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CAS No.: 1095173-27-5
Synonyms: PF-04449913;PF-4449913
PF-04449913 is a potent and orally bioavailable smoothened inhibitor. PF-04449913 binds to human SMO (amino acids 181-787) with an IC50 of 4 nM.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT03390296 | Acute Myeloid Leukemia | Phase 2 | Recruiting | December 2024 | United States, Texas ... more >> University of Texas MD Anderson Cancer Center Recruiting Houston, Texas, United States, 77030 Contact ndaver@mdanderson.org Collapse << |
NCT03162900 | Healthy Volunteers | Phase 1 | Completed | - | Belgium ... more >> Pfizer Clinical Research Unit Brussels, Belgium, B-1070 Collapse << |
NCT02430545 | Healthy Volunteers | Phase 1 | Completed | - | United States, Connecticut ... more >> New Haven Clinical Research Unit New Haven, Connecticut, United States, 06511 Collapse << |
实验方案
技术信息
CAS号 | 1095173-27-5 | 储存条件 |
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分子式 | C21H22N6O | 运输 | 蓝冰 | |||||||
分子量 | 374.44 | 别名 | PF-04449913;PF-4449913 | |||||||
溶解度 |
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动物实验配方 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT03390296 | Acute Myeloid Leukemia | Phase 2 | Recruiting | December 2024 | United States, Texas ... more >> University of Texas MD Anderson Cancer Center Recruiting Houston, Texas, United States, 77030 Contact ndaver@mdanderson.org Collapse << |
NCT03162900 | Healthy Volunteers | Phase 1 | Completed | - | Belgium ... more >> Pfizer Clinical Research Unit Brussels, Belgium, B-1070 Collapse << |
NCT02430545 | Healthy Volunteers | Phase 1 | Completed | - | United States, Connecticut ... more >> New Haven Clinical Research Unit New Haven, Connecticut, United States, 06511 Collapse << |
NCT03270878 | Healthy Volunteer Study | Phase 1 | Completed | - | United States, Connecticut ... more >> New Haven Clinical Research Unit New Haven, Connecticut, United States, 06511 Collapse << |
NCT03627754 | Hepatic Impairment | Phase 1 | Recruiting | January 1, 2020 | United States, Florida ... more >> Investigational Drug Services (IDS) University of Miami Hospitals and Clinics, Research Pharmacy Recruiting Miami, Florida, United States, 33136 University of Miami Division of Clinical Pharmacology Recruiting Miami, Florida, United States, 33136 Orlando Clinical Research Center Recruiting Orlando, Florida, United States, 32809 Collapse << |
NCT03416179 | Leukemia, Myeloid, Acute | Phase 3 | Recruiting | July 22, 2025 | - |
NCT02226172 | Primary Myelofibrosis; Post-po... more >>lycythemia Vera Myelofibrosis; Post-essential Thrombocythemia Myelofibrosis Collapse << | Phase 2 | Terminated | - | United States, Arizona ... more >> Mayo Clinic Building - Phoenix Phoenix, Arizona, United States, 85054 Mayo Clinic Hospital Phoenix, Arizona, United States, 85054 Mayo Clinic Scottsdale, Arizona, United States, 85259 United States, California UC San Diego Moores Cancer Center - Investigational Drug Services La Jolla, California, United States, 92037-0845 UCSD Medical Center Clinical Laboratory - La Jolla La Jolla, California, United States, 92037 University of California San Diego (UCSD) Moores Cancer Center La Jolla, California, United States, 92093-0698 UC San Diego Medical Center- Hillcrest San Diego, California, United States, 92103 United States, Michigan University of Michigan Ann Arbor, Michigan, United States, 48109 United States, New York Weill Cornell Medical College - New York-Presbyterian Hospital New York, New York, United States, 10021 Herbert Irving Comprehensive Cancer Center-Columbia University Medical Center New York, New York, United States, 10032 Weill Cornell Medical College-New York Presbyterian Hospital New York, New York, United States, 10065 United States, Ohio Cleveland Clinic - Taussig Cancer Institute Cleveland, Ohio, United States, 44195 United States, Utah Huntsman Cancer Institute-University of Utah Salt Lake City, Utah, United States, 84112 University of Utah, Huntsman Cancer Hospital Salt Lake City, Utah, United States, 84112 United States, Wisconsin Froedtert Hospital and Medical College of Wisconsin Milwaukee, Wisconsin, United States, 53226-3522 Japan Kobe University Hospital Kobe, Hyogo, Japan, 6500017 Osaka University Hopsital Suita-Shi, Osaka, Japan, 565-0871 Juntendo University Hospital Bunkyo-ku, Tokyo, Japan, 113-8431 Tokyo Medical University Hospital Tokyo, Japan, 160-0023 Collapse << |
NCT03130556 | Healthy Volunteers | Phase 1 | Completed | - | United States, Connecticut ... more >> Pfizer New Haven Clinical Research Unit New Haven, Connecticut, United States, 06511 Collapse << |
