400-920-2911 sales@csnpharm.cn
您的位置 : 首页 / Cell Cycle / PLK / CFI-400945
CAS No.: 1338806-73-7
Synonyms: CFI-400945 Free Base
CFI400945 is a potent and selective,orally bioavailable PLK4 inhibitor with an IC50 value of 2.8 ±1.4 nM have potential antineoplastic activity.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT03624543 | Breast Cancer | Phase 2 | Not yet recruiting | December 31, 2020 | - |
NCT01954316 | Advanced Cancer | Phase 1 | Recruiting | September 2018 | United States, California ... more >> UCLA Medical Center Recruiting Santa Monica, California, United States, 90404 Contact: Lisa Yonemoto 310-582-4069 lyonemoto@mednet.ucla.edu Principal Investigator: Zev Wainberg, MD Canada, Ontario Princess Margaret Cancer Centre Recruiting Toronto, Ontario, Canada, M5G 2M9 Contact: Philippe Bedard, M.D. 416-946-4534 Principal Investigator: Philippe Bedard, M.D. Collapse << |
NCT03187288 | Acute Myeloid Leukemia ... more >> Myelodysplastic Syndromes Relapsed Cancer Refractory Cancer Collapse << | Phase 1 | Recruiting | April 4, 2022 | Canada, Ontario ... more >> Juravinski Hospital and Cancer Centre Not yet recruiting Hamilton, Ontario, Canada, L8V 1C3 Contact: Brian Leber, M.D. 905-521-2100 ext 76384 Princess Margaret Cancer Centre Recruiting Toronto, Ontario, Canada, M5G 2M9 Contact: Karen Yee, M.D. 416-946-4495 Collapse << |
实验方案
技术信息
CAS号 | 1338806-73-7 | 储存条件 |
|
|
分子式 | C33H34N4O3 | 运输 | 蓝冰 | |
分子量 | 534.65 | 别名 | CFI-400945 Free Base |
Cell Lines | Concentration | Assay Type | Time | Activity Description | Data Sources |
---|
A549 cells | - | Growth inhibition assay | 5 days | Growth inhibition of human A549 cells after 5 days by SRB assay, GI50=0.005 μM | 25723005 |
HCC1954 cells | - | Growth inhibition assay | 5 days | Growth inhibition of human HCC1954 cells after 5 days by SRB assay, GI50=5 nM | 25723005 |
HMEC cells | - | Growth inhibition assay | 5 days | Growth inhibition of human HMEC cells after 5 days by SRB assay, GI50=9 μM | 25723005 |
MCF7 cells | - | Growth inhibition assay | 5 days | Growth inhibition of human MCF7 cells after 5 days by SRB assay, GI50=8 nM | 25723005 |
MDA-MB-231 cells | - | Growth inhibition assay | 5 days | Growth inhibition of human MDA-MB-231 cells after 5 days by SRB assay, GI50=8.6 μM | 25723005 |
MDA-MB-468 cells | - | Growth inhibition assay | 5 days | Growth inhibition of human MDA-MB-468 cells after 5 days by SRB assay, GI50=0.006 μM | 25723005 |
SW620 cells | - | Growth inhibition assay | 5 days | Growth inhibition of human SW620 cells after 5 days by SRB assay, GI50=0.38 μM | 25723005 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT03624543 | Breast Cancer | Phase 2 | Not yet recruiting | December 31, 2020 | - |
NCT01954316 | Advanced Cancer | Phase 1 | Recruiting | September 2018 | United States, California ... more >> UCLA Medical Center Recruiting Santa Monica, California, United States, 90404 Contact: Lisa Yonemoto 310-582-4069 lyonemoto@mednet.ucla.edu Principal Investigator: Zev Wainberg, MD Canada, Ontario Princess Margaret Cancer Centre Recruiting Toronto, Ontario, Canada, M5G 2M9 Contact: Philippe Bedard, M.D. 416-946-4534 Principal Investigator: Philippe Bedard, M.D. Collapse << |
NCT03187288 | Acute Myeloid Leukemia ... more >> Myelodysplastic Syndromes Relapsed Cancer Refractory Cancer Collapse << | Phase 1 | Recruiting | April 4, 2022 | Canada, Ontario ... more >> Juravinski Hospital and Cancer Centre Not yet recruiting Hamilton, Ontario, Canada, L8V 1C3 Contact: Brian Leber, M.D. 905-521-2100 ext 76384 Princess Margaret Cancer Centre Recruiting Toronto, Ontario, Canada, M5G 2M9 Contact: Karen Yee, M.D. 416-946-4495 Collapse << |
联系我们
官方电话:400-920-2911
二维码
微信公众号 CSN官网