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CAS No.: 1417329-24-8
Synonyms: HMTase Inhibitor IX
MM-102 is a high-affinity peptidomimetic MLL1 inhibitor with IC50 of 0.4 μM in a cell-free assay.
规格 | 价格 | 促销价格 | 库存 | 数量 |
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生物活性
动物研究 | |
剂量 | Mice: 15 mg/kg[2] (i.p.) |
给药途径 | i.p. |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT00985959 | Multiple Myeloma | Phase 1 | Completed | - | Japan ... more >> Fukuoka, Japan Hiroshima N/A, Japan Hitachi, Japan Isehara, Japan Kamogawa, Japan Kanazawa, Japan Kawagoe, Japan Kobe, Japan Koto-Ku, Japan Kumamoto, Japan Kurashiki, Japan Kurume, Japan Kyoto, Japan Nagasaki, Japan Nagoya, Japan Narita, Japan Niigata, Japan Okayama, Japan Osaka-Sayama, Japan Sapporo, Japan Shibukawa, Japan Suita, Japan Tokushima N/A, Japan Tokyo, Japan Toyama-City, Japan Toyohashi, Japan Utsunomiya, Japan Yokohama, Japan Collapse << |
NCT00985959 | - | - | Completed | - | - |
NCT02426723 | Multiple Myeloma | Phase 1 | Recruiting | - | United States, Texas ... more >> The University of Texas MD Anderson Cancer Center Recruiting Houston, Texas, United States, 77030 Principal Investigator: Elisabet Manasanch, MD Korea, Republic of Seoul National University Hospital Recruiting Seoul, Korea, Republic of Principal Investigator: Sung-Soo Yoon, MD Seoul St.Mary's Hospital Recruiting Seoul, Korea, Republic of Contact: Chang-Ki Min, MD Yonsei Severance Hospital Recruiting Seoul, Korea, Republic of Contact: Jin Seok Kim, MD Collapse << |
实验方案
技术信息
CAS号 | 1417329-24-8 | 储存条件 |
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分子式 | C35H49F2N7O4 | 运输 | 蓝冰 | |
分子量 | 669.80 | 别名 | HMTase Inhibitor IX |