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CAS No.: 136553-81-6
Synonyms: Cyclo(D-Trp-D-Asp-Pro-D-Val-Leu)
BQ-123 is a specific antagonist of endothelin A receptor (ETA) and the IC50 is 7.3 nM.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT00001624 | Hyperinsulinemia | Phase 1 | Completed | - | United States, Maryland ... more >> National Heart, Lung and Blood Institute (NHLBI) Bethesda, Maryland, United States, 20892 Collapse << |
NCT03038750 | - | - | Recruiting | July 2022 | United Kingdom ... more >> Department of Public Health and Primary Care Recruiting Cambridge, United Kingdom, CB1 8RN Contact: Dirk Paul, PhD 01223 761918 dsp35@medschl.cam.ac.uk Principal Investigator: Dirk Paul, PhD Collapse << |
NCT02966665 | Chronic Obstructive Pulmonary ... more >>Disease Pulmonary Artery Hypertension Heart Failure Hypertension Collapse << | Phase 1 | Recruiting | August 2020 | United States, Utah ... more >> George E Wahlen VA Medical Center Recruiting Salt Lake City, Utah, United States, 84132 Contact: Russell Richardson, Ph.D. 801-582-1565 r.richardson@hsc.utah.edu Contact: Ashley Nelson, MD 801-582-1565 ext 4127 ash.nelson@hsc.utah.edu Collapse << |
实验方案
技术信息
CAS号 | 136553-81-6 | 储存条件 |
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分子式 | C31H42N6O7 | 运输 | 蓝冰 | |||||
分子量 | 610.70 | 别名 | Cyclo(D-Trp-D-Asp-Pro-D-Val-Leu) | |||||
溶解度 |
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动物实验配方 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT00001624 | Hyperinsulinemia | Phase 1 | Completed | - | United States, Maryland ... more >> National Heart, Lung and Blood Institute (NHLBI) Bethesda, Maryland, United States, 20892 Collapse << |
NCT03038750 | - | - | Recruiting | July 2022 | United Kingdom ... more >> Department of Public Health and Primary Care Recruiting Cambridge, United Kingdom, CB1 8RN Contact: Dirk Paul, PhD 01223 761918 dsp35@medschl.cam.ac.uk Principal Investigator: Dirk Paul, PhD Collapse << |
NCT02966665 | Chronic Obstructive Pulmonary ... more >>Disease Pulmonary Artery Hypertension Heart Failure Hypertension Collapse << | Phase 1 | Recruiting | August 2020 | United States, Utah ... more >> George E Wahlen VA Medical Center Recruiting Salt Lake City, Utah, United States, 84132 Contact: Russell Richardson, Ph.D. 801-582-1565 r.richardson@hsc.utah.edu Contact: Ashley Nelson, MD 801-582-1565 ext 4127 ash.nelson@hsc.utah.edu Collapse << |
NCT00006071 | - | - | Completed | - | United States, Maryland ... more >> National Heart, Lung and Blood Institute (NHLBI) Bethesda, Maryland, United States, 20892 Collapse << |
NCT03679780 | Cardiovascular Diseases ... more >> Cardiovascular Risk Factor Vasoconstriction Collapse << | Phase 1 | Not yet recruiting | October 1, 2019 | United States, Texas ... more >> Engineering Research Building Not yet recruiting Arlington, Texas, United States, 76019 Contact: R. Matthew Brothers, PhD 8172723156 matthew.brothers@uta.edu Contact: John D Akins, MS 8172721835 john.akins@uta.edu Collapse << |
NCT00722215 | Chronic Kidney Disease ... more >> Proteinuria Collapse << | Phase 1 | Completed | - | United Kingdom ... more >> Clinical Research Centre, Western General Hospital Edinburgh, Scotland, United Kingdom, EH4 2XU Collapse << |
NCT00427232 | Coronary Vessels ... more >> Endothelins Vascular Resistance Collapse << | Phase 1 | Completed | - | Austria ... more >> Dept. of Internal Medicine II, Medical University of Vienna Vienna, Austria, A-1090 Collapse << |
NCT02987465 | - | - | Completed | - | United Kingdom ... more >> Addenbrooke's Hospital Cambridge, Cambridgeshire, United Kingdom, CB2 0QQ Collapse << |
NCT01395329 | Prehypertension ... more >> Hypertension Collapse << | Phase 4 | Completed | - | United States, Colorado ... more >> UC-Boulder Clinical and Translational Research Center Boulder, Colorado, United States, 80309 Collapse << |
NCT01395329 | - | - | Completed | - | - |
NCT00001527 | - | - | Completed | - | United States, Maryland ... more >> National Heart, Lung and Blood Institute (NHLBI) Bethesda, Maryland, United States, 20892 Collapse << |
NCT00115583 | Atherosclerosis, Coronary | Not Applicable | Completed | - | United States, Massachusetts ... more >> Brigham and Womens Hospital Boston, Massachusetts, United States, 02115 Collapse << |
NCT01119417 | Hypertension ... more >>Pure Autonomic Failure Multiple System Atrophy Collapse << | Phase 1 | Enrolling by invitation | December 2020 | United States, Tennessee ... more >> Vanderbilt University Nashville, Tennessee, United States, 37232 Collapse << |
NCT02062346 | Vasculitis | Not Applicable | Recruiting | August 2020 | United Kingdom ... more >> University of Edinburgh Recruiting Edinburgh, Midlothian, United Kingdom, EH16 4TJ University of Edinburgh Recruiting Edinburgh, United Kingdom Contact: Neeraj Dhaun Collapse << |
NCT02086253 | Healthy Conditions | Not Applicable | Completed | - | France ... more >> CHU - Hôpitaux de Rouen Rouen, Normandy, France, 76031 Collapse << |
NCT00745693 | Coronary Disease | Not Applicable | Completed | - | Sweden ... more >> Umeå University Umeå, Västerbottens, Sweden, SE-901 87 Collapse << |
NCT02124824 | Heart Failure | Early Phase 1 | Recruiting | September 1, 2019 | United States, Utah ... more >> VA Salt Lake City Health Care System, Salt Lake City, UT Recruiting Salt Lake City, Utah, United States, 84148 Contact: David W Wray, PhD 801-582-1565 ext 4162 walter.wray@hsc.utah.edu Contact: Douglas S Capps, BS (801) 582-1565 ext 4414 scott.capps@hsc.utah.edu Principal Investigator: David W. Wray, PhD Collapse << |
NCT00759408 | Pulmonary Hypertension | Phase 2 | Completed | - | United States, Massachusetts ... more >> Brigham and Women's Hospital Boston, Massachusetts, United States, 02115 Collapse << |
NCT00915070 | Healthy | Not Applicable | Completed | - | Austria ... more >> Department of Clinical Pharmacology, Medical University of Vienna Vienna, Austria, 1090 Collapse << |
NCT01658410 | Coronary Artery Disease ... more >> Aorto-coronary Bypass Grafting Collapse << | Phase 2 | Unknown | December 2016 | Austria ... more >> Medical University of Vienna Vienna, Austria, 1090 Collapse << |
NCT00759408 | - | - | Completed | - | - |
NCT00586820 | Myocardial Reperfusion Injury | Phase 2 | Completed | - | United States, Minnesota ... more >> Mayo Clinic Rochester, Minnesota, United States, 55905 Collapse << |
NCT00502528 | ST-Elevation Myocardial Infarc... more >>tion Collapse << | Phase 2 | Completed | - | Austria ... more >> Medical University of Vienna Vienna, Vienna-Austria, Austria, 1090 Collapse << |
NCT00586820 | - | - | Completed | - | - |
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