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CAS No.: 1058137-23-7
Synonyms: E-3810;AL-3810;德立替尼
E-3810 is a dual inhibitor of the VEGF and FGF receptors, potently and selectively inhibits VEGFR1, VEGFR2, VEGFR3, FGFR1 and FGFR2 with IC50 of 7 nM, 25 nM, 10 nM, 17.5 nM, and 82.5 nM, respectively.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT00838526 | Gastroesophageal Reflux Diseas... more >>e (GERD) Collapse << | Phase 3 | Completed | - | United States, Illinois ... more >> Ltd. Moline, Illinois, United States, 61265 Midwest Clinical Moline, Illinois, United States, 61265 Research Associates Moline, Illinois, United States, 61265 Moline, Illinois, United States, 61265 Collapse << |
NCT00132496 | - | - | Completed | - | - |
NCT00165841 | Gastroesophageal Reflux Diseas... more >>e Collapse << | Phase 2 | Completed | - | United States, California ... more >> Quality Care Medical Center Inc. Vista, California, United States, 92085 Collapse << |
实验方案
技术信息
CAS号 | 1058137-23-7 | 储存条件 |
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分子式 | C26H25N3O4 | 运输 | 蓝冰 | |||
分子量 | 443.49 | 别名 | E-3810;AL-3810;德立替尼 | |||
溶解度 |
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动物实验配方 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT00838526 | Gastroesophageal Reflux Diseas... more >>e (GERD) Collapse << | Phase 3 | Completed | - | United States, Illinois ... more >> Ltd. Moline, Illinois, United States, 61265 Midwest Clinical Moline, Illinois, United States, 61265 Research Associates Moline, Illinois, United States, 61265 Moline, Illinois, United States, 61265 Collapse << |
NCT00132496 | - | - | Completed | - | - |
NCT00165841 | Gastroesophageal Reflux Diseas... more >>e Collapse << | Phase 2 | Completed | - | United States, California ... more >> Quality Care Medical Center Inc. Vista, California, United States, 92085 Collapse << |
NCT00165841 | - | - | Completed | - | - |
NCT00658528 | - | - | Completed | - | - |
NCT00658632 | - | - | Completed | - | - |
NCT00132496 | Gastroesophageal Reflux Diseas... more >>e Collapse << | Phase 2 | Completed | - | - |
NCT00658632 | Gastroesophageal Reflux Diseas... more >>e (GERD) Collapse << | Phase 3 | Completed | - | - |
NCT00658775 | Gastroesophageal Reflux Diseas... more >>e (GERD) Collapse << | Phase 3 | Completed | - | - |
NCT00658775 | - | - | Completed | - | - |
NCT00658528 | Gastroesophageal Reflux Diseas... more >>e (GERD) Collapse << | Phase 3 | Completed | - | - |
NCT00839306 | Gastroesophageal Reflux Diseas... more >>e (GERD) Collapse << | Phase 3 | Completed | - | United States, Illinois ... more >> Associates, Ltd. Moline, Illinois, United States, 61265 Midwest Clinical Moline, Illinois, United States, 61265 Research Moline, Illinois, United States, 61265 Moline, Illinois, United States, 61265 Collapse << |
NCT00839306 | - | - | Completed | - | - |
NCT00911534 | Symptomatic Gastroesophageal R... more >>eflux Disease (sGERD) Collapse << | Phase 3 | Completed | - | - |
NCT01286194 | - | - | Completed | - | - |
