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CAS No.: 928037-13-2
Synonyms: E-7050
Golvatinib is a dual c-Met and VEGFR-2 inhibitor with IC50 of 14 nM and 16 nM.
规格 | 价格 | 促销价格 | 库存 | 数量 |
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生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT01355302 | Advanced or Metastatic Solid T... more >>umors Previously Untreated Gastric Cancer Collapse << | Phase 1 Phase 2 | Terminated(Sites not recruitin... more >>g) Collapse << | - | United States, Arizona ... more >> Arizona Oncology Associates, PC - CASA Tucson, Arizona, United States, 85715 United States, Florida Boca Raton Clinical Research Associates, Inc Plantation, Florida, United States, 33324 United States, Illinois Robert H. Lurie Comprenhensive Cancer Center of Northwestern University Chicago, Illinois, United States, 60611 United States, Michigan University of Michigan Comprehensive Cancer Center Ann Arbor, Michigan, United States, 48109 Barbara Ann Karmanos Cancer Institute Detroit, Michigan, United States, 48084 Henry Ford Medical Center Detroit, Michigan, United States, 48202 United States, North Carolina University of North Carolina at Chapel Hill Chapell Hill, North Carolina, United States, 27599 Duke University Medical Center Durham, North Carolina, United States, 27710 United States, Ohio Mercy Cancer Centerr at St. Anne Toledo, Ohio, United States, 43623 Russian Federation Chelyabinsk Regional Oncology Dispensary Chelyabinsk, Russian Federation, 454087 GOU VPO St-Petersburg SMA n/a Mechnikov Fed. Agen. of Healthcare and Social Developm. St Petersburg, Russian Federation, 195067 FSI "SRC of Oncology n. a. N.N.Petrov of Rosmedtekhnologiy" St Petersburg, Russian Federation, 197758 Ukraine SI Dnipropetrovsk Medical Academy of MOHU ch of Oncology and Medical Radiology Dnipropetrovsk, Ukraine, 49102 Municipal Clinical Medical and Prophylactic Institution Donetsk Regional Antitumor Centre Donetsk, Ukraine, 83092 Kyiv City Clinical Oncological Center Kyiv, Ukraine, 3115 Lviv State Oncol. Reg. Treatment and Diagnostic Center Lviv, Ukraine, 79031 United Kingdom Barts and the London NHS Trust London, Greater London, United Kingdom, EC1A 7BE Sarah Cannon Research UK London, Greater London, United Kingdom, W1G 6AD The Christie NHS Foundation Trust Manchester, Greater Manchester, United Kingdom, M20 4BX Collapse << |
NCT01355302 | - | - | Terminated(Sites not recruitin... more >>g) Collapse << | - | - |
实验方案
技术信息
CAS号 | 928037-13-2 | 储存条件 |
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分子式 | C33H37F2N7O4 | 运输 | 蓝冰 | |||||||||
分子量 | 633.69 | 别名 | E-7050 | |||||||||
溶解度 |
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动物实验配方 |
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