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CAS No.: 872599-83-2

Epelsiban Catalog No. CSN22158

Synonyms: GSK 557296;GSK-557,296-B

GSK 557296 is a potent, selective and orally bioavailable oxytocin receptor antagonist, with a pKi of 9.9 for human oxytocin receptor.

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  • 描述
  • 临床研究
  • NCT号适应症或疾病临床期招募状态预计完成时间地点
    NCT02794467AdenomyosisPhase 2Withdrawn(Study was prematurel... more >>y discontinued due to GSK's change in prioritization for the portfolio and is not due to any safety concerns or regulatory interaction.) Collapse <<October 2016United States, District of Col... more >>umbia GSK Investigational Site Washington, DC, District of Columbia, United States, 20036 United States, Florida GSK Investigational Site West Palm Beach, Florida, United States, 33409 United States, Illinois GSK Investigational Site Champaign, Illinois, United States, 61820 United States, Louisiana GSK Investigational Site Mandeville, Louisiana, United States, 70471 GSK Investigational Site Metairie, Louisiana, United States, 70006 United States, Nebraska GSK Investigational Site Lincoln, Nebraska, United States, 68510 United States, Nevada GSK Investigational Site Las Vegas, Nevada, United States, 89128 United States, New Jersey GSK Investigational Site Lawrenceville, New Jersey, United States, 08648 United States, North Carolina GSK Investigational Site Durham, North Carolina, United States, 27713 GSK Investigational Site Raleigh, North Carolina, United States, 27612 United States, Ohio GSK Investigational Site Englewood, Ohio, United States, 45322 United States, Pennsylvania GSK Investigational Site Pittsburgh, Pennsylvania, United States, 15206 United States, Texas GSK Investigational Site Houston, Texas, United States, 77030 Collapse <<
    NCT02257359Embryo TransferPhase 1Completed-United States, Kansas ... more >> GSK Investigational Site Overland Park, Kansas, United States, 66211 Collapse <<
    NCT02213029Embryo TransferPhase 1Terminated-United States, California ... more >> GSK Investigational Site Glendale, California, United States, 91206 United States, Maryland GSK Investigational Site Baltimore, Maryland, United States, 21225 Collapse <<
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实验方案

技术信息

CAS号 872599-83-2 储存条件
分子式 C30H38N4O4 运输 蓝冰
分子量 518.65 别名 GSK 557296;GSK-557,296-B

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