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CAS No.: 1015787-98-0
Synonyms: MK-7264;AF-219;RO-4926219
Gefapixant is an orally active P2X3 receptor (P2X3R) antagonist with IC50s of ~30 nM versus recombinant hP2X3 homotrimers and 100-250 nM at hP2X2/3 heterotrimeric receptors.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT02612623 | Refractory Chronic Cough | Phase 2 | Completed | - | United States, California ... more >> Afferent Investigative Site Mission Viejo, California, United States Afferent Investigative Site San Jose, California, United States United States, Colorado Afferent Investigative Site Colorado Springs, Colorado, United States United States, Florida Afferent Investigative Site Largo, Florida, United States United States, North Carolina Afferent Investigative Site Charlotte, North Carolina, United States United States, Oklahoma Afferent Investigative Site Tulsa, Oklahoma, United States United States, Texas Afferent Investigative Site Dallas, Texas, United States Afferent Investigative Site San Antonio, Texas, United States United States, Washington Afferent Investigative Site Bellevue, Washington, United States United States, Wisconsin Afferent Investigative Site Greenfield, Wisconsin, United States Collapse << |
NCT01554579 | Osteoarthritis of the Knee | Phase 2 | Completed | - | - |
NCT01554579 | - | - | Completed | - | - |
实验方案
技术信息
CAS号 | 1015787-98-0 | 储存条件 |
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分子式 | C14H19N5O4S | 运输 | 蓝冰 | |
分子量 | 353.40 | 别名 | MK-7264;AF-219;RO-4926219 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT02612623 | Refractory Chronic Cough | Phase 2 | Completed | - | United States, California ... more >> Afferent Investigative Site Mission Viejo, California, United States Afferent Investigative Site San Jose, California, United States United States, Colorado Afferent Investigative Site Colorado Springs, Colorado, United States United States, Florida Afferent Investigative Site Largo, Florida, United States United States, North Carolina Afferent Investigative Site Charlotte, North Carolina, United States United States, Oklahoma Afferent Investigative Site Tulsa, Oklahoma, United States United States, Texas Afferent Investigative Site Dallas, Texas, United States Afferent Investigative Site San Antonio, Texas, United States United States, Washington Afferent Investigative Site Bellevue, Washington, United States United States, Wisconsin Afferent Investigative Site Greenfield, Wisconsin, United States Collapse << |
NCT01554579 | Osteoarthritis of the Knee | Phase 2 | Completed | - | - |
NCT01554579 | - | - | Completed | - | - |
NCT01569438 | - | - | Completed | - | - |
NCT02612610 | Refractory Chronic Cough | Phase 2 | Completed | - | - |
NCT01432730 | Chronic Cough | Phase 2 | Completed | - | United Kingdom ... more >> North West Lung Research Centre, Wythenshawe Hospital Manchester, United Kingdom, M23 9LT Collapse << |
NCT03449134 | Chronic Cough | Phase 3 | Recruiting | July 10, 2020 | - |
NCT02612610 | - | - | Completed | - | - |
NCT01569438 | Bladder Pain Syndrome | Phase 2 | Completed | - | - |
NCT02502097 | Idiopathic Pulmonary Fibrosis ... more >> Cough Collapse << | Phase 2 | Completed | - | - |
NCT02349425 | Refractory Chronic Cough | Phase 2 | Completed | - | - |
NCT03654326 | Endometriosis-related Pain | Phase 2 | Recruiting | October 22, 2019 | - |
NCT03108924 | Renal Insufficiency | Phase 1 | Completed | - | United States, Florida ... more >> Clinical Pharmacology of Miami ( Site 0001) Hialeah, Florida, United States, 33014 Orlando Clinical Research Center ( Site 0002) Orlando, Florida, United States, 32809 Collapse << |
NCT03449147 | Chronic Cough | Phase 3 | Recruiting | January 8, 2021 | - |
NCT03569033 | Acute Cough | Phase 2 | Recruiting | June 21, 2019 | United Kingdom ... more >> Hvivo Service Limited. Queen Mary BioEnterprises ( Site 0003) Recruiting London, United Kingdom, E1 2AX Contact: Study Coordinator +442077561300 Collapse << |
NCT02476890 | Refractory Chronic Cough | Phase 2 | Completed | - | - |
