400-920-2911 sales@csnpharm.cn
您的位置 : 首页 / Protein Tyrosine Kinase/RTK / c-Kit / Dovitinib lactate hydrate
CAS No.: 915769-50-5
Synonyms: TKI258 lactate hydrate;CHIR-258 lactate hydrate;TKI-258
Dovitinib lactate is the Lactate of Dovitinib, which is a multitargeted RTK inhibitor, mostly for class III (FLT3/c-Kit) with IC50 of 1 nM/2 nM, also potent to class IV (FGFR1/3) and class V (VEGFR1-4) RTKs with IC50 of 8-13 nM, less potent to InsR, EGFR, c-Met, EphA2, Tie2, IGFR1 and HER2.
生物活性
实验方案
技术信息
CAS号 | 915769-50-5 | 储存条件 |
|
|
分子式 | C24H29FN6O5 | 运输 | 蓝冰 | |
分子量 | 500.52 | 别名 | TKI258 lactate hydrate;CHIR-258 lactate hydrate;TKI-258;CHIR-258;Dovitinib lactate |
联系我们
官方电话:400-920-2911
二维码
微信公众号 CSN官网