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CAS No.: 1009583-20-3
Synonyms: Bms-816336
BMS-816336, a hydroxyl-substituted adamantyl acetamide, has been identified as a potent inhibitor against human 11β-hydroxysteroid dehydrogenase type 1(11β-HSD1) enzyme (IC50 3.0 nM) with > 10000 fold selectivity over human 11β-hydroxysteroid dehydrogenase type 2(11β-HSD2).
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT00979368 | Diabetes Mellitus, Non-Insulin... more >>-Dependent Dyslipidemia Collapse << | Phase 1 | Completed | - | Australia, Victoria ... more >> Local Institution Melbourne, Victoria, Australia, 3004 Collapse << |
实验方案
技术信息
CAS号 | 1009583-20-3 | 储存条件 |
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分子式 | C21H27NO3 | 运输 | 蓝冰 | |
分子量 | 341.44 | 别名 | Bms-816336 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT00979368 | Diabetes Mellitus, Non-Insulin... more >>-Dependent Dyslipidemia Collapse << | Phase 1 | Completed | - | Australia, Victoria ... more >> Local Institution Melbourne, Victoria, Australia, 3004 Collapse << |
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