER |
| SK-NEP-1 | - | Growth Inhibition Assay | - | IC50=2.044 μM | SANGER |
| SK-N-FI | - | Growth Inhibition Assay | - | IC50=26.1162 μM | SANGER |
| SK-OV-3 | - | Growth Inhibition Assay | - | IC50=33.8854 μM | SANGER |
| SK-PN-DW | - | Growth Inhibition Assay | - | IC50=5.43589 μM | SANGER |
| SK-UT-1 | - | Growth Inhibition Assay | - | IC50=7.54829 μM | SANGER |
| SN12C | - | Growth Inhibition Assay | - | IC50=32.8815 μM | SANGER |
| SNB75 | - | Growth Inhibition Assay | - | IC50=14.3893 μM | SANGER |
| SNU-387 | - | Growth Inhibition Assay | - | IC50=6.99516 μM | SANGER |
| SNU-423 | - | Growth Inhibition Assay | - | IC50=7.29452 μM | SANGER |
| SNU-449 | - | Growth Inhibition Assay | - | IC50=8.75265 μM | SANGER |
| SNU-C2B | - | Growth Inhibition Assay | - | IC50=3.39097 μM | SANGER |
| SW1573 | - | Growth Inhibition Assay | - | IC50=6.78319 μM | SANGER |
| SW1710 | - | Growth Inhibition Assay | - | IC50=2.30661 μM | SANGER |
| SW1783 | - | Growth Inhibition Assay | - | IC50=16.9998 μM | SANGER |
| SW48 | - | Growth Inhibition Assay | - | IC50=3.43358 μM | SANGER |
| SW626 | - | Growth Inhibition Assay | - | IC50=4.89697 μM | SANGER |
| SW684 | - | Growth Inhibition Assay | - | IC50=13.1861 μM | SANGER |
| SW756 | - | Growth Inhibition Assay | - | IC50=9.55361 μM | SANGER |
| SW780 | - | Growth Inhibition Assay | - | IC50=8.18821 μM | SANGER |
| SW872 | - | Growth Inhibition Assay | - | IC50=43.2123 μM | SANGER |
| SW954 | - | Growth Inhibition Assay | - | IC50=2.8583 μM | SANGER |
| SW962 | - | Growth Inhibition Assay | - | IC50=12.8223 μM | SANGER |
| SW982 | - | Growth Inhibition Assay | - | IC50=5.13374 μM | SANGER |
| T47D | - | Growth Inhibition Assay | - | IC50=5.9612 μM | SANGER |
| T98G | - | Growth Inhibition Assay | - | IC50=3.28216 μM | SANGER |
| TCCSUP | - | Growth Inhibition Assay | - | IC50=5.71778 μM | SANGER |
| TE-1 | - | Growth Inhibition Assay | - | IC50=5.03666 μM | SANGER |
| TE-10 | - | Growth Inhibition Assay | - | IC50=5.44893 μM | SANGER |
| TE-11 | - | Growth Inhibition Assay | - | IC50=27.7342 μM | SANGER |
| TE-5 | - | Growth Inhibition Assay | - | IC50=33.1368 μM | SANGER |
| TE-6 | - | Growth Inhibition Assay | - | IC50=8.23788 μM | SANGER |
| TE-8 | - | Growth Inhibition Assay | - | IC50=3.19231 μM | SANGER |
| TE-9 | - | Growth Inhibition Assay | - | IC50=2.17376 μM | SANGER |
| TGBC11TKB | - | Growth Inhibition Assay | - | IC50=9.19205 μM | SANGER |
| TGBC1TKB | - | Growth Inhibition Assay | - | IC50=7.15277 μM | SANGER |
| TGW | - | Growth Inhibition Assay | - | IC50=1.05124 μM | SANGER |
| TI-73 | - | Growth Inhibition Assay | - | IC50=9.03496 μM | SANGER |
| TK10 | - | Growth Inhibition Assay | - | IC50=5.36086 μM | SANGER |
| TYK-nu | - | Growth Inhibition Assay | - | IC50=3.53676 μM | SANGER |
| U-118-MG | - | Growth Inhibition Assay | - | IC50=32.5441 μM | SANGER |
| U251 | - | Growth Inhibition Assay | - | IC50=2.73032 μM | SANGER |
| U-266 | - | Growth Inhibition Assay | - | IC50=4.61032 μM | SANGER |
| U-87-MG | - | Growth Inhibition Assay | - | IC50=6.83826 μM | SANGER |
| UACC-62 | - | Growth Inhibition Assay | - | IC50=15.966 μM | SANGER |
| UM-UC-3 | - | Growth Inhibition Assay | - | IC50=8.7139 μM | SANGER |
| VM-CUB-1 | - | Growth Inhibition Assay | - | IC50=5.23439 μM | SANGER |
| VMRC-RCZ | - | Growth Inhibition Assay | - | IC50=39.0054 μM | SANGER |
| YAPC | - | Growth Inhibition Assay | - | IC50=35.9533 μM | SANGER |
| YH-13 | - | Growth Inhibition Assay | - | IC50=11.4742 μM | SANGER |
| YKG-1 | - | Growth Inhibition Assay | - | IC50=1.98432 μM | SANGER |
| 靶点 | Description | IC50 |
|---|---|---|
| RSK1 | IC50:31nM | |
| RSK2 | IC50:24nM | |
| RSK3 | IC50:18nM | |
| RSK4 | IC50:15nM |
