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CAS No.: 314245-33-5
IU1 is a cell-permeable, reversible and selective proteasome inhibitor of human USP14 with IC50 of 4.7 μ M, 25-fold selective to IsoT.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT01578473 | Peyronie's Disease | Phase 1 | Completed | - | United States, Massachusetts ... more >> Men's Health Boston Chestnut Hill, Massachusetts, United States, 02467 Collapse << |
NCT01354704 | Deep Vein Thrombosis ... more >> Venous Thrombosis Adverse Effect of Anticoagulants Collapse << | Phase 4 | Completed | - | Tunisia ... more >> Hospital Charle Nicolle Tunis, Tunis BAB SOUIKA, Tunisia, 1006 Collapse << |
NCT01774812 | Cardiovascular Disease ... more >> Sudden Cardiac Death Collapse << | Phase 2 | Completed | - | Canada, Alberta ... more >> Northland Hemodialysis Clinic Calgary, Alberta, Canada, T2L 2J8 Foothills Medical Centre - University of Calgary Calgary, Alberta, Canada, T2N 2T9 Sheldon M. Chumir Health Centre Calgary, Alberta, Canada, T2R 0X7 Collapse << |
实验方案
技术信息
CAS号 | 314245-33-5 | 储存条件 |
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分子式 | C18H21FN2O | 运输 | 蓝冰 | |
分子量 | 300.37 | 别名 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT01578473 | Peyronie's Disease | Phase 1 | Completed | - | United States, Massachusetts ... more >> Men's Health Boston Chestnut Hill, Massachusetts, United States, 02467 Collapse << |
NCT01354704 | Deep Vein Thrombosis ... more >> Venous Thrombosis Adverse Effect of Anticoagulants Collapse << | Phase 4 | Completed | - | Tunisia ... more >> Hospital Charle Nicolle Tunis, Tunis BAB SOUIKA, Tunisia, 1006 Collapse << |
NCT01774812 | Cardiovascular Disease ... more >> Sudden Cardiac Death Collapse << | Phase 2 | Completed | - | Canada, Alberta ... more >> Northland Hemodialysis Clinic Calgary, Alberta, Canada, T2L 2J8 Foothills Medical Centre - University of Calgary Calgary, Alberta, Canada, T2N 2T9 Sheldon M. Chumir Health Centre Calgary, Alberta, Canada, T2R 0X7 Collapse << |
NCT01806792 | Postmenopausal Women Osteoporo... more >>sis Collapse << | Phase 3 | Completed | - | Korea, Republic of ... more >> Chung-ang university hospital Seoul, Korea, Republic of, 156-755 Collapse << |
NCT02417207 | Hepatitis B L... more >>iver Transplantation Collapse << | Phase 4 | Unknown | April 2018 | China, Guangdong ... more >> Wang Guoying Guangzhou, Guangdong, China, 510630 Collapse << |
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