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CAS No.: 210354-22-6
GW274150 is an arginine-competitive, NADPH-dependent iNOS inhibitor that has been identified from a series of acetamide amino acids that have a high selectivity for iNOS vs both eNOS (> 260-fold) and nNOS (> 219-fold) and high bioavailability (> 90%) after oral administration.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT00379990 | Arthritis, Rheumatoid | Phase 2 | Completed | - | Serbia ... more >> GSK Investigational Site Belgrade, Serbia, 11000 United Kingdom GSK Investigational Site London, United Kingdom, W6 8LH Collapse << |
NCT00273013 | Asthma | Phase 1 | Completed | - | United Kingdom ... more >> GSK Investigational Site Manchester, Lancashire, United Kingdom, M23 9LT GSK Investigational Site London, United Kingdom, SE1 9RT Collapse << |
NCT00370435 | Arthritis, Rheumatoid | Phase 2 | Completed | - | United Kingdom ... more >> GSK Investigational Site London, United Kingdom, W6 8LH Collapse << |
实验方案
技术信息
CAS号 | 210354-22-6 | 储存条件 |
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分子式 | C8H17N3O2S | 运输 | 蓝冰 | |
分子量 | 219.30 | 别名 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT00379990 | Arthritis, Rheumatoid | Phase 2 | Completed | - | Serbia ... more >> GSK Investigational Site Belgrade, Serbia, 11000 United Kingdom GSK Investigational Site London, United Kingdom, W6 8LH Collapse << |
NCT00273013 | Asthma | Phase 1 | Completed | - | United Kingdom ... more >> GSK Investigational Site Manchester, Lancashire, United Kingdom, M23 9LT GSK Investigational Site London, United Kingdom, SE1 9RT Collapse << |
NCT00370435 | Arthritis, Rheumatoid | Phase 2 | Completed | - | United Kingdom ... more >> GSK Investigational Site London, United Kingdom, W6 8LH Collapse << |
NCT00242866 | Migraine Disorders | Phase 2 | Completed | - | - |
NCT00319137 | Migraine Disorders ... more >> Migraine Collapse << | Phase 2 | Completed | - | Australia, South Australia ... more >> GSK Investigational Site Adelaide, South Australia, Australia, 5000 New Zealand GSK Investigational Site Auckland, New Zealand, 1311 GSK Investigational Site Christchurch, New Zealand, 8001 GSK Investigational Site Hamilton, New Zealand, 2001 GSK Investigational Site Wellington, New Zealand, 6035 Collapse << |
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