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CAS No.: 76541-72-5
Synonyms: SR-202
SR 202 is a selective PPARγ antagonist which attenuates troglitazone-induced PPARγ transcriptional activity with IC50 value of 140μM. It inhibits PPARγ-dependent adipocyte differentiation and growth in vitro and in vivo and improves insulin sensitivity in diabetic ob/ob mice and increases HDL levels in rats in vivo.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT01309542 | Major Depressive Disorder | Phase 3 | Completed | - | - |
NCT01414920 | Diabetes Mellitus, Type 2 | Phase 2 | Completed | - | - |
NCT00201981 | Keratoconjunctivitis Sicca | Phase 3 | Completed | - | - |
实验方案
技术信息
CAS号 | 76541-72-5 | 储存条件 |
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分子式 | C11H17ClO7P2 | 运输 | 蓝冰 | |||
分子量 | 358.65 | 别名 | SR-202 | |||
溶解度 |
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动物实验配方 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT01309542 | Major Depressive Disorder | Phase 3 | Completed | - | - |
NCT01414920 | Diabetes Mellitus, Type 2 | Phase 2 | Completed | - | - |
NCT00201981 | Keratoconjunctivitis Sicca | Phase 3 | Completed | - | - |
NCT00848107 | Systemic Sclerosis | Phase 2 | Terminated(The TDE-DU-202 exte... more >>nsion study was discontinued after the randomized, placebo-controlled TDE-DU-201 study did not meet its primary efficacy objective.) Collapse << | - | - |
NCT02909725 | Sedentary Lifestyle ... more >> Diabetes Mellitus, Gestational Collapse << | Not Applicable | Unknown | December 2016 | United States, Iowa ... more >> Iowa State University Recruiting Ames, Iowa, United States, 50011 Contact: Caroline McKinney, BS 515-202-5569 clmck@iastate.edu Contact: Christina Campbell, PhD 515-294-4260 ccampbel@iastate.edu Principal Investigator: Christina Campbell, PhD Collapse << |
NCT01104870 | Pulmonary Hypertension | Phase 2 | Completed | - | United States, Arizona ... more >> St. Joseph's Hospital and Medical Center Phoenix, Arizona, United States, 85013 University of Arizona Tucson, Arizona, United States, 87524 United States, California University of California Los Angeles Pulmonary Division Los Angeles, California, United States, 90095 University of California Davis Medical Center Sacramento, California, United States, 95817 United States, New York University of Rochester Medical Center, Mary Parkes Center Rochester, New York, United States, 14623 United States, Ohio The Carl and Edyth Lindner Research Center at The Christ Hospital Cincinnati, Ohio, United States, 45219 University of Cincinnati Cincinnati, Ohio, United States, 45267 The Ohio State University Medical Center Columbus, Ohio, United States, 43221 United States, Pennsylvania University of Pittsburgh Medical Center Pittsburgh, Pennsylvania, United States, 15213 Collapse << |
NCT02160730 | Cushings Disease | Phase 2 | Terminated(NIH grant ended.) | - | United States, California ... more >> Cedars-Sinai Medical Center Los Angeles, California, United States, 90048 Collapse << |
NCT00848107 | - | - | Terminated(The TDE-DU-202 exte... more >>nsion study was discontinued after the randomized, placebo-controlled TDE-DU-201 study did not meet its primary efficacy objective.) Collapse << | - | - |
NCT00151398 | Alzheimer Disease | Phase 2 | Completed | - | - |
NCT01546649 | Premenopausal Breast Cancer | Phase 3 | Completed | - | Japan ... more >> Nagoya-shi, Aichi, Japan Fukushima-shi, Fukushima, Japan Maebashi-shi, Gunma, Japan Ohta-shi, Gunma, Japan Sapporo-shi, Hokkaido, Japan Isehara-shi, Kanagawa, Japan Yokohama-shi, Kanagawa, Japan Kumamoto-shi, Kumamoto, Japan Kyoto-shi, Kyoto, Japan Nigata-shi, Nigata, Japan Kurashiki-shi, Okayama, Japan Osaka-shi, Osaka, Japan Suita-shi, Osaka, Japan Kita-adachi-gun, Saitama, Japan Shinjuku-ku, Tokyo, Japan Collapse << |
NCT01546649 | - | - | Completed | - | - |
NCT00654927 | Multiple Sclerosis | Phase 3 | Completed | - | - |
NCT00053417 | - | - | Completed | - | - |
NCT00709371 | Obesity | Phase 2 | Completed | - | - |
NCT01027949 | Pulmonary Arterial Hypertensio... more >>n Collapse << | Phase 3 | Active, not recruiting | December 2020 | - |
NCT01104870 | - | - | Completed | - | - |
NCT01235221 | Multiple Sclerosis | Phase 3 | Completed | - | Canada, Alberta ... more >> Foothills Medical Center Calgary, Alberta, Canada Canada, British Columbia University of British Columbia Vancouver, British Columbia, Canada Canada, New Brunswick River Valley Health Fredericton, New Brunswick, Canada Canada, Nova Scotia QEII Health Sciences Centre Halifax, Nova Scotia, Canada Canada, Ontario Ottawa Hospital General Campus Ottawa, Ontario, Canada Collapse << |
NCT00654927 | - | - | Completed | - | - |
NCT02393612 | Peripheral Arterial Disease | Phase 3 | Completed | - | - |
NCT00053417 | Multiple Sclerosis | Phase 2 | Completed | - | - |
NCT00526136 | Atrial Fibrillation | Phase 2 | Completed | - | - |
NCT02547428 | Attention-Deficit Hyperactivit... more >>y Disorder Collapse << | Phase 2 | Completed | - | United States, California ... more >> Newport Beach, California, United States United States, Florida Bradenton, Florida, United States Maitland, Florida, United States United States, Nevada Las Vegas, Nevada, United States United States, North Carolina Durham, North Carolina, United States Collapse << |
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