NCT02790840 | Healthy | Phase 1 | Completed | - | United States, Arizona ... more >> Celerion Tempe, Arizona, United States, 85283 Collapse << |
NCT03696108 | Chronic Cough | Phase 3 | Recruiting | October 6, 2020 | Japan ... more >> Oishi Clinic ( Site 3818) Recruiting Kasuya-gun, Fukuoka, Japan, 811-2310 Contact: Study Coordinator +81929381900 Nagata Hospital ( Site 3815) Recruiting Yanagawa, Fukuoka, Japan, 832-0059 Contact: Study Coordinator +81944723501 Japan Community Health care Organization Kanazawa Hospital ( Site 3817) Recruiting Kanazawa, Ishikawa, Japan, 920-8610 Contact: Study Coordinator +81762522200 Matsusaka City Hospital ( Site 3825) Recruiting Matsusaka, Mie, Japan, 515-8544 Contact: Study Coordinator +81598231515 Sugiura Clinic ( Site 3806) Recruiting Kawaguchi, Saitama, Japan, 332-0012 Contact: Study Coordinator +81482225015 National Hospital Organization Matsue Medical Center ( Site 3848) Recruiting Matsue, Shimane, Japan, 690-8556 Contact: Study Coordinator +81852216131 Kiheibashi Otolaryngology ( Site 3828) Recruiting Kodaira, Tokyo, Japan, 187-0044 Contact: Study Coordinator +81423323387 Tochigi Takao Clinic ( Site 3833) Recruiting Kagoshima, Japan, 890-0073 Contact: Study Coordinator +81998138111 Nagano Red Cross Hospital ( Site 3859) Recruiting Nagano, Japan, 380-8582 Contact: Study Coordinator +81262264131 Saiseikai Niigata Daini Hospital ( Site 3831) Recruiting Niigata, Japan, 950-1104 Contact: Study Coordinator +81252336161 Oita Red Cross Hospital ( Site 3837) Recruiting Oita, Japan, 870-0033 Contact: Study Coordinator +81975326181 Yamagata Clinic ( Site 3813) Recruiting Oita, Japan, 870-0921 Contact: Study Coordinator +81975562456 Chibana Clinic ( Site 3809) Recruiting Okinawa, Japan, 904-2143 Contact: Study Coordinator +81989391301 Ito ENT Clinic ( Site 3816) Recruiting Shizuoka, Japan, 420-0803 Contact: Study Coordinator +81542651000 Collapse << |
NCT02492776 | Healthy | Phase 1 | Completed | - | United States, Arizona ... more >> Celerion Tempe, Arizona, United States, 85283 Collapse << |
NCT01993329 | Asthma | Phase 1 | Completed | - | United Kingdom ... more >> Medicines Evaluation Unit Manchester, United Kingdom, M23 9QZ Collapse << |
NCT02477709 | Idiopathic Pulmonary Fibrosis | Phase 2 | Completed | - | United States, North Carolina ... more >> American Health Research Charlotte, North Carolina, United States, 28207 Collapse << |
NCT02476890 | - | - | Completed | - | - |
NCT02477709 | - | - | Completed | - | - |
NCT02229877 | Healthy Volunteers | Phase 1 | Completed | - | United States, Arizona ... more >> Celerion Tempe, Arizona, United States, 85283 Collapse << |
NCT02397460 | Refractory Chronic Cough | Phase 2 | Completed | - | United Kingdom ... more >> The Medicines Evaluation Unit Manchester, United Kingdom, M23 9QZ Collapse << |
NCT03482713 | Chronic Cough | Phase 2 | Completed | - | Japan ... more >> Nagoya City University Hospital ( Site 3328) Nagoya, Aichi, Japan, 467-8602 Idaimae Minamiyojo Int Clinic ( Site 3321) Sapporo, Hokkaido, Japan, 064-0804 Tsumura Cardiovascular-internal-medicine Clinic ( Site 3314) Kakogawa, Hyogo, Japan, 675-0101 Hitachi, Ltd. Hitachinaka General Hospital ( Site 3301) Hitachinaka, Ibaraki, Japan, 312-0057 Saiseikai Kanazawa Hospital ( Site 3337) Kanazawa, Ishikawa, Japan, 920-0353 Komatsu Municipal Hospital ( Site 3308) Komatsu, Ishikawa, Japan, 923-8560 Kamei Internal Medicine and Respiratory Clinic ( Site 3309) Takamatsu, Kagawa, Japan, 761-8073 Yokohama City Minato Red Cross Hospital ( Site 3306) Yokohama, Kanagawa, Japan, 231-8682 Matsusaka City Hospital ( Site 3325) Matsusaka, Mie, Japan, 515-8544 Nagaoka Red Cross Hospital ( Site 3307) Nagaoka, Niigata, Japan, 940-2085 Kawaguchi Respiratory Clinic ( Site 3304) Higashiosaka, Osaka, Japan, 577-0843 Fukushima Medical University Hospital ( Site 3338) Fukushima, Japan, 960-1295 Doujin Memorial Medical Foundation, Meiwa Hospital ( Site 3310) Tokyo, Japan, 101-0041 Nihonbashi Medical & Allergy Clinic ( Site 3334) Tokyo, Japan, 103-0022 Fukuwa Clinic ( Site 3311) Tokyo, Japan, 103-0027 Showa University Hospital ( Site 3331) Tokyo, Japan, 142-8666 Collapse << |
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