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CAS No.: 1338806-73-7

CFI-400945 Catalog No. CSN15736

Synonyms: CFI-400945 Free Base

CFI400945 is a potent and selective,orally bioavailable PLK4 inhibitor with an IC50 value of 2.8 ±1.4 nM have potential antineoplastic activity.

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靶点选择性

生物活性

  • 描述
  • 细胞研究
  • Cell Data
  • 更多
  • 临床研究
  • NCT号适应症或疾病临床期招募状态预计完成时间地点
    NCT03624543Breast CancerPhase 2Not yet recruitingDecember 31, 2020-
    NCT01954316Advanced CancerPhase 1RecruitingSeptember 2018United States, California ... more >> UCLA Medical Center Recruiting Santa Monica, California, United States, 90404 Contact: Lisa Yonemoto    310-582-4069    lyonemoto@mednet.ucla.edu    Principal Investigator: Zev Wainberg, MD          Canada, Ontario Princess Margaret Cancer Centre Recruiting Toronto, Ontario, Canada, M5G 2M9 Contact: Philippe Bedard, M.D.    416-946-4534       Principal Investigator: Philippe Bedard, M.D. Collapse <<
    NCT03187288Acute Myeloid Leukemia ... more >> Myelodysplastic Syndromes Relapsed Cancer Refractory Cancer Collapse <<Phase 1RecruitingApril 4, 2022Canada, Ontario ... more >> Juravinski Hospital and Cancer Centre Not yet recruiting Hamilton, Ontario, Canada, L8V 1C3 Contact: Brian Leber, M.D.    905-521-2100 ext 76384       Princess Margaret Cancer Centre Recruiting Toronto, Ontario, Canada, M5G 2M9 Contact: Karen Yee, M.D.    416-946-4495 Collapse <<

实验方案

技术信息

CAS号 1338806-73-7 储存条件
分子式 C33H34N4O3 运输 蓝冰
分子量 534.65 别名 CFI-400945 Free Base

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