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CAS No.: 1075236-89-3
Synonyms: GSK2140944;GSK-2140944E
Gepotidacin is a first in class triazaacenaphthylene antibiotic that inhibits bacterial type II DNA replication by inhibiting the activity of bacterial topoisomerase and has in vitro activity against susceptible and drug-resistant pathogens.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT02202187 | Infections, Respiratory Tract | Phase 1 | Completed | - | United States, Minnesota ... more >> GSK Investigational Site Minneapolis, Minnesota, United States, 55404 Collapse << |
NCT01706315 | Infections, Respiratory Tract | Phase 1 | Completed | - | United States, Kansas ... more >> GSK Investigational Site Overland Park, Kansas, United States, 66211 Collapse << |
NCT02045849 | Infections, Bacterial | Phase 1 | Completed | - | United States, Kansas ... more >> GSK Investigational Site Overland Park, Kansas, United States, 66211 Collapse << |
实验方案
技术信息
CAS号 | 1075236-89-3 | 储存条件 |
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分子式 | C24H28N6O3 | 运输 | 蓝冰 | |
分子量 | 448.52 | 别名 | GSK2140944;GSK-2140944E |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT02202187 | Infections, Respiratory Tract | Phase 1 | Completed | - | United States, Minnesota ... more >> GSK Investigational Site Minneapolis, Minnesota, United States, 55404 Collapse << |
NCT01706315 | Infections, Respiratory Tract | Phase 1 | Completed | - | United States, Kansas ... more >> GSK Investigational Site Overland Park, Kansas, United States, 66211 Collapse << |
NCT02045849 | Infections, Bacterial | Phase 1 | Completed | - | United States, Kansas ... more >> GSK Investigational Site Overland Park, Kansas, United States, 66211 Collapse << |
NCT01934205 | Infections, Bacterial | Phase 1 | Completed | - | United States, Maryland ... more >> GSK Investigational Site Baltimore, Maryland, United States, 21225 Collapse << |
NCT02294682 | Gonorrhea | Phase 2 | Completed | - | United States, California ... more >> GSK Investigational Site Fountain Valley, California, United States, 92708 GSK Investigational Site Los Angeles, California, United States, 90028 GSK Investigational Site Los Angeles, California, United States, 90069 GSK Investigational Site Palm Springs, California, United States, 92262 GSK Investigational Site San Francisco, California, United States, 94103 United States, Florida GSK Investigational Site Orlando, Florida, United States, 32806 United States, Georgia GSK Investigational Site Atlanta, Georgia, United States, 30308 United States, Indiana GSK Investigational Site Indianapolis, Indiana, United States, 46202 United States, Louisiana GSK Investigational Site New Orleans, Louisiana, United States, 70119 United States, Nebraska GSK Investigational Site Omaha, Nebraska, United States, 68114 United States, Ohio GSK Investigational Site Cleveland, Ohio, United States, 44109 United States, Pennsylvania GSK Investigational Site Jenkintown, Pennsylvania, United States, 19046 Puerto Rico GSK Investigational Site San Juan, Puerto Rico, 00927 United Kingdom GSK Investigational Site London, United Kingdom, SW10 9NH Collapse << |
NCT02045797 | Infections, Bacterial | Phase 2 | Completed | - | - |
NCT01615796 | Infections, Respiratory Tract | Phase 1 | Completed | - | Australia, New South Wales ... more >> GSK Investigational Site Randwick, New South Wales, Australia, 2031 Collapse << |
NCT02000765 | Infections, Respiratory Tract | Phase 1 | Completed | - | United Kingdom ... more >> GSK Investigational Site London, United Kingdom, NW10 7NS Collapse << |
NCT02257398 | Infections, Respiratory Tract | Phase 1 | Completed | - | United States, Texas ... more >> GSK Investigational Site Austin, Texas, United States, 78744 Collapse << |
NCT02045797 | - | - | Completed | - | - |
NCT02853435 | Infections, Bacterial | Phase 1 | Completed | - | United States, California ... more >> GSK Investigational Site Anaheim, California, United States, 92801 United States, Texas GSK Investigational Site Austin, Texas, United States, 78744 Collapse << |
NCT02729038 | Infections, Bacterial | Phase 1 | Completed | - | United States, Florida ... more >> GSK Investigational Site Miami, Florida, United States, 33136 GSK Investigational Site Orlando, Florida, United States, 32809 United States, Minnesota GSK Investigational Site Minneapolis, Minnesota, United States, 55404 Collapse << |
NCT02294682 | - | - | Completed | - | - |
NCT03562117 | Infections, Bacterial | Phase 1 | Recruiting | April 10, 2019 | United States, Florida ... more >> GSK Investigational Site Recruiting Miami, Florida, United States, 33136 Contact: US GSK Clinical Trials Call Center 877-379-3718 GSKClinicalSupportHD@gsk.com Contact: EU GSK Clinical Trials Call Center +44 (0) 20 8990 4466 GSKClinicalSupportHD@gsk.com GSK Investigational Site Recruiting Orlando, Florida, United States, 32809 Contact: US GSK Clinical Trials Call Center 877-379-3718 GSKClinicalSupportHD@gsk.com Contact: EU GSK Clinical Trials Call Center +44 (0) 20 8990 4466 GSKClinicalSupportHD@gsk.com Collapse << |
NCT02729038 | - | - | Completed | - | - |
NCT03568942 | Infections, Bacterial | Phase 2 | Recruiting | December 14, 2018 | United States, California ... more >> GSK Investigational Site Recruiting La Mesa, California, United States, 91942 Contact: US GSK Clinical Trials Call Center 877-379-3718 GSKClinicalSupportHD@gsk.com Contact: EU GSK Clinical Trials Call Center +44 (0) 20 8990 4466 GSKClinicalSupportHD@gsk.com Collapse << |
NCT02853435 | - | - | Completed | - | - |
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