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CAS No.: 1445993-26-9
Synonyms: ABBV-075;米维布塞
Mivebresib, also known as ABBV-075, is an inhibitor of bormodomain and extra terminal domain (BET). The Ki values of BRD2, BRD4, BRDT are 1 nM - 2.2 nM.
规格 | 价格 | 促销价格 | 库存 | 数量 |
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生物活性
靶点 | Bromodomain 3 Ki:12.2nM | Bromodomain 2 Ki:1-2.2nM | Bromodomain 4 Ki:1-2.2nM | Bromodomain testis-specific Protein Ki:1-2.2nM | Bromodomain CREBBP Kd:87μM | 更多 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT02391480 | Cancer Breast... more >> Cancer Non-Small Cell Lung Cancer Acute Myeloid Leukemia (AML) Multiple Myeloma Prostate Cancer Small Cell Lung Cancer Non-Hodgkins Lymphoma Collapse << | Phase 1 | Recruiting | October 22, 2019 | United States, Arizona ... more >> Scottsdale Healthcare /ID# 132963 Recruiting Scottsdale, Arizona, United States, 85258-4566 United States, California City of Hope /ID# 154053 Recruiting Duarte, California, United States, 91010 UC Davis Comp Cancer Ctr /ID# 154644 Recruiting Sacramento, California, United States, 95817 United States, Connecticut Yale University /ID# 136982 Recruiting New Haven, Connecticut, United States, 06510 United States, Illinois University of Chicago /ID# 155453 Recruiting Chicago, Illinois, United States, 60637-1443 United States, Indiana Indiana Univ School Medicine /ID# 132946 Active, not recruiting Indianapolis, Indiana, United States, 46202 United States, North Carolina Duke Univ Med Ctr /ID# 154647 Recruiting Durham, North Carolina, United States, 27710 United States, Texas Mary Crowley Cancer Research /ID# 154059 Recruiting Dallas, Texas, United States, 75246 Univ TX, MD Anderson /ID# 132276 Recruiting Houston, Texas, United States, 77030 UT MD Anderson Cancer Center /ID# 164122 Recruiting Houston, Texas, United States, 77030 Collapse << |
实验方案
技术信息
CAS号 | 1445993-26-9 | 储存条件 |
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分子式 | C22H19F2N3O4S | 运输 | 蓝冰 | |||||||
分子量 | 459.47 | 别名 | ABBV-075;米维布塞 | |||||||
溶解度 |
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动物实验配方 |