NCT01546038 | Acute Myeloid Leukemia | Phase 2 | Active, not recruiting | June 2019 | - |
NCT02226172 | - | - | Terminated | - | - |
NCT01842646 | Myelodysplastic Syndrome (MDS)... more >> Chronic Myelomonocytic Leukemia (CMML) Collapse << | Phase 2 | Active, not recruiting | March 2020 | United States, Florida ... more >> H. Lee Moffitt Cancer Center and Research Institute Tampa, Florida, United States, 33612 Collapse << |
NCT01842646 | - | - | Active, not recruiting | - | - |
NCT03466450 | Glioblastoma | Phase 1 Phase 2 | Recruiting | March 2021 | Spain ... more >> Institut Catalá de Oncología Badalona/Hospital Germans Trias i Pujol Recruiting Badalona, Barcelona, Spain, 08916 Contact: Carmen Balañá, M.D. +34 972 22 58 34 cbalana@iconcologia.net Principal Investigator: Carmen Balañá, M.D. Institut Catalá de Oncología Girona/Hospital Universitari Dr. Josep Trueta Recruiting Girona, Spain, 17007 Contact: Sonia del Barco, M.D. +34 972 22 58 34 ext 7977 sdelbarco@iconcologia.net Principal Investigator: Sonia del Barco, M.D. Hospital Universitario Ramón y Cajal Recruiting Madrid, Spain Contact: Mª Ángeles Vaz 91 336 80 00 ext 7977 mavaz4@gmail.com Principal Investigator: Mª Ángeles Vaz, M.D. Hospital Universitario y Politécnico La Fe Recruiting Valencia, Spain, 46009 Contact: José Muñoz Langa, M.D. +34 934344412 munyoz_joslan@gva.es Principal Investigator: José Muñoz Langa, M.D. Collapse << |
NCT00953758 | Hematologic Malignancies | Phase 1 | Completed | - | United States, California ... more >> Pfizer Investigational Site La Jolla, California, United States, 92037 Pfizer Investigational Site La Jolla, California, United States, 92093 Pfizer Investigational Site San Diego, California, United States, 92103 United States, Texas Pfizer Investigational Site Houston, Texas, United States, 77030-4009 United States, Washington Pfizer Investigational Site Seattle, Washington, United States, 98109-1023 Italy Pfizer Investigational Site Bologna, Italy, 40138 Collapse << |
NCT02367456 | Myelodysplastic Syndrome ... more >> Acute Myeloid Leukemia Collapse << | Phase 2 | Recruiting | October 10, 2021 | - |
NCT01546038 | - | - | Active, not recruiting | - | - |
NCT02038777 | Acute Myeloid Leukemia | Phase 1 | Recruiting | October 31, 2019 | Japan ... more >> Japanese Red Cross Nagoya First Hospital Recruiting Nagoya, Aichi, Japan, 453-8511 Kobe University Hospital Recruiting Kobe-shi, Hyogo, Japan, 650-0017 Tohoku University Hospital Recruiting Sendai, Miyagi, Japan, 980-8574 National Cancer Center Hospital Recruiting Chuo-ku, Tokyo, Japan, 104-0045 Akita University Hospital Recruiting Akita, Japan, 010-8543 Kyushu University Hospital Recruiting Fukuoka, Japan, 812-8582 Tokyo Medical University Hospital Recruiting Tokyo, Japan, 160-0023 Collapse << |
NCT01286467 | Solid Tumors | Phase 1 | Completed | - | United States, California ... more >> Pfizer Investigational Site Los Angeles, California, United States, 90033 United States, Colorado Pfizer Investigational Site Aurora, Colorado, United States, 80045 United States, Massachusetts Pfizer Investigational Site Boston, Massachusetts, United States, 02115 Collapse << |
NCT02110342 | Healthy | Phase 1 | Completed | - | United States, Wisconsin ... more >> Pfizer Investigational Site Madison, Wisconsin, United States, 53704 Collapse << |
NCT03596567 | Renal Impairment | Phase 1 | Completed | - | United States, Florida ... more >> University of Miami Division of Clinical Pharmacology Miami, Florida, United States, 33136 University of Miami, Sylvester Comprehensive Cancer Center Miami, Florida, United States, 33136 United States, Minnesota Prism Clinical Research LLC Saint Paul, Minnesota, United States, 55114 Collapse << |
NCT01841333 | Adult Acute Myeloid Leukemia i... more >>n Remission Recurrent Adult Acute Myeloid Leukemia Collapse << | Phase 2 | Recruiting | April 2020 | United States, Colorado ... more >> University of Colorado Cancer Center Recruiting Aurora, Colorado, United States, 80045 Contact: Emily Denoncourt, RN, BSN, OCN 720-848-0566 emily.denoncourt@ucdenver.edu Principal Investigator: Dan A Pollyea, MD, MS United States, Ohio Ohio State University Not yet recruiting Columbus, Ohio, United States, 43210 Contact: Steve Devine, MD 614-293-5655 Principal Investigator: Steve Devine, MD Collapse << |
NCT01749085 | Healthy Volunteers | Phase 1 | Completed | - | United States, Connecticut ... more >> Pfizer Investigational Site New Haven, Connecticut, United States, 06511 Collapse << |
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