NCT02109016 | Non-Small Cell Lung Cancer ... more >> Squamous Non-Small Cell Lung Cancer NSCLC Small Cell Lung Cancer SCLC Lung Cancer Advanced Lung Cancer Metastatic Lung Cancer Stage IV Lung Cancer Collapse << | Phase 2 | Terminated | - | United States, California ... more >> University of California, Los Angeles Los Angeles, California, United States, 90095 United States, Colorado University of Colorado Aurora, Colorado, United States, 80045 United States, District of Columbia Georgetown University Washington, District of Columbia, United States, 20007 United States, Georgia Emory University Atlanta, Georgia, United States, 30322 United States, Maryland Associates in Oncology and Hematology Rockville, Maryland, United States, 20850 United States, Pennsylvania University of Pittsburgh Medical Center Pittsburgh, Pennsylvania, United States, 15232 United States, Tennessee Tennessee Oncology Nashville, Tennessee, United States, 37203 France CHU Caen, Hôpital de la Côte de Nacre Caen, France, 14033 CHRU Lille, Hôpital Albert Calmette Lille, France, 59037 Hôpital Nord Marseille, France, 13915 Institut Gustave-Roussy Villejuif, France, 94805 Germany Universität Duisburg-Essen Essen, Germany, 45147 Hospital Grosshansdorf Grosshansdorf, Germany, 22927 Pius Hospital Oldenburg Oldenburg, Germany, 26121 Italy Ospedale San Raffaele Milano, Italy, 20132 Fondazione IRCCS Istituto Nazionale Tumori Milano, Italy, 20133 AOU San Luigi Gonzaga Orbassano, Italy, 10043 Ospedale S. Maria della Misericordia Perugia, Italy, 06156 Spain Hospital Universitari Vall d'Hebrón Barcelona, Cataluña, Spain, 8035 Collapse << |
NCT01153659 | Healthy | Phase 1 | Completed | - | United States, Oklahoma ... more >> Oklahoma Foundation for Digestive Research Oklahoma City, Oklahoma, United States, 73104 Collapse << |
NCT00236184 | Heartburn | Phase 3 | Completed | - | United States, California ... more >> Jeffrey L. Newman Vista, California, United States, 92084 Collapse << |
NCT00236197 | Heartburn | Phase 3 | Completed | - | United States, New York ... more >> New York Center For Clinical Research Lake Success, New York, United States, 11042 Collapse << |
NCT00911534 | - | - | Completed | - | - |
NCT00838526 | - | - | Completed | - | - |
NCT01085708 | Healthy | Phase 1 | Completed | - | - |
NCT00236184 | - | - | Completed | - | - |
NCT01085695 | Healthy | Phase 1 | Completed | - | - |
NCT01202071 | Healthy | Phase 2 | Completed | - | Japan ... more >> Toshima-ku, Tokyo, Japan Collapse << |
NCT00236197 | - | - | Completed | - | - |
NCT01089543 | Functional Dyspepsia | Phase 2 | Completed | - | Japan ... more >> Nagoya, Aichi, Japan Chikushino, Fukuoka, Japan Kitakyushu, Fukuoka, Japan Maebashi, Gunma, Japan Sapporo, Hokkaido, Japan Kobe, Hyogo, Japan Nishinomiya, Hyogo, Japan Tsuchiura, Ibaraki, Japan Takamatsu, Kagawa, Japan Yokohama, Kanagawa, Japan Sendai, Miyagi, Japan Yufu, Oita, Japan Nakagami, Okinawa, Japan Hirakata, Osaka, Japan Moriguchi, Osaka, Japan Suita, Osaka, Japan Takatsuki, Osaka, Japan Karatsu, Saga, Japan Kusatsu, Shiga, Japan Izumo, Shimane, Japan Fujieda, Shizuoka, Japan Hamamatsu, Shizuoka, Japan Otawara, Tochigi, Japan Shimotsuga, Tochigi, Japan Bunkyo, Tokyo, Japan Mitaka, Tokyo, Japan Nakano, Tokyo, Japan Ota, Tokyo, Japan Setagaya, Tokyo, Japan Shibuya, Tokyo, Japan Shinagawa, Tokyo, Japan Akita, Japan Fukuoka, Japan Gifu, Japan Hiroshima, Japan Kagoshima, Japan Kochi, Japan Kumamoto, Japan Kyoto, Japan Miyazaki, Japan Oita, Japan Osaka, Japan Saga, Japan Saitama, Japan Shizuoka, Japan Yamagata, Japan Collapse << |
