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CAS No.: 1219168-18-9
Synonyms: Compound C dihydrochloride;BML-275 dihydrochloride;BML-275 2HCl
Dorsomorphin 2HCl is a selective AMPK inhibitor with Ki value of 109 nM.
生物活性
靶点 | AMPK Ki:109nM |
实验方案
技术信息
CAS号 | 1219168-18-9 | 储存条件 |
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分子式 | C24H27Cl2N5O | 运输 | 蓝冰 | |||||
分子量 | 472.41 | 别名 | Compound C dihydrochloride;BML-275 dihydrochloride;BML-275 2HCl;Compound C 2HCl;Dorsomorphin (hydrochloride);BML-275;Compound C;CpdC;Dorsomorphin HCl | |||||
溶解度 |
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动物实验配方 |
Cell Lines | Concentration | Assay Type | Time | Activity Description | Data Sources |
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mouse C2C12 cells | 4 μM | Function assay | - | Inhibition of BMPR1-mediated osteoblast differentiation in BMP4-stimulated mouse C2C12 cells assessed as decrease in alkaline phosphatase level at 4 uM by spectrophotometry | 18026094 |
靶点 | Description | IC50 |
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AMPK | Ki:109nM |
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