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CAS No.: 130308-48-4
Synonyms: HOE 140;Firazyr;艾替班特
Icatibant is a selective and specific antagonist of bradykinin B2 receptor with IC50 and Ki of 1.07 nM and 0.798 nM respectively.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT02584959 | Hereditary Angioedema (HAE) | Phase 3 | Completed | - | - |
NCT02584959 | - | - | Completed | - | - |
NCT02826356 | - | - | Completed | - | France ... more >> Hospices Civils de Lyon, Département d'Anesthésie-Réanimation, Hôpital Edouard Herriot, Lyon, France. Lyon, France, 69003 Collapse << |
实验方案
技术信息
CAS号 | 130308-48-4 | 储存条件 |
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分子式 | C59H89N19O13S | 运输 | 蓝冰 | |
分子量 | 1304.52 | 别名 | HOE 140;Firazyr;艾替班特 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT02584959 | Hereditary Angioedema (HAE) | Phase 3 | Completed | - | - |
NCT02584959 | - | - | Completed | - | - |
NCT02826356 | - | - | Completed | - | France ... more >> Hospices Civils de Lyon, Département d'Anesthésie-Réanimation, Hôpital Edouard Herriot, Lyon, France. Lyon, France, 69003 Collapse << |
NCT03005184 | Heart Failure NYHA Class I ... more >> Heart Failure NYHA Class II Heart Failure NYHA Class III Collapse << | Phase 2 | Withdrawn(Study is being redes... more >>igned and submitted as a new study.) Collapse << | January 2020 | United States, Tennessee ... more >> Vanderbilt University Medical Center Nashville, Tennessee, United States, 37232 Collapse << |
NCT00965393 | Ischaemic Heart Diseases | Not Applicable | Completed | - | United Kingdom ... more >> University of Edinburgh, 49 Little France Crescent Edinburgh, United Kingdom, EH16 4SB Collapse << |
NCT00965120 | Ischaemic Heart Diseases | Not Applicable | Completed | - | United Kingdom ... more >> University of Edinburgh, 49 Little France Crescent Edinburgh, United Kingdom, EH16 4SB Collapse << |
NCT00223704 | Cardiopulmonary Bypass ... more >> Inflammation Fibrinolysis Surgery Collapse << | Phase 2 Phase 3 | Completed | - | United States, Tennessee ... more >> TN Valley Healthcare System Nashville, Tennessee, United States, 37212 Vanderbilt University Nashville, Tennessee, United States, 37232 Collapse << |
NCT00223704 | - | - | Completed | - | - |
NCT01574248 | ACE Inhibitor-associated Angio... more >>edema Collapse << | Phase 4 | Terminated(DSMC recommended di... more >>scontinuation for futility and feasibility) Collapse << | - | United States, California ... more >> University of California, San Diego San Diego, California, United States, 92093 United States, Tennessee Vanderbilt University Medical Center Nashville, Tennessee, United States, 37235 Collapse << |
NCT01154361 | Angioedema | Phase 2 | Completed | - | Germany ... more >> Klinikum rechts der Isar Hals-Nasen-Ohrenklinik der TUM Munich, Bavaria, Germany, 81675 Collapse << |
NCT01574248 | - | - | Terminated(DSMC recommended di... more >>scontinuation for futility and feasibility) Collapse << | - | - |
NCT00517582 | Angioneurotic Edema | Phase 1 | Terminated(This study was stop... more >>ped to allow initiation of a mult-center study) Collapse << | - | United States, Tennessee ... more >> Vanderbilt University Medical Center Nashville, Tennessee, United States, 37205 Collapse << |
NCT01034969 | - | - | Recruiting | May 24, 2023 | - |
NCT03177798 | Hemodialysis-Induced Symptom ... more >> Mitochondrial Diseases Collapse << | Phase 2 | Active, not recruiting | December 31, 2018 | United States, Tennessee ... more >> Vanderbilt University Medical Center Nashville, Tennessee, United States, 37232 Collapse << |
NCT00500656 | Hereditary Angioedema | Phase 3 | Completed | - | Italy ... more >> Università degli Studi di Milano, Dipartimento di Medicina Interna Milano, Italy, 20123 Collapse << |
NCT00097695 | Angioedema | Phase 3 | Completed | - | United States, District of Col... more >>umbia Georgetown University Hospital, Lombardi Cancer Center Washington, District of Columbia, United States, 20007-2197 Collapse << |