NCT00165672 | Non-erosive Gastroesophageal R... more >>eflux Disease Collapse << | Phase 3 | Completed | - | Japan ... more >> Nagoya, Aichi-Prefecture, Japan, 467-0001 Fukuoka, Fukuoka-Prefecture, Japan, 810-0001 Fukuoka, Fukuoka-Prefecture, Japan, 811-0213 Yukuhashi, Fukuoka-Prefecture, Japan, 824-0026 Hiroshima, Hiroshima-Prefecture, Japan, 734-0037 Osaka, Osaka-Prefecture, Japan, 530-0012 Osaka, Osaka-Prefecture, Japan, 545-0051 Saga, Saga-Prefecture, Japan, 849-0937 Otsu, Shiga-Prefecture, Japan, 520-2121 Izumo, Shimane-Prefecture, Japan, 693-0021 Bunkyo-ku, Tokyo, Japan, 113-0022 Shinjuku-ku, Tokyo, Japan, 162-0052 Ube, Yamaguchi-Prefecture, Japan, 755-0046 Collapse << |
NCT01202071 | - | - | Completed | - | - |
NCT01089543 | - | - | Completed | - | - |
NCT02135107 | Gastroesophageal Reflux Diseas... more >>e Collapse << | Phase 3 | Completed | - | - |
NCT02747797 | Advanced Cancer | Phase 2 | Withdrawn(Drug Supply No Longe... more >>r Available) Collapse << | April 2022 | United States, California ... more >> UC San Diego Moores Cancer Center La Jolla, California, United States, 92093 Collapse << |
NCT02135107 | - | - | Completed | - | - |
NCT00770913 | - | - | Completed | - | - |
NCT00165646 | Non-erosive Gastroesophageal R... more >>eflux Disease Collapse << | Phase 3 | Completed | - | Japan ... more >> Aichi-Gun, Aichi-Prefecture, Japan, 480-1103 Nagoya, Aichi-Prefecture, Japan, 466-0065 Nagoya, Aichi-Prefecture, Japan, 467-0001 Chikushino, Fukuoka-Prefecture, Japan, 818-0024 Chikushino, Fukuoka-Prefecture, Japan, 818-0067 Fukuoka, Fukuoka-Prefecture, Japan, 813-0003 Kita-kyushu, Fukuoka-Prefecture, Japan, 807-1262 Maebashi, Gunma-Prefecture, Japan, 371-0034 Hiroshima, Hiroshima-Prefecture, Japan, 730-0052 Hiroshima, Hiroshima-Prefecture, Japan, 734-0037 Sapporo, Hokkaido-Prefecture, Japan, 003-0021 Sapporo, Hokkaido-Prefecture, Japan, 060-0061 Sapporo, Hokkaido-Prefecture, Japan, 060-0814 Kochi, Kochi-Prefecture, Japan, 780-0901 Kyoto, Kyoto-Prefecture, Japan, 602-0000 Kyoto, Kyoto-Prefecture, Japan, 606-8397 Sandai, Miyagi-Prefecture, Japan, 980-0872 Sendai, Miyagi-Prefecture, Japan, 984-0075 Moriguchi, Osaka-Prefecture, Japan, 570-0021 Osaka, Osaka-Prefecture, Japan, 530-0012 Osaka, Osaka-Prefecture, Japan, 536-0002 Osaka, Osaka-Prefecture, Japan, 545-0051 Saga, Saga-Prefecture, Japan, 849-0937 Kawaguchi, Saitama-Prefecture, Japan, 332-0021 Izumo, Shimane-Prefecture, Japan, 693-0021 Matsue, Shimane-Prefecture, Japan, 690-0886 Hamamatsu, Shizuoka-Prefecture, Japan, 431-3125 Shinagawa-ku, Tokyo, Japan, 140-0011 Shinjuku-ku, Tokyo, Japan, 162-0052 Sanyoonoda, Yamaguchi-Prefecture, Japan, 756-0076 Sanyoonoda, Yamaguchi-Prefecture, Japan, 757-0002 Ube, Yamaguchi-Prefecture, Japan, 755-0004 Ube, Yamaguchi-Prefecture, Japan, 755-0046 Ube, Yamaguchi-Prefecture, Japan, 755-0067 Ube, Yamaguchi-Prefecture, Japan, 755-0077 Collapse << |
NCT00165672 | - | - | Completed | - | - |
NCT01283945 | Solid Tumors | Phase 1 Phase 2 | Completed | - | France ... more >> Institute Gustave Roussy Villejuif, Paris, France, 94805 Hopital Louis Pradel Lyon, France, 69677 Italy European Institute of Oncology Milano, Italy, 20141 Spain Vall d' Hebron University Hospital Barcellona, Spain Collapse << |
NCT01398410 | Gastric Ulcers Duodenal Ulcers... more >> Caused by Low-dose Aspirin Collapse << | Phase 2 Phase 3 | Completed | - | - |
NCT00770913 | Refractory Reflux Esophagitis | Phase 2 Phase 3 | Completed | - | - |
NCT01397448 | Gastric or Duodenal Ulcers Cau... more >>sed by Low-dose Aspirin Collapse << | Phase 2 Phase 3 | Completed | - | - |
NCT01398410 | - | - | Completed | - | - |
NCT01397448 | - | - | Completed | - | - |
NCT00165646 | - | - | Completed | - | - |
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