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CAS No.: 895519-90-1
Synonyms: HHGV678
Flumatinib is a multi-kinase inhibitor with IC50 Values of 1.2 nM, 307.6 nM and 2662 nM for c-Abl, PDGFRβ and c-Kit respectively.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT02204644 | CML, CML-CP,MMR,TKI | Phase 3 | Completed | - | China, Tianjin ... more >> Hospital of Blood Diseases, Chinese Academy of Medical Sciences Tianjin, Tianjin, China, 300020 Collapse << |
NCT01503502 | Myelogenous Leukemia, Chronic | Phase 2 | Unknown | December 2014 | China, Beijing ... more >> Peking University People's Hospital Beijing, Beijing, China, 100044 China, Hubei Union Hospital Tongji Medical College Huazhong University of Science and technology Wuhan, Hubei, China, 430022 China, Jiangsu The First Rffiurted Hospital of Soochow University Suzhou, Jiangsu, China, 215006 China, Shanghai Ruijin Hospital Shanghai, Shanghai, China, 200025 China, Tianjin Institute of Hematology & Blood Diseases Hospital, Chinese Academy of Medical Sciences & Peking Union Medical College Tianjin, Tianjin, China, 300020 Collapse << |
NCT02511340 | Chronic Myelogenous Leukemia | Phase 2 | Unknown | December 2015 | China, Hubei ... more >> Union Hospital Tongji Medical College Huazhong University of Science and technology Wuhan, Hubei, China, 430022 Collapse << |
实验方案
技术信息
CAS号 | 895519-90-1 | 储存条件 |
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分子式 | C29H29F3N8O | 运输 | 蓝冰 | |
分子量 | 562.59 | 别名 | HHGV678 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT02204644 | CML, CML-CP,MMR,TKI | Phase 3 | Completed | - | China, Tianjin ... more >> Hospital of Blood Diseases, Chinese Academy of Medical Sciences Tianjin, Tianjin, China, 300020 Collapse << |
NCT01503502 | Myelogenous Leukemia, Chronic | Phase 2 | Unknown | December 2014 | China, Beijing ... more >> Peking University People's Hospital Beijing, Beijing, China, 100044 China, Hubei Union Hospital Tongji Medical College Huazhong University of Science and technology Wuhan, Hubei, China, 430022 China, Jiangsu The First Rffiurted Hospital of Soochow University Suzhou, Jiangsu, China, 215006 China, Shanghai Ruijin Hospital Shanghai, Shanghai, China, 200025 China, Tianjin Institute of Hematology & Blood Diseases Hospital, Chinese Academy of Medical Sciences & Peking Union Medical College Tianjin, Tianjin, China, 300020 Collapse << |
NCT02511340 | Chronic Myelogenous Leukemia | Phase 2 | Unknown | December 2015 | China, Hubei ... more >> Union Hospital Tongji Medical College Huazhong University of Science and technology Wuhan, Hubei, China, 430022 Collapse << |
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