CAS No.: 176977-56-3
LY320135 Catalog No. CSN19472
Synonyms: Ly320135
LY-320135 is a potent and selective Canniboid CB1 receptor antagonist/inverse agonist. LY-320135 is selective (~70 fold) over Canniboid CB2 receptors. This compound shows weak binding to both 5-HT2 (Ki = 6.4 μM) and muscarinic receptors (Ki = 2.1 μM).
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纯度 & 质量文件
批次:
靶点选择性
生物活性
- 描述
- 参考文献
- [1] Pertwee RG. Inverse agonism and neutral antagonism at cannabinoid CB1 receptors. Life Sci. 2005 Feb 4;76(12):1307-24.
- [2] Holland M, John Challiss RA, et al. Cannabinoid CB1 receptors fail to cause relaxation, but couple via Gi/Go to the inhibition of adenylyl cyclase in carotid artery smooth muscle. Br J Pharmacol. 1999 Oct;128(3):597-604.
实验方案
- 计算器
- 储存液制备
技术信息
| CAS号 | 176977-56-3 | 储存条件 |
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| 分子式 | C24H17NO4 | 运输 | 蓝冰 | |
| 分子量 | 383.40 | 别名 | Ly320135 |
