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CAS No.: 1379545-95-5
Synonyms: MSC2363318A;HTI-286 HCl;SPA 110 HCl
MSC2363318A, also known as M2698, is an orally available inhibitor of the serine/threonine protein kinases ribosomal protein S6 Kinase (p70S6K) and Akt (protein kinase B), with potential antineoplastic activity.
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生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT01971515 | Solid Tumor | Phase 1 | Completed | - | United States, Alabama ... more >> University of Alabama at Birmingham Birmingham, Alabama, United States, 35294 United States, California Cedars Sinai Medical Center Los Angeles, California, United States, 90048 University of California at San Diego, Moores Cancer Center San Diego, California, United States, 92093 United States, Florida Sylvester Comprehensive Cancer Center Miami, Florida, United States, 33136 United States, Louisiana Metairie Oncology Metairie, Louisiana, United States, 70006 United States, Massachusetts Massachusetts General Hospital Boston, Massachusetts, United States, 02114 United States, Michigan Karmanos Cancer Institute Detroit, Michigan, United States, 48201 Henry Ford Hospital Detroit, Michigan, United States, 48202 United States, Missouri Washington University School of Medicine Saint Louis, Missouri, United States, 63110 United States, New York Mount Sinai New York, New York, United States, 10029 United States, South Carolina Medical University of South Carolina Charleston, South Carolina, United States, 29425 United States, Texas Mary Crowley Cancer Research Center Dallas, Texas, United States, 75251 MD Anderson Cancer Center Houston, Texas, United States, 77030 University of Texas Health Science Center at San Antonio San Antonio, Texas, United States, 78229 United States, Vermont Fletcher Allen Health Care, Inc. Burlington, Vermont, United States, 05401 Collapse << |
实验方案
技术信息
CAS号 | 1379545-95-5 | 储存条件 |
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分子式 | C21H19ClF3N5O | 运输 | 蓝冰 | |
分子量 | 449.86 | 别名 | MSC2363318A;HTI-286 HCl;SPA 110 HCl |