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CAS No.: 1271022-90-2
Synonyms: BMS-911543
BMS-911543 is a selective ATP-competitive JAK2 inhibitor with IC50 value of 1.1 nM, with much less potency against JAK1, JAK3 and TYK2 with IC50 values of 360nM, 75 nM and 66nM.
规格 | 价格 | 促销价格 | 库存 | 数量 |
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生物活性
动物研究 | ||||||||||||||||||||||||||||||||||||
剂量 | Mice: 3 mg/kg - 30 mg/kg[3] (p.o.); 2 mg/kg[1] (i.v.) Rat: 1 mg/kg[1] (i.v./p.o.) | |||||||||||||||||||||||||||||||||||
给药途径 | p.o., i.v. | |||||||||||||||||||||||||||||||||||
动物药代数据 |
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NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT01236352 | Cancer | Phase 1 Phase 2 | Completed | - | United States, Minnesota ... more >> Mayo Clinic Rochester, Minnesota, United States, 55905 United States, New York The Mount Sinai School Of Medicine New York, New York, United States, 10029 United States, Texas The University Of Texas Md Anderson Cancer Center Houston, Texas, United States, 77030 Australia, Victoria Local Institution East Melbourne, Victoria, Australia, 3002 Local Institution Melbourne, Victoria, Australia, 3050 Collapse << |
实验方案
技术信息
CAS号 | 1271022-90-2 | 储存条件 |
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分子式 | C23H28N8O | 运输 | 蓝冰 | |||||
分子量 | 432.52 | 别名 | BMS-911543 | |||||
溶解度 |
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动物实验配方 |