NCT00303056 | Joint Disease | Phase 2 | Completed | - | United States, New Jersey ... more >> Administrative Office Bridgewater, New Jersey, United States, 08807 Austria Administrative Office Vienna, Austria, DCA 1220 Czech Republic Administrative Office Praha, Czech Republic, 160 00 Germany Administrative Office Berlin, Germany, D-10785 Poland Administrative Office Warszawa, Poland, 02-672 Collapse << |
NCT01457430 | Hereditary Angioedema | Phase 4 | Completed | - | United States, California ... more >> San Diego Veterans Affairs Medical Center La Jolla, California, United States UCLA - David Geffen School of Medicine Los Angeles, California, United States United States, Maryland Institute for Allergy and Asthma Wheaton, Maryland, United States, 20902 United States, Pennsylvania Penn State University Hershey, Pennsylvania, United States, 17033 United States, Texas AARA Research Center Dallas, Texas, United States, 75231 Collapse << |
NCT00912093 | Hereditary Angioedema | Phase 3 | Completed | - | - |
NCT00097695 | - | - | Completed | - | - |
NCT01457430 | - | - | Completed | - | - |
NCT01919801 | Angiotensin Converting Enzyme ... more >>Inhibitor Induced Angioedema Collapse << | Phase 3 | Completed | - | - |
NCT00500656 | - | - | Completed | - | - |
NCT01919801 | - | - | Completed | - | - |
NCT00997204 | Hereditary Angioedema | Phase 3 | Completed | - | Argentina ... more >> Hospital Britanico Unidad de Alergia Buenos Aires, Argentina, C1035AAT Austria Universitätsklinik für Dermatologie und Venerologie Graz, Austria, 8036 Denmark Odense Universitetshospital-OUH Odense, I og Alergicentret, Denmark France Centre Hospitalier Universitaire/ Service de Dermatologie Angers, Angers Cedex 09, France, 49933 Hospital Edouaed Herriot Lyon, Cedex 03, France, 69437 Clinique Universitaire de Medicine/ Centre National de reference Grenoble, Grenoble Cedex 09, France, 38043 Hopital Claude Huriex/ Service de medicine interne Lille, Lille Cedex, France, 59037 Hopital Europeen Georges Pompidou Immunologie Clinique Paris, Paris Cedex 15, France, 75015 Germany Universitätsmedizin Berlin, Klinik für Dermatologie, Venerologie und Allergologie, Charité Berlin, Germany, 10117 Universitäts-Hals-Nasen-Ohren-Klinik Essen, Universität Duisburg-Essen Essen, Germany, 45127 Klinkum der Johann Wolfgang Goethe-Universitat Frankfurt am Main, Germany, 60590 Hautklinik und Poliklinik, Universitätsmedizin der Johannes Gutenberg-Universität Mainz, Germany, 55101 Israel Bnai-Zion M.C. Clinical Immunology and Allergy Division Haifa, Israel, 31048 Tel Aviv Sourasky Medical Center - Allergy Unit Tel Aviv, Israel, 64239 The Chaim Sheba Medical Center, The Allergy and Clinical Immunology Unit Tel Hashomer, Israel, 52621 Italy Ospedale Luigi Sacco Milano, Italy, 20157 Universita degli Studi di Napoli 'Federico II' Napoli,, Italy, 80131 Spain Hospital Universitario Vall de Hebrón / Sección de Alergia, Escola Infermeria Barcelona, Spain, 08035 Hospital General Universitario Gregorio Maranon Madrid, Spain, 28007 Hospital Universitario La Paz, Servicio de Alergia Madrid, Spain, 28046 Hospital Universitario La Fe, Servicio de Alergia Valencia, Spain, 46009 Switzerland Luzerner Kantonsspital Luzern, Switzerland Universitätsspital Zürich / Dermatologische Klinik Zurich, Switzerland, 8091 United Kingdom Southmead Hospital, Department of Immunology Bristol, United Kingdom, BS10 5NB Barts & The London NHS Trust, Pathology and Pharmacy Building London, United Kingdom, E1 2ES Derriford Combined Laboratory, Department of Clinical Immunology & Allergy Plymouth, United Kingdom, PL6 8DH Collapse << |
NCT00997204 | - | - | Completed | - | - |
NCT02045264 | Hereditary Angioedema (HAE) | Phase 1 | Completed | - | United States, California ... more >> PAREXEL Glendale, California, United States, 91206 Collapse << |
NCT02045264 | - | - | Completed | - | - |
NCT00912093 | - | - | Completed | - | - |
NCT01386658 | Hereditary Angioedema (HAE) | Phase 3 | Completed | - | - |
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