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CAS No.: 217094-32-1
Synonyms: K-604 HCl;K-604 Hydrochloride;K-604
K-604 is a potent and selective acyl-CoA:cholesterol acyltransferase 1 (ACAT-1) inhibitor. K-604 inhibits against acyl-coenzyme A (acyl-CoA):cholesterol O-acyltransferase-1 (ACAT1, SOAT1) activitiy in a selective (IC50 = 450 nM vs. 102.85 μ M against human ACAT1 and ACAT2, respectively) and acyl-CoA-competitive (Ki = 378 nM against oleoyl-coA) manner.
生物活性
实验方案
技术信息
CAS号 | 217094-32-1 | 储存条件 |
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分子式 | C23H32Cl2N6OS3 | 运输 | 蓝冰 | |
分子量 | 575.64 | 别名 | K-604 HCl;K-604 Hydrochloride;K-604 |
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