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CAS No.: 2289690-31-7
Synonyms: NUCC-0196361
MYCi361 is a MYC inhibitor with Kd value of 3.2μM. It engages MYC inside cells, disrupts MYC/MAX dimers, and impairs MYC-driven gene expression. MYCi361 suppressed in vivo tumor growth in mice, increased tumor immune cell infiltration, upregulated PD-L1 on tumors, and sensitized tumors to anti-PD1 immunotherapy.
生物活性
实验方案
技术信息
CAS号 | 2289690-31-7 | 储存条件 |
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分子式 | C26H16ClF9N2O2 | 运输 | 蓝冰 | |||||||
分子量 | 594.86 | 别名 | NUCC-0196361 | |||||||
溶解度 |
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动物实验配方 |
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