400-920-2911 sales@csnpharm.cn
您的位置 : 首页 / PI3K/Akt/mTOR / Akt / GSK2110183 analog 1 HCl
CAS No.: 2070009-64-0
Synonyms: Afuresertib-F;GSK-2110183-analog;Afuresertib-F HCl
GSK2110183 HCl is an orally bioavailable, selective, ATP-competitive and potent pan-Akt inhibitor with IC50s of 0.08/2/2.6 nM for Akt1/Akt2/Akt3 respectively.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT01445587 | Cancer | Phase 2 | Withdrawn(Based on the clinica... more >>l activity, not safety data, of the AKT inhibitor, GSK has decided at this time to suspend further development of GSK2110183 as monotherapy.) Collapse << | November 2011 | Australia, Victoria ... more >> GSK Investigational Site Melbourne, Victoria, Australia, 3004 Collapse << |
实验方案
技术信息
CAS号 | 2070009-64-0 | 储存条件 |
|
|
分子式 | C18H17Cl3F2N4OS | 运输 | 蓝冰 | |
分子量 | 481.77 | 别名 | Afuresertib-F;GSK-2110183-analog;Afuresertib-F HCl;Afuresertib-F hydrochloride |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT01445587 | Cancer | Phase 2 | Withdrawn(Based on the clinica... more >>l activity, not safety data, of the AKT inhibitor, GSK has decided at this time to suspend further development of GSK2110183 as monotherapy.) Collapse << | November 2011 | Australia, Victoria ... more >> GSK Investigational Site Melbourne, Victoria, Australia, 3004 Collapse << |
联系我们
官方电话:400-920-2911
二维码
微信公众号 CSN官网