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CAS No.: 1206123-37-6

Etrasimod Catalog No. CSN18981

Synonyms: APD334

Etrasimod is a potent, selective and orally available antagonist of the sphingosine-1-phosphate-1 (S1P1) receptor with an IC50 value of 1.88 nM in CHO cells.

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生物活性

  • 描述
  • 临床研究
  • NCT号适应症或疾病临床期招募状态预计完成时间地点
    NCT03072953Pyoderma GangrenosumPhase 2Terminated(Terminated [Sponsor... more >> decision to terminate the study]) Collapse <<-Australia, New South Wales ... more >> Westmead Hospital Westmead, New South Wales, Australia, 2145 Australia, Queensland Veracity Clinical Research Woolloongabba, Queensland, Australia, 4102 Australia, Victoria Eastern Clinical Research Unit Box Hill, Victoria, Australia, 3128 Royal Melbourne Hospital Parkville, Victoria, Australia, 3050 Australia, Western Australia Fremantle Dermatology Fremantle, Western Australia, Australia, 6160 New Zealand Braemar Day Hospital Hamilton, New Zealand Collapse <<
    NCT03139032Inflammatory Bowel Diseases ... more >> Skin Extra-intestinal Manifestations Collapse <<Phase 2Terminated(Sponsor decision to... more >> terminate the study) Collapse <<-Belgium ... more >> Arena 2001 Leuven, Belgium Germany Arena 1001 Hamburg, Germany Serbia Arena 3001 Belgrade, Serbia Collapse <<
    NCT03155932Primary Biliary CholangitisPhase 2RecruitingDecember 2019United States, California ... more >> Gastroenterology and Hepatology, UC Davis Medical Center Not yet recruiting Sacramento, California, United States, 95817 Principal Investigator: Chris Bowlus, MD          United States, Texas Baylor College of Medicine Recruiting Houston, Texas, United States, 77030 Principal Investigator: John Vierling, MD          Texas Liver Institute Recruiting San Antonio, Texas, United States, 78215 Principal Investigator: Eric Lawitz, MD          United States, Washington Swedish Medical Center Not yet recruiting Seattle, Washington, United States, 98104 Principal Investigator: Kris Kowdley, MD          Australia, New South Wales Royal Prince Alfred Hospital Recruiting Camperdown, New South Wales, Australia Contact: Simone Strasser, Prof          Australia, Queensland Sunshine Coast University Hospital Recruiting Birtinya, Queensland, Australia Contact: James OBeirne, Prof          Australia, Victoria Alfred Health Recruiting Melbourne, Victoria, Australia, 3004 Contact: William Kemp, Prof          New Zealand Auckland City Hospital Recruiting Grafton, Auckland, New Zealand Contact: Dominic Ray-Chaudhuri, Dr          Christchurch Clinical Studies Trust Recruiting Christchurch, New Zealand Contact: Jeffrey Ngu, Dr Collapse <<
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技术信息

CAS号 1206123-37-6 储存条件
分子式 C26H26F3NO3 运输 蓝冰
分子量 457.48 别名 APD334

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