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CAS No.: 1190932-38-7
Synonyms: RNR Inhibitor COH29
COH29 is a potent ribonucleotide reductase (RNR) inhibitor with anticancer activity with IC50 value of 8 μM in KB cell.
生物活性
靶点 | Ribonucleotide Reductase IC50:8μM |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT02112565 | Unspecified Adult Solid Tumor,... more >> Protocol Specific Collapse << | Phase 1 | Recruiting | November 2019 | United States, California ... more >> City of Hope Medical Center Recruiting Duarte, California, United States, 91010 Contact: Joseph Chao 626-471-9200 jchao@coh.org Principal Investigator: Joseph Chao Collapse << |
实验方案
技术信息
CAS号 | 1190932-38-7 | 储存条件 |
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分子式 | C22H16N2O5S | 运输 | 蓝冰 | |||||
分子量 | 420.44 | 别名 | RNR Inhibitor COH29 | |||||
溶解度 |
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动物实验配方 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT02112565 | Unspecified Adult Solid Tumor,... more >> Protocol Specific Collapse << | Phase 1 | Recruiting | November 2019 | United States, California ... more >> City of Hope Medical Center Recruiting Duarte, California, United States, 91010 Contact: Joseph Chao 626-471-9200 jchao@coh.org Principal Investigator: Joseph Chao Collapse << |
靶点 | Description | IC50 |
---|---|---|
Ribonucleotide Reductase | IC50:8μM |
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