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CAS No.: 550999-75-2
Synonyms: EVP-6124;MT-4666
EVP-6124 is a partial agonist of α7 neuronal nicotinic acetylcholine receptors (nAChRs) and shows selectivity for α7 nAChRs and did not activate or inhibit heteromeric α4β2 nAChRs.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT02327182 | Alzheimer's Disease | Phase 3 | Terminated(This study was term... more >>inated due to the benefit-risk balance of MT-4666.) Collapse << | - | Japan ... more >> Investigational site Osaka, Kansai, Japan Collapse << |
NCT01073228 | Alzheimer's Disease ... more >> Central Nervous System Diseases Cognition Collapse << | Phase 2 | Completed | - | - |
NCT00766363 | Alzheimer's Disease ... more >> Central Nervous System Diseases Collapse << | Phase 1 | Completed | - | United States, California ... more >> Pacific Research Network, Inc. San Diego, California, United States, 92103 United States, Florida MD Clinical Hallandale Beach, Florida, United States, 33009 United States, New Jersey Comprehensive Clinical Research Berlin, New Jersey, United States, 08009 Global Medical Institutes, LLC Princeton, New Jersey, United States, 08540 Collapse << |
实验方案
技术信息
CAS号 | 550999-75-2 | 储存条件 |
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分子式 | C16H17ClN2OS | 运输 | 蓝冰 | |
分子量 | 320.84 | 别名 | EVP-6124;MT-4666 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT02327182 | Alzheimer's Disease | Phase 3 | Terminated(This study was term... more >>inated due to the benefit-risk balance of MT-4666.) Collapse << | - | Japan ... more >> Investigational site Osaka, Kansai, Japan Collapse << |
NCT01073228 | Alzheimer's Disease ... more >> Central Nervous System Diseases Cognition Collapse << | Phase 2 | Completed | - | - |
NCT00766363 | Alzheimer's Disease ... more >> Central Nervous System Diseases Collapse << | Phase 1 | Completed | - | United States, California ... more >> Pacific Research Network, Inc. San Diego, California, United States, 92103 United States, Florida MD Clinical Hallandale Beach, Florida, United States, 33009 United States, New Jersey Comprehensive Clinical Research Berlin, New Jersey, United States, 08009 Global Medical Institutes, LLC Princeton, New Jersey, United States, 08540 Collapse << |
NCT01556763 | Schizophrenia ... more >> Schizoaffective Disorder Central Nervous System Diseases Collapse << | Phase 1 | Completed | - | United States, Kansas ... more >> Clinical Research Institute Wichita, Kansas, United States, 67211 Collapse << |
NCT00968851 | Schizophrenia ... more >> Central Nervous System Diseases Cognition Collapse << | Phase 2 | Completed | - | - |
NCT01716975 | Schizophrenia ... more >> Impaired Cognition Collapse << | Phase 3 | Completed | - | - |
NCT01556763 | - | - | Completed | - | - |
NCT01480232 | Nicotine Dependence ... more >> Smoking Cessation Collapse << | Phase 2 | Terminated(Study has been put ... more >>on clinical hold by FDA) Collapse << | - | United States, Massachusetts ... more >> Massachusetts General Hospital Boston, Massachusetts, United States, 02114 Collapse << |
NCT00766363 | - | - | Completed | - | - |
NCT01969123 | Alzheimer's Disease ... more >> Dementia Collapse << | Phase 3 | Terminated(Study has been susp... more >>ended due to clinical hold.) Collapse << | January 2017 | - |
NCT01487135 | Healthy Subjects ... more >> Cardiac Repolarization Collapse << | Phase 1 | Completed | - | - |
NCT01714661 | Schizophrenia ... more >> Impaired Cognition Collapse << | Phase 3 | Completed | - | - |
NCT02004392 | Alzheimer's Disease ... more >> Dementia Collapse << | Phase 3 | Terminated(Study has been susp... more >>ended due to clinical hold.) Collapse << | August 2017 | - |
NCT01969136 | Alzheimer's Disease ... more >> Dementia Collapse << | Phase 3 | Terminated(Study has been susp... more >>ended due to clinical hold.) Collapse << | January 2017 | - |
NCT01480232 | - | - | Terminated(Study has been put ... more >>on clinical hold by FDA) Collapse << | - | - |
NCT02246075 | Alzheimer's Disease ... more >> Dementia Cognition Collapse << | Phase 2 | Withdrawn(Forum has decided no... more >>t to proceed with this study at this time.) Collapse << | - | United States, Florida ... more >> Delray Beach, Florida, United States United States, New Mexico Albuquerque, New Mexico, United States Collapse << |
NCT01984723 | Renal Impairment | Phase 1 | Completed | - | Czech Republic ... more >> Jankovcova 1569/2c, 17000 Praha 7, Czech Republic Hungary Rottenbiller u. 13 H-1077 Budapest, Hungary Collapse << |
NCT01984736 | Hepatic Impairment | Phase 1 | Completed | - | Czech Republic ... more >> Jankovcova 1569/2c, 17000 Praha 7, Czech Republic Poland Ul. Seczkowa 20B/8, Warszawa, Mazowieckie, 02-793, Poland Slovakia Bardosova 2/A 83101 Bratislava, Slovakia Collapse << |
NCT01714713 | Schizophrenia ... more >> Impaired Cognition Collapse << | Phase 3 | Completed | - | - |
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