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CAS No.: 885060-09-3
Synonyms: ARRY-520
ARRY-520 is a synthetic, small molecule kinesin spindle protein (KSP) inhibitor with IC50 of 6 nM.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT02092922 | Advanced Multiple Myeloma | Phase 2 | Completed | - | - |
NCT01989325 | Advanced Multiple Myeloma | Phase 2 | Completed | - | - |
NCT02384083 | Multiple Myeloma | Phase 1 Phase 2 | Active, not recruiting | December 2019 | Spain ... more >> Instoitut Català d'Oncologia Badalona, Spain, 08916 Hospital Clinico Universitario Barcelona, Spain, 08036 Hospital Doce de Octubre Madrid, Spain, 28041 Hospital Morales Messeguer Murcia, Spain, 30008 Clínica Universitaria de Navarra Pamplona, Spain, 31008 Hoapital Clinico Universitario Salamanca Salamanca, Spain, 37007 Hospital General de Segovia Segovia, Spain, 40002 Hospital Virgen del Rocío Sevilla, Spain, 41013 Hospital Universitario Dr Peset Valencia, Spain, 46017 Hospital Lozano Blesa Zaragoza, Spain, 50009 Collapse << |
实验方案
技术信息
CAS号 | 885060-09-3 | 储存条件 |
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分子式 | C20H22F2N4O2S | 运输 | 蓝冰 | |
分子量 | 420.48 | 别名 | ARRY-520 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT02092922 | Advanced Multiple Myeloma | Phase 2 | Completed | - | - |
NCT01989325 | Advanced Multiple Myeloma | Phase 2 | Completed | - | - |
NCT02384083 | Multiple Myeloma | Phase 1 Phase 2 | Active, not recruiting | December 2019 | Spain ... more >> Instoitut Català d'Oncologia Badalona, Spain, 08916 Hospital Clinico Universitario Barcelona, Spain, 08036 Hospital Doce de Octubre Madrid, Spain, 28041 Hospital Morales Messeguer Murcia, Spain, 30008 Clínica Universitaria de Navarra Pamplona, Spain, 31008 Hoapital Clinico Universitario Salamanca Salamanca, Spain, 37007 Hospital General de Segovia Segovia, Spain, 40002 Hospital Virgen del Rocío Sevilla, Spain, 41013 Hospital Universitario Dr Peset Valencia, Spain, 46017 Hospital Lozano Blesa Zaragoza, Spain, 50009 Collapse << |
NCT00462358 | Advanced Solid Tumors | Phase 1 | Completed | - | United States, Maryland ... more >> Marlene and Stewart Greenebaum Cancer Center Baltimore, Maryland, United States, 21201 United States, Michigan Wayne State University, Karmanos Cancer Institute Detroit, Michigan, United States, 48201 Collapse << |
NCT01372540 | Plasma Cell Leukemia ... more >> Recurrent Plasma Cell Myeloma Refractory Plasma Cell Myeloma Collapse << | Phase 1 | Active, not recruiting | February 24, 2019 | United States, Texas ... more >> M D Anderson Cancer Center Houston, Texas, United States, 77030 Collapse << |
NCT01248923 | Multiple Myeloma, Plasma Cell ... more >>Leukemia Collapse << | Phase 1 | Completed | - | United States, Alabama ... more >> Clearview Cancer Institute Huntsville, Alabama, United States, 35805 United States, Arizona Arizona Clinical Research Center, Inc. Tucson, Arizona, United States, 85715 United States, California City of Hope Duarte, California, United States, 91010 United States, Georgia Emory University, Winship Cancer Institute Atlanta, Georgia, United States, 30322 United States, Maryland Associates in Oncology/Hematology Rockville, Maryland, United States, 20850 United States, Michigan University of Michigan Comprehensive Cancer Center Ann Arbor, Michigan, United States, 48109 Karmanos Cancer Institute Detroit, Michigan, United States, 48201 United States, New York NYU Cancer Center New York, New York, United States, 10016 Mount Sinai Medical Center New York, New York, United States, 10029 United States, South Carolina Charleston Hematology Oncology Associates Charleston, South Carolina, United States, 29414 United States, Tennessee The Jones Clinic Germantown, Tennessee, United States, 38138 Vanderbilt-Ingram Cancer Center Nashville, Tennessee, United States, 37212 United States, Texas Baylor Charles A. Sammons Cancer Center at Dallas Dallas, Texas, United States, 75246 Collapse << |
NCT00637052 | Advanced MDS ... more >>Acute Myeloid Leukemia Collapse << | Phase 1 Phase 2 | Completed | - | United States, Georgia ... more >> Emory University School of Medicine, Winship Cancer Center Atlanta, Georgia, United States, 30322 United States, Texas University of Texas, M.D. Anderson Cancer Center Houston, Texas, United States, 77030 Collapse << |
NCT00821249 | Multiple Myeloma ... more >> Plasma Cell Leukemia Collapse << | Phase 1 Phase 2 | Completed | - | United States, Georgia ... more >> Emory University, Winship Cancer Institute Atlanta, Georgia, United States, 30322 United States, Michigan Karmanos Cancer Institute Detroit, Michigan, United States, 48201 United States, Pennsylvania Fox Chase Cancer Center Philadelphia, Pennsylvania, United States, 19111 United States, Texas MD Anderson Cancer Center Houston, Texas, United States, 77030 United States, Washington Fred Hutchinson Cancer Research Center Seattle, Washington, United States, 98109 Collapse << |
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