CAS No.: 138908-40-4
CL 316243/CL316243 二钠盐 Catalog No. CSN20033
Synonyms: CL 316,243 (sodium salt);BTA-243 Disodium Salt;CL-316,243
CL-316243 is a potent and highly selective β3-adrenoceptor agonist (EC50 = 3 nM) and > 10000-fold selective over β1 and β2 receptors. CL-316243 restores the expression of down-regulated fatty acid oxidation genes in type 2 diabetic mice.
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纯度 & 质量文件
批次:
靶点选择性
生物活性
- 描述
- 参考文献
- [1] Park JW, Jung KH, et al. 18F-FDG PET/CT monitoring of β3 agonist-stimulated brown adipocyte recruitment in white adipose tissue. J Nucl Med. 2015 Jan;56(1):153-8.
- [2] Ohsaka Y, Nomura Y. CL316243 induces phosphatidylinositol 3,4,5-triphosphate production in rat adipocytes in an adenosine deaminase-, pertussis toxin-, or wortmannin-sensitive manner. Physiol Res. 2016 Jul 18;65(3):543-6.
实验方案
- 计算器
- 储存液制备
技术信息
| CAS号 | 138908-40-4 | 储存条件 |
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| 分子式 | C20H18ClNNa2O7 | 运输 | 蓝冰 | |
| 分子量 | 465.79 | 别名 | CL 316,243 (sodium salt);BTA-243 Disodium Salt;CL-316,243;CL316,243. HP 186;HP-186 |
